Quantitative Structure-Activity Relationships of Antibacterial Agents, 7-Heterocyclic Amine Substituted 1-Cyclopropyl-6,8-difluoro-4-oxoquinoline-3-carboxylic Acids.

Tetsuo OKADA; Kiyoshi EZUMI; Masumi YAMAKAWA; Hisao SATO; Teruji TSUJI; Tadahiko TSUSHIMA; Kiyoshi MOTOKAWA; Yoshihide KOMATSU

doi:10.1248/cpb.41.126

Quantitative Structure-Activity Relationships of Antibacterial Agents, 7-Heterocyclic Amine Substituted 1-Cyclopropyl-6,8-difluoro-4-oxoquinoline-3-carboxylic Acids.

Chemical and Pharmaceutical Bulletin ◽

10.1248/cpb.41.126 ◽

1993 ◽

Vol 41 (1) ◽

pp. 126-131 ◽

Cited By ~ 22

Author(s):

Tetsuo OKADA ◽

Kiyoshi EZUMI ◽

Masumi YAMAKAWA ◽

Hisao SATO ◽

Teruji TSUJI ◽

...

Keyword(s):

Carboxylic Acids ◽

Antibacterial Agents ◽

Heterocyclic Amine ◽

Quantitative Structure ◽

Structure Activity Relationships ◽

Structure Activity ◽

Quantitative Structure Activity Relationships ◽

Substituted 1

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ChemInform Abstract: Quantitative Structure-Activity Relationships of Antibacterial Agents, 7-Heterocyclic Amine Substituted 1-Cyclopropyl-6,8-difluoro-4- oxoquinoline-3-carboxylic Acids.

ChemInform ◽

10.1002/chin.199325281 ◽

2010 ◽

Vol 24 (25) ◽

pp. no-no

Author(s):

T. OKADA ◽

K. EZUMI ◽

M. YAMAKAWA ◽

H. SATO ◽

T. TSUJI ◽

...

Keyword(s):

Carboxylic Acids ◽

Antibacterial Agents ◽

Heterocyclic Amine ◽

Quantitative Structure ◽

Structure Activity Relationships ◽

Structure Activity ◽

Quantitative Structure Activity Relationships ◽

Substituted 1

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Novel and Selective 5-HT2C/2BReceptor Antagonists as Potential Anxiolytic Agents: Synthesis, Quantitative Structure−Activity Relationships, and Molecular Modeling of Substituted 1-(3-Pyridylcarbamoyl)indolines

Journal of Medicinal Chemistry ◽

10.1021/jm970741j ◽

1998 ◽

Vol 41 (10) ◽

pp. 1598-1612 ◽

Cited By ~ 47

Author(s):

Steven M. Bromidge ◽

Steven Dabbs ◽

David T. Davies ◽

D. Malcolm Duckworth ◽

Ian T. Forbes ◽

...

Keyword(s):

Molecular Modeling ◽

Quantitative Structure ◽

Structure Activity Relationships ◽

Structure Activity ◽

Quantitative Structure Activity Relationships ◽

Substituted 1

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Quantitative Structure−Activity Relationships among Macrolide Antibacterial Agents: In Vitro and in Vivo Potency againstPasteurella multocida

Journal of Medicinal Chemistry ◽

10.1021/jm960436i ◽

1997 ◽

Vol 40 (9) ◽

pp. 1340-1346 ◽

Cited By ~ 90

Author(s):

James W. McFarland ◽

Cynthia M. Berger ◽

Susan A. Froshauer ◽

Shigeru F. Hayashi ◽

Scott J. Hecker ◽

...

Keyword(s):

Antibacterial Agents ◽

Quantitative Structure ◽

Structure Activity Relationships ◽

Structure Activity ◽

Quantitative Structure Activity Relationships

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Quantitative structure-activity relationships of heterocyclic amine mutagens formed during the cooking of food

Environmental and Molecular Mutagenesis ◽

10.1002/em.2850170103 ◽

1991 ◽

Vol 17 (1) ◽

pp. 4-19 ◽

Cited By ~ 37

Author(s):

F. T. Hatch ◽

M. G. Knize ◽

J. S. Felton ◽

R. W. Morgan

Keyword(s):

Heterocyclic Amine ◽

Quantitative Structure ◽

Structure Activity Relationships ◽

Structure Activity ◽

Quantitative Structure Activity Relationships

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Quantum-mechanically calculated properties for the development of quantitative structure-activity relationships (QSAR'S). pKA-values of phenols and aromatic and aliphatic carboxylic acids

