Synthesis and Biological Evaluation of Orally Active Prodrugs of Indomethacin

Babasaheb P. Bandgar; Rajendra Janardan Sarangdhar; Santosh Viswakarma; Fakrudeen Ali Ahamed

doi:10.1021/jm101085j

Synthesis and Biological Evaluation of Orally Active Prodrugs of Indomethacin

Journal of Medicinal Chemistry ◽

10.1021/jm101085j ◽

2011 ◽

Vol 54 (5) ◽

pp. 1191-1201 ◽

Cited By ~ 43

Author(s):

Babasaheb P. Bandgar ◽

Rajendra Janardan Sarangdhar ◽

Santosh Viswakarma ◽

Fakrudeen Ali Ahamed

Keyword(s):

Biological Evaluation ◽

Orally Active ◽

Synthesis And Biological Evaluation

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Design, synthesis and biological evaluation of (2S,3R,4R,5S,6R)-5-fluoro-6-(hydroxymethyl)-2-aryltetrahydro-2H-pyran-3,4-diols as potent and orally active SGLT dual inhibitors

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2018.09.025 ◽

2018 ◽

Vol 28 (21) ◽

pp. 3446-3453 ◽

Cited By ~ 2

Author(s):

Guozhang Xu ◽

Michael D. Gaul ◽

Gee-Hong Kuo ◽

Fuyong Du ◽

June Zhi Xu ◽

...

Keyword(s):

Biological Evaluation ◽

Design Synthesis ◽

Dual Inhibitors ◽

Orally Active ◽

Synthesis And Biological Evaluation

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Synthesis and Biological Evaluation ofN-Heterocyclic Indolyl Glyoxylamides as Orally Active Anticancer Agents

Journal of Medicinal Chemistry ◽

10.1021/jm020471r ◽

2003 ◽

Vol 46 (9) ◽

pp. 1706-1715 ◽

Cited By ~ 114

Author(s):

Wen-Tai Li ◽

Der-Ren Hwang ◽

Ching-Ping Chen ◽

Chien-Wei Shen ◽

Chen-Long Huang ◽

...

Keyword(s):

Anticancer Agents ◽

Biological Evaluation ◽

Orally Active ◽

Synthesis And Biological Evaluation

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Synthesis and Biological Evaluation of [4-(2-Phenylethenesulfonylmethyl)phenyl]-quinazolin-4-yl-amines as Orally Active Anticancer Agents.

ChemInform ◽

10.1002/chin.200417153 ◽

2004 ◽

Vol 35 (17) ◽

Author(s):

Vedula M. Sharma ◽

et al. et al.

Keyword(s):

Anticancer Agents ◽

Biological Evaluation ◽

Orally Active ◽

Synthesis And Biological Evaluation

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Synthesis and biological evaluation of taxinine analogues as orally active multidrug resistance reversal agents in cancer

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2004.06.089 ◽

2004 ◽

Vol 14 (18) ◽

pp. 4767-4770 ◽

Cited By ~ 17

Author(s):

Xin Zhao ◽

Jun Gu ◽

Dali Yin ◽

Xiaoguang Chen

Keyword(s):

Multidrug Resistance ◽

Biological Evaluation ◽

Reversal Agents ◽

Resistance Reversal ◽

Orally Active ◽

Synthesis And Biological Evaluation

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Synthesis and biological evaluation of ester prodrugs of benzafibrate as orally active hypolipidemic agents

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2012.08.036 ◽

2012 ◽

Vol 57 ◽

pp. 217-224 ◽

Cited By ~ 7

Author(s):

Babasaheb P. Bandgar ◽

Rajendra J. Sarangdhar ◽

Khan Fruthous ◽

Jeyamurugan Mookkan ◽

Shilpee Chaudhary ◽

...

