scholarly journals Chemoproteomic Study Uncovers HemK2/KMT9 As a New Target for NTMT1 Bisubstrate Inhibitors

2021 ◽  
Author(s):  
Dongxing Chen ◽  
Ying Meng ◽  
Dan Yu ◽  
Nicholas Noinaj ◽  
Xiaodong Cheng ◽  
...  
Keyword(s):  
Bisubstrate Inhibitors

scholarly journals Novel Bisubstrate Inhibitors for Protein N-Terminal Acetyltransferase D

2021 ◽  
Author(s):  
Youchao Deng ◽  
Sunbin Deng ◽  
Yi-Hsun Ho ◽  
Sarah M. Gardner ◽  
Zhi Huang ◽  
...  
Keyword(s):  
Bisubstrate Inhibitors

scholarly journals Structure-Based Design, Synthesis, and in vitro Evaluation of Bisubstrate Inhibitors for CatecholO-Methyltransferase (COMT)

2000 ◽  
Vol 6 (6) ◽  
pp. 971-982 ◽  
Author(s):  
Birgit Masjost ◽  
Patrick Ballmer ◽  
Edilio Borroni ◽  
Gerhard Zürcher ◽  
Fritz K. Winkler ◽  
...  
Keyword(s):  
Design Synthesis ◽  
In Vitro Evaluation ◽  
Bisubstrate Inhibitors

Unexpected CK2β-antagonistic functionality of bisubstrate inhibitors targeting protein kinase CK2

2020 ◽  
Vol 96 ◽  
pp. 103608 ◽  
Author(s):  
Markus Pietsch ◽  
Kaido Viht ◽  
Alexander Schnitzler ◽  
Ramesh Ekambaram ◽  
Michaela Steinkrüger ◽  
...  
Keyword(s):  
Protein Kinase ◽  
Protein Kinase Ck2 ◽  
Kinase Ck2 ◽  
Bisubstrate Inhibitors

scholarly journals Bisubstrate inhibitors to target histone acetyltransferase 1

2019 ◽  
Vol 93 (5) ◽  
pp. 865-873 ◽  
Author(s):  
Liza Ngo ◽  
Tyler Brown ◽  
Yujun G. Zheng
Keyword(s):  
Histone Acetyltransferase ◽  
Bisubstrate Inhibitors

Molecular Recognition at the Active Site of Catechol‐ O ‐methyltransferase (COMT): Adenine Replacements in Bisubstrate Inhibitors

2011 ◽  
Vol 17 (23) ◽  
pp. 6369-6381 ◽  
Author(s):  
Manuel Ellermann ◽  
Ralph Paulini ◽  
Roland Jakob‐Roetne ◽  
Christian Lerner ◽  
Edilio Borroni ◽  
...  
Keyword(s):  
Molecular Recognition ◽  
Active Site ◽  
Bisubstrate Inhibitors

scholarly journals Design of potential bisubstrate inhibitors against Mycobacterium tuberculosis (Mtb) 1-deoxy-d-xylulose 5-phosphate reductoisomerase (Dxr)—evidence of a novel binding mode

MedChemComm ◽  
2013 ◽  
Vol 4 (7) ◽  
pp. 1099 ◽  
Author(s):  
Géraldine San Jose ◽  
Emily R. Jackson ◽  
Eugene Uh ◽  
Chinchu Johny ◽  
Amanda Haymond ◽  
...  
Keyword(s):  
Mycobacterium Tuberculosis ◽  
Binding Mode ◽  
Bisubstrate Inhibitors

Synthesis and Biological Evaluation of Potent Bisubstrate Inhibitors of the Enzyme CatecholO-Methyltransferase (COMT) Lacking a Nitro Group

2006 ◽  
Vol 89 (9) ◽  
pp. 1856-1887 ◽  
Author(s):  
Ralph Paulini ◽  
Christian Lerner ◽  
François Diederich ◽  
Roland Jakob-Roetne ◽  
Gerhard Zürcher ◽  
...  
Keyword(s):  
Nitro Group ◽  
Biological Evaluation ◽  
Bisubstrate Inhibitors ◽  
Synthesis And Biological Evaluation
Sign in / Sign up

Export Citation Format

Share Document