peptide isosteres Latest Research Papers

Late-stage C(sp2)–H and C(sp3)–H glycosylation of C-aryl/alkyl glycopeptides: mechanistic insights and fluorescence labeling

Chemical Science ◽

10.1039/d0sc01260b ◽

2020 ◽

Vol 11 (25) ◽

pp. 6521-6526 ◽

Cited By ~ 9

Author(s):

Jun Wu ◽

Nikolaos Kaplaneris ◽

Shaofei Ni ◽

Felix Kaltenhäuser ◽

Lutz Ackermann

Keyword(s):

Amino Acids ◽

Late Stage ◽

Fluorescence Labeling ◽

Palladium Catalyzed ◽

Peptide Isosteres

C–H glycosylations of complex amino acids and peptides were accomplished through the assistance of triazole peptide-isosteres. The palladium-catalyzed glycosylation provided access to complex C-glycosides and fluorescent-labeled glycoamino acids.

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Allylic Amines as Key Building Blocks in the Synthesis of (E)-Alkene Peptide Isosteres

Organic Process Research & Development ◽

10.1021/op2002613 ◽

2012 ◽

Vol 16 (1) ◽

pp. 26-34 ◽

Cited By ~ 60

Author(s):

Erin M. Skoda ◽

Gary C. Davis ◽

Peter Wipf

Keyword(s):

Building Blocks ◽

Allylic Amines ◽

Peptide Isosteres

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ChemInform Abstract: Cyclopropanes as Conformationally Restricted Peptide Isosteres. Design and Synthesis of Novel Collagenase Inhibitors.

ChemInform ◽

10.1002/chin.199334255 ◽

2010 ◽

Vol 24 (34) ◽

pp. no-no

Author(s):

S. F. MARTIN ◽

C. J. OALMANN ◽

S. LIRAS

Keyword(s):

Conformationally Restricted ◽

Design And Synthesis ◽

Peptide Isosteres

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ChemInform Abstract: Use of an Alanine-Derived β-Keto Sulfone in the Synthesis of Peptide Isosteres.

ChemInform ◽

10.1002/chin.199322178 ◽

2010 ◽

Vol 24 (22) ◽

pp. no-no

Author(s):

B. LYGO

Keyword(s):

Peptide Isosteres

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ChemInform Abstract: Fluoroolefin Peptide Isosteres - Tools for Controlling Peptide Conformations.

ChemInform ◽

10.1002/chin.199501214 ◽

2010 ◽

Vol 26 (1) ◽

pp. no-no

Author(s):

L. G. BOROS ◽

B. DE CORTE ◽

R. H. GIMI ◽

J. T. WELCH ◽

Y. WU ◽

...

Keyword(s):

Peptide Conformations ◽

Peptide Isosteres

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ChemInform Abstract: Allylsilanes in Organic Synthesis: Stereoselective Synthesis of trans- Alkene Peptide Isosteres.

ChemInform ◽

10.1002/chin.199604141 ◽

2010 ◽

Vol 27 (4) ◽

pp. no-no

Author(s):

M. J. DALY ◽

R. A. WARD ◽

D. F. THOMPSON ◽

G. PROCTER

Keyword(s):

Organic Synthesis ◽

Stereoselective Synthesis ◽

Peptide Isosteres

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ChemInform Abstract: Novel Peptide Isosteres That Were Designed to Inhibit the Binding of the HIV Surface Glycoprotein (gp120) to the T Cell Surface Glycoprotein CD4.

ChemInform ◽

10.1002/chin.199838236 ◽

2010 ◽

Vol 29 (38) ◽

pp. no-no

Author(s):

M. G. B. DREW ◽

S. GORSUCH ◽

J. MANN ◽

S. YOSHIDA

Keyword(s):

T Cell ◽

Cell Surface ◽

Surface Glycoprotein ◽

Cell Surface Glycoprotein ◽

Glycoprotein Gp120 ◽

Peptide Isosteres

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ChemInform Abstract: General Asymmetric Synthesis of Hydroxymethylene and Hydroxyethylene Peptide Isosteres.

