A Slow-Tight Binding Inhibitor of Dopamine β-Monooxygenase:  A Transition State Analogue for the Product Release Step†

Sanjeewa P. Dharmasena; D. Shyamali Wimalasena; Kandatege Wimalasena

doi:10.1021/bi0262606

A Slow-Tight Binding Inhibitor of Dopamine β-Monooxygenase: A Transition State Analogue for the Product Release Step†

Biochemistry ◽

10.1021/bi0262606 ◽

2002 ◽

Vol 41 (41) ◽

pp. 12414-12420 ◽

Cited By ~ 7

Author(s):

Sanjeewa P. Dharmasena ◽

D. Shyamali Wimalasena ◽

Kandatege Wimalasena

Keyword(s):

Transition State ◽

Tight Binding ◽

Product Release ◽

Transition State Analogue

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Effect of alcohol configuration on tight binding inhibition of HIV protease by hydroxyethylamine transition-state analogue inhibitors

Peptides 1990 ◽

10.1007/978-94-011-3034-9_327 ◽

1991 ◽

pp. 790-791

Author(s):

Daniel H. Rich ◽

Jeremy Green ◽

J. V. N. Vara Prasad ◽

C. Q. Sun ◽

Mihaly Toth ◽

...

Keyword(s):

Transition State ◽

Tight Binding ◽

Hiv Protease ◽

Transition State Analogue ◽

Binding Inhibition ◽

Transition State Analogue Inhibitors

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Origin of Tight Binding of a Near-Perfect Transition-State Analogue by Cytidine Deaminase: Implications for Enzyme Catalysis

Journal of the American Chemical Society ◽

10.1021/ja0439625 ◽

2005 ◽

Vol 127 (9) ◽

pp. 3191-3197 ◽

Cited By ~ 28

Author(s):

Haobo Guo ◽

Niny Rao ◽

Qin Xu ◽

Hong Guo

Keyword(s):

Transition State ◽

Enzyme Catalysis ◽

Cytidine Deaminase ◽

Tight Binding ◽

Transition State Analogue

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Ketone-substrate analogues of Clostridium histolyticum collagenases: tight-binding transition-state analogue inhibitors

Biochemistry ◽

10.1021/bi00412a016 ◽

1988 ◽

Vol 27 (12) ◽

pp. 4299-4304 ◽

Cited By ~ 9

Author(s):

Kasim A. Mookhtiar ◽

Damian Grobelny ◽

Richard E. Galardy ◽

Harold E. Van Wart

Keyword(s):

Transition State ◽

Tight Binding ◽

Clostridium Histolyticum ◽

Substrate Analogues ◽

Transition State Analogue ◽

Transition State Analogue Inhibitors

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Faculty Opinions recommendation of L-Enantiomers of transition state analogue inhibitors bound to human purine nucleoside phosphorylase.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1097544.553622 ◽

2008 ◽

Author(s):

Wayne Guida

Keyword(s):

Transition State ◽

Purine Nucleoside Phosphorylase ◽

Purine Nucleoside ◽

Nucleoside Phosphorylase ◽

Transition State Analogue ◽

Transition State Analogue Inhibitors

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Crystallization and preliminary x-ray studies of spinach ribulose 1,5-bisphosphate carboxylase/oxygenase complexed with activator and a transition state analogue.

Journal of Biological Chemistry ◽

10.1016/s0021-9258(17)43825-7 ◽

1983 ◽

Vol 258 (23) ◽

pp. 14088-14090

Author(s):

I Andersson ◽

A C Tjäder ◽

E Cedergren-Zeppezauer ◽

C I Brändén

Keyword(s):

Transition State ◽

Bisphosphate Carboxylase ◽

X Ray ◽

Transition State Analogue

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A metabolically stable tight-binding transition-state inhibitor of glyoxalase-I

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2006.08.121 ◽

2006 ◽

Vol 16 (23) ◽

pp. 6039-6042 ◽

Cited By ~ 14

Author(s):

Swati S. More ◽

Robert Vince

Keyword(s):

Transition State ◽

Tight Binding ◽

Glyoxalase I

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Crystal structure of cobra-venom phospholipase A2 in a complex with a transition-state analogue

Science ◽

10.1126/science.2274787 ◽

1990 ◽

Vol 250 (4987) ◽

pp. 1560-1563 ◽

Cited By ~ 227

Author(s):

S. White ◽

D. Scott ◽

Z. Otwinowski ◽

M. Gelb ◽

P. Sigler

Keyword(s):

Crystal Structure ◽

Transition State ◽

Phospholipase A2 ◽

Cobra Venom ◽

Transition State Analogue

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An Esterolytic Imprinted Polymer Prepared via a Silica-Supported Transition State Analogue

Chemistry of Materials ◽

10.1021/cm0352394 ◽

2004 ◽

Vol 16 (14) ◽

pp. 2745-2749 ◽

Cited By ~ 21

Author(s):

Kristian Lettau ◽

Axel Warsinke ◽

André Laschewsky ◽

Klaus Mosbach ◽

Ecevit Yilmaz ◽

...

Keyword(s):

Transition State ◽

Imprinted Polymer ◽

Transition State Analogue

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A new class of C-nucleoside analogues. 1-(S)-aryl-1,4-dideoxy-1,4-imino-D-ribitols, transition state analogue inhibitors of nucleoside hydrolase

Tetrahedron Letters ◽

10.1016/s0040-4039(00)79290-2 ◽

1993 ◽

Vol 34 (45) ◽

pp. 7213-7216 ◽

Cited By ~ 51

Author(s):

Benjamin A. Horenstein ◽

Roger F. Zabinski ◽

Vern L. Schramm

Keyword(s):

Transition State ◽

Nucleoside Analogues ◽

New Class ◽

Nucleoside Hydrolase ◽

Transition State Analogue ◽

Transition State Analogue Inhibitors

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Transition State Analogue Inhibitors of 5′-Deoxyadenosine/5′-Methylthioadenosine Nucleosidase from Mycobacterium tuberculosis

Biochemistry ◽

10.1021/acs.biochem.7b00576 ◽

2017 ◽

Vol 56 (38) ◽

pp. 5090-5098 ◽

Cited By ~ 9

Author(s):

Hilda A. Namanja-Magliano ◽

Gary B. Evans ◽

Rajesh K. Harijan ◽

Peter C. Tyler ◽

Vern L. Schramm

Keyword(s):

Mycobacterium Tuberculosis ◽

Transition State ◽

Transition State Analogue ◽

Transition State Analogue Inhibitors

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