Non-peptidic Inhibitors of Human Leukocyte Elastase. 1. The Design and Synthesis of Pyridone-Containing Inhibitors

1994 ◽  
Vol 37 (19) ◽  
pp. 3090-3099 ◽  
Author(s):  
Peter Warner ◽  
Rosalyn C. Green ◽  
Bruce Gomes ◽  
Anne M. Strimpler
Keyword(s):  
Human Leukocyte ◽  
Leukocyte Elastase ◽  
Design And Synthesis ◽  
Elastase 1 ◽  
Human Leukocyte Elastase ◽  
Peptidic Inhibitors

Design and Synthesis of Hydrazinopeptides and Their Evaluation as Human Leukocyte Elastase Inhibitors

1998 ◽  
Vol 41 (24) ◽  
pp. 4833-4843 ◽  
Author(s):  
Laure Guy ◽  
Joëlle Vidal ◽  
André Collet ◽  
Augustin Amour ◽  
Michèle Reboud-Ravaux
Keyword(s):  
Human Leukocyte ◽  
Leukocyte Elastase ◽  
Design And Synthesis ◽  
Human Leukocyte Elastase

Design and synthesis of 4H-3,1-benzoxazin-4-ones as potent alternate substrate inhibitors of human leukocyte elastase

1990 ◽  
Vol 33 (2) ◽  
pp. 464-479 ◽  
Author(s):  
Allen Krantz ◽  
Robin W. Spencer ◽  
Tim F. Tam ◽  
Teng Jiam Liak ◽  
Leslie J. Copp ◽  
...  
Keyword(s):  
Human Leukocyte ◽  
Leukocyte Elastase ◽  
Design And Synthesis ◽  
Human Leukocyte Elastase ◽  
Alternate Substrate

Orally active .beta.-lactam inhibitors of human leukocyte elastase-1. Activity of 3,3-diethyl-2-azetidinones

1992 ◽  
Vol 35 (21) ◽  
pp. 3745-3754 ◽  
Author(s):  
Shrenik K. Shah ◽  
Conrad P. Dorn ◽  
Paul E. Finke ◽  
Jeffrey J. Hale ◽  
William K. Hagmann ◽  
...  
Keyword(s):  
Human Leukocyte ◽  
Beta Lactam ◽  
Leukocyte Elastase ◽  
Elastase 1 ◽  
Human Leukocyte Elastase ◽  
Orally Active

Design of Orally Active, Non-Peptidic Inhibitors of Human Leukocyte Elastase

1994 ◽  
Vol 37 (9) ◽  
pp. 1259-1261 ◽  
Author(s):  
Frederick J. Brown ◽  
Donald W. Andisik ◽  
Peter R. Bernstein ◽  
Craig B. Bryant ◽  
Chris Ceccarelli ◽  
...  
Keyword(s):  
Human Leukocyte ◽  
Leukocyte Elastase ◽  
Human Leukocyte Elastase ◽  
Peptidic Inhibitors ◽  
Orally Active

Peptidyl Carbamates as Human Leukocyte Elastase Inhibitors: Design and Synthesis of Desmosine-Like Tetrapeptidyl Carbamate Inhibitors

1993 ◽  
Vol 7 (4) ◽  
pp. 275-301 ◽  
Author(s):  
George A. Digenis ◽  
William R. Banks ◽  
Masasuki Kato ◽  
William F. Rencher ◽  
Bushra J. Agha
Keyword(s):  
Human Leukocyte ◽  
Leukocyte Elastase ◽  
Design And Synthesis ◽  
Human Leukocyte Elastase ◽  
Carbamate Inhibitors

Inhibition of human leukocyte elastase. 1. Inhibition by C-7-substituted cephalosporin tert-butyl esters

1990 ◽  
Vol 33 (9) ◽  
pp. 2513-2521 ◽  
Author(s):  
James B. Doherty ◽  
Bonnie M. Ashe ◽  
Peter L. Barker ◽  
Thomas J. Blacklock ◽  
John W. Butcher ◽  
...  
Keyword(s):  
Human Leukocyte ◽  
Leukocyte Elastase ◽  
Tert Butyl ◽  
Butyl Esters ◽  
Elastase 1 ◽  
Human Leukocyte Elastase

ChemInform Abstract: Orally Active β-Lactam Inhibitors of Human Leukocyte Elastase-1. Activity of 3,3-Diethyl-2-azetidinones.

ChemInform ◽  
2010 ◽  
Vol 24 (20) ◽  
pp. no-no
Author(s):  
S. K. SHAH ◽  
C. P. JUN. DORN ◽  
P. E. FINKE ◽  
J. J. HALE ◽  
W. K. HAGMANN ◽  
...  
Keyword(s):  
Human Leukocyte ◽  
Leukocyte Elastase ◽  
Elastase 1 ◽  
Human Leukocyte Elastase ◽  
Orally Active
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