Chemosphere ◽

10.1016/0045-6535(89)90503-1 ◽

1989 ◽

Vol 19 (10-11) ◽

pp. 1595-1609 ◽

Cited By ~ 43

Author(s):

C. Grüber ◽

V. Buß

Keyword(s):

Carboxylic Acids ◽

Quantitative Structure ◽

Pka Values ◽

Structure Activity Relationships ◽

Structure Activity ◽

Quantitative Structure Activity Relationships ◽

Aliphatic Carboxylic Acids

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3D-Quantitative Structure-Activity Relationships for Hydrophobic Interactions: Comparative Molecular Field Analysis (CoMFA) including Molecular Lipophilicity Potentials as Applied to the Glycine Conjugation of Aromatic as well as Aliphatic Carboxylic Acids

Quantitative Structure-Activity Relationships ◽

10.1002/qsar.19960150303 ◽

1996 ◽

Vol 15 (3) ◽

pp. 194-200 ◽

Cited By ~ 4

Author(s):

Takashi Masuda ◽

Katsuhiko Nakamura ◽

Takahiro Jikihara ◽

Fumiyo Kasuya ◽

Kazuo Igarashi ◽

...

Keyword(s):

Carboxylic Acids ◽

Hydrophobic Interactions ◽

Field Analysis ◽

Molecular Field ◽

Comparative Molecular Field Analysis ◽

Quantitative Structure ◽

Structure Activity Relationships ◽

Structure Activity ◽

Quantitative Structure Activity Relationships ◽

Aliphatic Carboxylic Acids

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Mechanistic interpretation of the genotoxicity of nitrofurans (antibacterial agents) using quantitative structure-activity relationships and comparative molecular field analysis

Journal of Medicinal Chemistry ◽

10.1021/jm00060a008 ◽

1993 ◽

Vol 36 (8) ◽

pp. 1007-1016 ◽

Cited By ~ 58

Author(s):

Asim Kumar Debnath ◽

Corwin Hansch ◽

Ki H. Kim ◽

Yvonne C. Martin

Keyword(s):

Antibacterial Agents ◽

Field Analysis ◽

Molecular Field ◽

Comparative Molecular Field Analysis ◽

Quantitative Structure ◽

Structure Activity Relationships ◽

Molecular Field Analysis ◽

Structure Activity ◽

Quantitative Structure Activity Relationships

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Quantitative Structure-Activity Relationships of Potential Antimalarial Drugs Active Against Chloroquine-Resistant Plasmodium Falciparum

Planta Medica ◽

10.1055/s-2008-1075144 ◽

2008 ◽

Vol 74 (03) ◽

Author(s):

SJ Hocart ◽

H Liu ◽

D De ◽

FM Krogstad ◽

DJ Krogstad

Keyword(s):

Plasmodium Falciparum ◽

Antimalarial Drugs ◽

Quantitative Structure ◽

Structure Activity Relationships ◽

Structure Activity ◽

Quantitative Structure Activity Relationships

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Parabolic Quantitative Structure–Activity Relationships and Photodynamic Therapy: Application of a Three-Compartment Model with Clearance to the In Vivo Quantitative Structure–Activity Relationships of a Congeneric Series of Pyropheophorbide Derivatives Used as Photosensitizers for Photodynamic Therapy

Photochemistry and Photobiology ◽

10.1562/0031-8655(1999)070<0781:pqsrap>2.3.co;2 ◽

1999 ◽

Vol 70 (5) ◽

pp. 781 ◽

Cited By ~ 2

Author(s):

W. R. Potter ◽

B. W. Henderson ◽

D. A. Bellnier ◽

R. K. Pandey ◽

L. A. Vaughan ◽

...

Keyword(s):

Photodynamic Therapy ◽

Compartment Model ◽

Quantitative Structure ◽

Structure Activity Relationships ◽

Structure Activity ◽

Three Compartment Model ◽

Quantitative Structure Activity Relationships

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Binding Affinity of Triphenyl Acrylonitriles to Estrogen Receptors: Quantitative Structure-Activity Relationships

Folia Medica ◽

10.2478/v10153-010-0005-2 ◽

2010 ◽

Vol 52 (3) ◽

Cited By ~ 1

Author(s):

Sorana Bolboacă ◽

Monica Marta ◽

Lorentz Jäntschi

Keyword(s):

Estrogen Receptors ◽

Binding Affinity ◽

Quantitative Structure ◽

Structure Activity Relationships ◽

Structure Activity ◽

Quantitative Structure Activity Relationships

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