Process Research and Scale-up of a Commercialisable Route to Maraviroc (UK-427,857), a CCR-5 Receptor Antagonist

2008 ◽  
Vol 12 (6) ◽  
pp. 1104-1113 ◽  
Author(s):  
Jens Åhman ◽  
Melissa Birch ◽  
Sarah J. Haycock-Lewandowski ◽  
James, Long ◽  
Alexander Wilder
Keyword(s):  
Receptor Antagonist ◽  
Scale Up ◽  
Process Research

Process Research for (+)-Ambrisentan, an Endothelin-A Receptor Antagonist

2018 ◽  
Vol 22 (9) ◽  
pp. 1200-1207 ◽  
Author(s):  
Wei-Dong Feng ◽  
Song-Ming Zhuo ◽  
Jun Yu ◽  
Chuan-Meng Zhao ◽  
Fu-Li Zhang
Keyword(s):  
Receptor Antagonist ◽  
Process Research ◽  
Endothelin A Receptor ◽  
Endothelin A

Process Research and Initial Scale-Up of ABT-839: A Farnesyltransferase Inhibitor

2003 ◽  
pp. 59-69 ◽  
Author(s):  
Todd S. McDermott ◽  
Ramiya Premchandron ◽  
Anne E. Bailey ◽  
Lakshmi Bhagavatula ◽  
Howard E. Morton
Keyword(s):  
Scale Up ◽  
Process Research ◽  
Farnesyltransferase Inhibitor ◽  
Initial Scale

Process research toward scale-up and industrial preparation of RPR 109891 (Klerval™)

2006 ◽  
pp. 126-128
Author(s):  
James J. Mencel ◽  
Benoit J. Vanasse ◽  
Richard G. Woodward ◽  
James P. Sherbine ◽  
Robert C. Liu ◽  
...  
Keyword(s):  
Scale Up ◽  
Process Research ◽  
Industrial Preparation

Process Research and Development and Scale-up of a 4,4-Difluoro-3,3-dimethylproline Derivative

2008 ◽  
Vol 12 (2) ◽  
pp. 322-338 ◽  
Author(s):  
Francesco Rossi ◽  
Francesco Corcella ◽  
Francesco Saverio Caldarelli ◽  
Franco Heidempergher ◽  
Chiara Marchionni ◽  
...  
Keyword(s):  
Research And Development ◽  
Scale Up ◽  
Process Research

Process Research on a Phenoxybutyric Acid LTB4 Receptor Antagonist. Efficient Kilogram-Scale Synthesis of a 3,5-Bisarylphenol Core

2012 ◽  
Vol 17 (1) ◽  
pp. 114-119 ◽  
Author(s):  
Lianhe Shu ◽  
Ping Wang ◽  
Roumen Radinov ◽  
Romyr Dominique ◽  
James Wright ◽  
...  
Keyword(s):  
Receptor Antagonist ◽  
Process Research ◽  
Ltb4 Receptor

Development and Scale-Up of an Optimized Route to the Pyridazin-3-one Histamine H3 Receptor Antagonist CEP-32215

2013 ◽  
Vol 17 (5) ◽  
pp. 846-853 ◽  
Author(s):  
Yi Wang ◽  
Katrin Przyuski ◽  
Renee C. Roemmele ◽  
Robert L. Hudkins ◽  
Roger P. Bakale
Keyword(s):  
Receptor Antagonist ◽  
Scale Up ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Histamine H3

Process Research and Development of a MTP Inhibitor: Another Case of Disappearing Polymorphs upon Scale-up

2010 ◽  
Vol 14 (4) ◽  
pp. 878-882 ◽  
Author(s):  
Mahavir Prashad ◽  
Paul Sutton ◽  
Raeann Wu ◽  
Bin Hu ◽  
James Vivelo ◽  
...  
Keyword(s):  
Research And Development ◽  
Scale Up ◽  
Process Research
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