Bisubstrate inhibitors to target histone acetyltransferase 1

Liza Ngo; Tyler Brown; Yujun G. Zheng

doi:10.1111/cbdd.13476

Bisubstrate inhibitors to target histone acetyltransferase 1

Chemical Biology & Drug Design ◽

10.1111/cbdd.13476 ◽

2019 ◽

Vol 93 (5) ◽

pp. 865-873 ◽

Cited By ~ 8

Author(s):

Liza Ngo ◽

Tyler Brown ◽

Yujun G. Zheng

Keyword(s):

Histone Acetyltransferase ◽

Bisubstrate Inhibitors

Download Full-text

New Potent Bisubstrate Inhibitors of Histone Acetyltransferase p300: Design, Synthesis and Biological Evaluation

Chemical Biology & Drug Design ◽

10.1111/j.1747-0285.2010.01056.x ◽

2010 ◽

Vol 77 (1) ◽

pp. 86-92 ◽

Cited By ~ 14

Author(s):

Franciane Ho A Kwie ◽

Martine Briet ◽

David Soupaya ◽

Pascal Hoffmann ◽

Marie Maturano ◽

...

Keyword(s):

Histone Acetyltransferase ◽

Biological Evaluation ◽

Design Synthesis ◽

Bisubstrate Inhibitors ◽

Synthesis And Biological Evaluation ◽

Acetyltransferase P300

Download Full-text

Assays of nucleosome assembly and the inhibition of histone acetyltransferase activity. (6) Reconstitution of chromatin; (7) Analysis of nucleoproteins on an agarose gel; and (8) Purification of reconstituted chromatin on a sucrose gradient

Protocol Exchange ◽

10.1038/nprot.2007.338 ◽

2007 ◽

Author(s):

Takahito Yamasaki ◽

Takehide Murata ◽

Chunyuan Jin ◽

Kohsuke Kato ◽

Michiya Noguchi ◽

...

Keyword(s):

Sucrose Gradient ◽

Histone Acetyltransferase ◽

Agarose Gel ◽

Nucleosome Assembly ◽

Acetyltransferase Activity ◽

Histone Acetyltransferase Activity

Download Full-text

Assays of nucleosome assembly and the inhibition of histone acetyltransferase activity. (5) Preparation of core histones

Protocol Exchange ◽

10.1038/nprot.2007.337 ◽

2007 ◽

Author(s):

Takahito Yamasaki ◽

Takehide Murata ◽

Chunyuan Jin ◽

Kohsuke Kato ◽

Michiya Noguchi ◽

...

Keyword(s):

Histone Acetyltransferase ◽

Nucleosome Assembly ◽

Acetyltransferase Activity ◽

Core Histones ◽

Histone Acetyltransferase Activity

Download Full-text

Histone acetyltransferase HTATIP - [Isoform 1]

Targeted Protein Database ◽

10.2970/tpdb.2008.136 ◽

2008 ◽

Author(s):

Lise Mattera

Keyword(s):

Histone Acetyltransferase

Download Full-text

Faculty Opinions recommendation of Tetrahymena histone acetyltransferase A: a homolog to yeast Gcn5p linking histone acetylation to gene activation.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1003340.30205 ◽

2001 ◽

Author(s):

Michael Meisterernst

Keyword(s):

Histone Acetylation ◽

Histone Acetyltransferase ◽

Gene Activation

Download Full-text

Faculty Opinions recommendation of CBP histone acetyltransferase activity is a critical component of memory consolidation.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1020555.232666 ◽

2004 ◽

Author(s):

Hilmar Bading

Keyword(s):

Memory Consolidation ◽

Histone Acetyltransferase ◽

Critical Component ◽

Acetyltransferase Activity ◽

Histone Acetyltransferase Activity

Download Full-text

Faculty Opinions recommendation of Fungal Rtt109 histone acetyltransferase is an unexpected structural homolog of metazoan p300/CBP.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1115528.573845 ◽

2008 ◽

Author(s):

Xiaodong Cheng

Keyword(s):

Histone Acetyltransferase

Download Full-text

Faculty Opinions recommendation of Fungal Rtt109 histone acetyltransferase is an unexpected structural homolog of metazoan p300/CBP.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1115528.571568 ◽

2008 ◽

Author(s):

Stephen Jackson

Keyword(s):

Histone Acetyltransferase

Download Full-text

Faculty Opinions recommendation of Members of the GCN5 histone acetyltransferase complex regulate PLETHORA-mediated root stem cell niche maintenance and transit amplifying cell proliferation in Arabidopsis.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1161841.623456 ◽

2009 ◽

Author(s):

Elena Alvarez-Buylla ◽

Adriana Garay

Keyword(s):

Cell Proliferation ◽

Stem Cell ◽

Stem Cell Niche ◽

Histone Acetyltransferase ◽

Root Stem Cell ◽

Cell Niche

Download Full-text

Faculty Opinions recommendation of A barcode screen for epigenetic regulators reveals a role for the NuB4/HAT-B histone acetyltransferase complex in histone turnover.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.14257968.15771073 ◽

2012 ◽

Author(s):

Alain Verreault ◽

Benoit Guillemette

Keyword(s):

Histone Acetyltransferase ◽

Epigenetic Regulators

Download Full-text