ChemInform ◽

10.1002/chin.199852094 ◽

2010 ◽

Vol 29 (52) ◽

pp. no-no

Author(s):

Y. AOYAGI ◽

R. M. WILLIAMS

Keyword(s):

Asymmetric Synthesis ◽

Peptide Isosteres

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ChemInform Abstract: Methyl- and (Trifluoromethyl)alkene Peptide Isosteres: Synthesis and Evaluation of Their Potential as β-Turn Promoters and Peptide Mimetics.

ChemInform ◽

10.1002/chin.199906171 ◽

2010 ◽

Vol 30 (6) ◽

pp. no-no

Author(s):

P. WIPF ◽

T. C. HENNINGER ◽

S. J. GEIB

Keyword(s):

Peptide Mimetics ◽

Peptide Isosteres

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ChemInform Abstract: Investigations on the Enzyme Specificity of Clostripain: A New Efficient Biocatalyst for the Synthesis of Peptide Isosteres.

ChemInform ◽

10.1002/chin.200024043 ◽

2010 ◽

Vol 31 (24) ◽

pp. no-no

Author(s):

Robert Guenther ◽

Anja Stein ◽

Frank Bordusa

Keyword(s):

Enzyme Specificity ◽

Peptide Isosteres

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peptide isosteres
Recently Published Documents

TOTAL DOCUMENTS

H-INDEX

Late-stage C(sp2)–H and C(sp3)–H glycosylation of C-aryl/alkyl glycopeptides: mechanistic insights and fluorescence labeling

Allylic Amines as Key Building Blocks in the Synthesis of (E)-Alkene Peptide Isosteres

ChemInform Abstract: Cyclopropanes as Conformationally Restricted Peptide Isosteres. Design and Synthesis of Novel Collagenase Inhibitors.

ChemInform Abstract: Use of an Alanine-Derived β-Keto Sulfone in the Synthesis of Peptide Isosteres.

ChemInform Abstract: Fluoroolefin Peptide Isosteres - Tools for Controlling Peptide Conformations.

ChemInform Abstract: Allylsilanes in Organic Synthesis: Stereoselective Synthesis of trans- Alkene Peptide Isosteres.

ChemInform Abstract: Novel Peptide Isosteres That Were Designed to Inhibit the Binding of the HIV Surface Glycoprotein (gp120) to the T Cell Surface Glycoprotein CD4.

ChemInform Abstract: General Asymmetric Synthesis of Hydroxymethylene and Hydroxyethylene Peptide Isosteres.

ChemInform Abstract: Methyl- and (Trifluoromethyl)alkene Peptide Isosteres: Synthesis and Evaluation of Their Potential as β-Turn Promoters and Peptide Mimetics.

ChemInform Abstract: Investigations on the Enzyme Specificity of Clostripain: A New Efficient Biocatalyst for the Synthesis of Peptide Isosteres.

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peptide isosteresRecently Published Documents

TOTAL DOCUMENTS

H-INDEX

Late-stage C(sp2)–H and C(sp3)–H glycosylation of C-aryl/alkyl glycopeptides: mechanistic insights and fluorescence labeling

Allylic Amines as Key Building Blocks in the Synthesis of (E)-Alkene Peptide Isosteres

ChemInform Abstract: Cyclopropanes as Conformationally Restricted Peptide Isosteres. Design and Synthesis of Novel Collagenase Inhibitors.

ChemInform Abstract: Use of an Alanine-Derived β-Keto Sulfone in the Synthesis of Peptide Isosteres.

ChemInform Abstract: Fluoroolefin Peptide Isosteres - Tools for Controlling Peptide Conformations.

ChemInform Abstract: Allylsilanes in Organic Synthesis: Stereoselective Synthesis of trans- Alkene Peptide Isosteres.

ChemInform Abstract: Novel Peptide Isosteres That Were Designed to Inhibit the Binding of the HIV Surface Glycoprotein (gp120) to the T Cell Surface Glycoprotein CD4.

ChemInform Abstract: General Asymmetric Synthesis of Hydroxymethylene and Hydroxyethylene Peptide Isosteres.

ChemInform Abstract: Methyl- and (Trifluoromethyl)alkene Peptide Isosteres: Synthesis and Evaluation of Their Potential as β-Turn Promoters and Peptide Mimetics.

ChemInform Abstract: Investigations on the Enzyme Specificity of Clostripain: A New Efficient Biocatalyst for the Synthesis of Peptide Isosteres.

peptide isosteres
Recently Published Documents