Keyword(s):

Biological Evaluation ◽

Hypolipidemic Agents ◽

Orally Active ◽

Synthesis And Biological Evaluation ◽

Ester Prodrugs

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Design, Synthesis and Biological Evaluation of a Novel Series of Potent, Orally Active Adenosine A1 Receptor Antagonists with High Blood-Brain Barrier Permeability

Chemical and Pharmaceutical Bulletin ◽

10.1248/cpb.49.988 ◽

2001 ◽

Vol 49 (8) ◽

pp. 988-998 ◽

Cited By ~ 21

Author(s):

Satoru KURODA ◽

Fujiko TAKAMURA ◽

Yoshiyuki TENDA ◽

Hiromichi ITANI ◽

Yasuyo TOMISHIMA ◽

...

Keyword(s):

Blood Brain Barrier ◽

Biological Evaluation ◽

Brain Barrier ◽

Receptor Antagonists ◽

Design Synthesis ◽

Barrier Permeability ◽

Blood Brain Barrier Permeability ◽

Brain Barrier Permeability ◽

Orally Active ◽

Synthesis And Biological Evaluation

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Design, synthesis, and biological evaluation of triazolopiperazine-based β-amino amides as potent, orally active dipeptidyl peptidase IV (DPP-4) inhibitors

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2007.07.100 ◽

2007 ◽

Vol 17 (21) ◽

pp. 5934-5939 ◽

Cited By ~ 29

Author(s):

Jennifer E. Kowalchick ◽

Barbara Leiting ◽

KellyAnn D. Pryor ◽

Frank Marsilio ◽

Joseph K. Wu ◽

...

Keyword(s):

Dipeptidyl Peptidase ◽

Biological Evaluation ◽

Dipeptidyl Peptidase Iv ◽

Design Synthesis ◽

Orally Active ◽

Synthesis And Biological Evaluation ◽

Amino Amides

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Synthesis and biological evaluation of 2-amino-1-thiazolyl imidazoles as orally active anticancer agents

Investigational New Drugs ◽

10.1007/s10637-010-9547-7 ◽

2010 ◽

Vol 30 (1) ◽

pp. 164-175 ◽

Cited By ~ 5

Author(s):

Wen-Tai Li ◽

Der-Ren Hwang ◽

Jen-Shin Song ◽

Ching-Ping Chen ◽

Tung-Wei Chen ◽

...

Keyword(s):

Anticancer Agents ◽

Biological Evaluation ◽

Orally Active ◽

Synthesis And Biological Evaluation

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Design, Synthesis, and Biological Evaluation of (2R,αS)-3,4-Dihydro-2-[3-(1,1,2,2-tetrafluoroethoxy)phenyl]-5-[3-(trifluoromethoxy)-phenyl]-α-(trifluoromethyl)-1(2H)-quinolineethanol as Potent and Orally Active Cholesteryl Ester Transfer Protein Inhibitor

Journal of Medicinal Chemistry ◽

10.1021/jm801319d ◽

2009 ◽

Vol 52 (6) ◽

pp. 1768-1772 ◽

Cited By ~ 31

Author(s):

Gee-Hong Kuo ◽

Thomas Rano ◽

Patricia Pelton ◽

Keith T. Demarest ◽

Alan C. Gibbs ◽

...

Keyword(s):

Cholesteryl Ester ◽

Cholesteryl Ester Transfer Protein ◽

Biological Evaluation ◽

Protein Inhibitor ◽

Design Synthesis ◽

Transfer Protein ◽

Orally Active ◽

Synthesis And Biological Evaluation

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A Simple Stereoselective Synthesis and Biological Evaluation of FR181157: Orally Active Prostacyclin Mimetic.

ChemInform ◽

10.1002/chin.200414227 ◽

2004 ◽

Vol 35 (14) ◽

Author(s):

Kouji Hattori ◽

Seiichiro Tabuchi ◽

Osamu Okitsu ◽

Kiyoshi Taniguchi

Keyword(s):

Stereoselective Synthesis ◽

Biological Evaluation ◽

Orally Active ◽

Synthesis And Biological Evaluation

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