scholarly journals Design, Synthesis and Evaluation of 2,4‐Diaminoquinazoline Derivatives as Potential Tubulin Polymerization Inhibitors

ChemMedChem ◽  
2020 ◽  
Vol 15 (19) ◽  
pp. 1802-1812
Author(s):  
Frida S. Herrera‐Vázquez ◽  
Félix Matadamas‐Martínez ◽  
Rodrigo Aguayo‐Ortiz ◽  
Laura Dominguez ◽  
Teresa Ramírez‐Apan ◽  
...  
Keyword(s):  
Tubulin Polymerization ◽  
Design Synthesis ◽  
Tubulin Polymerization Inhibitors

Design, synthesis and antiproliferative activity of the new conjugates of E7010 and resveratrol as tubulin polymerization inhibitors

2016 ◽  
Vol 14 (4) ◽  
pp. 1382-1394 ◽  
Author(s):  
Ahmed Kamal ◽  
Md. Ashraf ◽  
Shaik Thokhir Basha ◽  
S. M. Ali Hussaini ◽  
Shamshair Singh ◽  
...  
Keyword(s):  
Antiproliferative Activity ◽  
Tubulin Polymerization ◽  
Design Synthesis ◽  
New Class ◽  
Tubulin Polymerization Inhibitors ◽  
Amine Conjugates

A new class of (E)-N-phenyl-3-styrylpyridin-2-amine conjugates were designed and synthesized on the basis of E7010 and resveratrol scaffolds.

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