Development and Scale-Up of an Optimized Route to the Pyridazin-3-one Histamine H3 Receptor Antagonist CEP-32215

2013 ◽  
Vol 17 (5) ◽  
pp. 846-853 ◽  
Author(s):  
Yi Wang ◽  
Katrin Przyuski ◽  
Renee C. Roemmele ◽  
Robert L. Hudkins ◽  
Roger P. Bakale
Keyword(s):  
Receptor Antagonist ◽  
Scale Up ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Histamine H3

Ameliorating effects of histamine H3 receptor antagonist E177 on acute pentylenetetrazole-induced memory impairments in rats

2021 ◽  
Vol 405 ◽  
pp. 113193
Author(s):  
Alaa Alachkar ◽  
Mohamed Lotfy ◽  
Ernest Adeghate ◽  
Dorota Łażewska ◽  
Katarzyna Kieć-Kononowicz ◽  
...  
Keyword(s):  
Receptor Antagonist ◽  
Histamine H3 Receptor ◽  
Memory Impairments ◽  
H3 Receptor ◽  
Histamine H3

P1-235: Effects of the novel histamine H3 receptor antagonist S 38093 in a non-human primate model of cognitive dysfunction

2009 ◽  
Vol 5 (4S_Part_8) ◽  
pp. P245-P245
Author(s):  
Jay S. Schneider ◽  
Emmanuel Decamp ◽  
Michael Hill ◽  
Erwan Bezard ◽  
Alan Crossman ◽  
...  
Keyword(s):  
Receptor Antagonist ◽  
Cognitive Dysfunction ◽  
The Novel ◽  
Primate Model ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Human Primate ◽  
Histamine H3

scholarly journals Influence of a selective histamine H3 receptor antagonist on hypothalamic neural activity, food intake and body weight

2005 ◽  
Vol 29 (12) ◽  
pp. 1402-1412 ◽  
Author(s):  
K Malmlöf ◽  
F Zaragoza ◽  
V Golozoubova ◽  
H H F Refsgaard ◽  
T Cremers ◽  
...  
Keyword(s):  
Body Weight ◽  
Food Intake ◽  
Receptor Antagonist ◽  
Neural Activity ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Histamine H3

Anticonvulsant and procognitive properties of the non-imidazole histamine H3 receptor antagonist DL77 in male adult rats

2016 ◽  
Vol 106 ◽  
pp. 46-55 ◽  
Author(s):  
Bassem Sadek ◽  
Ali Saad ◽  
Dhanasekaran Subramanian ◽  
Mohamed Shafiullah ◽  
Dorota Łażewska ◽  
...  
Keyword(s):  
Receptor Antagonist ◽  
Adult Rats ◽  
Male Adult ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Histamine H3

Histamine H3 receptor antagonist decreases cue-induced alcohol reinstatement in mice

2016 ◽  
Vol 106 ◽  
pp. 156-163 ◽  
Author(s):  
Saara Nuutinen ◽  
Tiia Mäki ◽  
Stanislav Rozov ◽  
Pia Bäckström ◽  
Petri Hyytiä ◽  
...  
Keyword(s):  
Receptor Antagonist ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Histamine H3

Pharmacokinetics and tissue distribution of the new non-imidazole histamine H3 receptor antagonist 1-[3-(4-tert-butylphenoxy) propyl]piperidine in rats

Xenobiotica ◽  
2015 ◽  
Vol 45 (10) ◽  
pp. 912-920 ◽  
Author(s):  
Malgorzata Szafarz ◽  
Agata Kryczyk ◽  
Dorota Lazewska ◽  
Katarzyna Kiec-Kononowicz ◽  
Elzbieta Wyska
Keyword(s):  
Receptor Antagonist ◽  
Tissue Distribution ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Histamine H3
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