glycogen phosphorylase inhibitor Latest Research Papers

Glycogen phosphorylase inhibitor, 2,3‐bis[(2E)‐3‐(4‐hydroxyphenyl)prop‐2‐enamido] butanedioic acid (BF142), improves baseline insulin secretion of MIN6 insulinoma cells

PLoS ONE ◽

10.1371/journal.pone.0236081 ◽

2020 ◽

Vol 15 (9) ◽

pp. e0236081

Author(s):

Lilla Nagy ◽

Ferenc Béke ◽

László Juhász ◽

Tünde Kovács ◽

Éva Juhász-Tóth ◽

...

Keyword(s):

Insulin Secretion ◽

Glycogen Phosphorylase ◽

Butanedioic Acid ◽

Insulinoma Cells ◽

Glycogen Phosphorylase Inhibitor

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Synthetic flavonoid derivatives targeting the glycogen phosphorylase inhibitor site: QM/MM-PBSA motivated synthesis of substituted 5,7-dihydroxyflavones, crystallography, in vitro kinetics and ex-vivo cellular experiments reveal novel potent inhibitors

Bioorganic Chemistry ◽

10.1016/j.bioorg.2020.104003 ◽

2020 ◽

Vol 102 ◽

pp. 104003 ◽

Cited By ~ 1

Author(s):

Ben A. Chetter ◽

Efthimios Kyriakis ◽

Daniel Barr ◽

Aikaterini G. Karra ◽

Elisabeth Katsidou ◽

...

Keyword(s):

Glycogen Phosphorylase ◽

Ex Vivo ◽

In Vitro Kinetics ◽

Glycogen Phosphorylase Inhibitor

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Effects of Intracerebroventricular Glycogen Phosphorylase Inhibitor CP-316,819 Infusion on Hypothalamic Glycogen Content and Metabolic Neuron AMPK Activity and Neurotransmitter Expression in Male Rat

Journal of Molecular Neuroscience ◽

10.1007/s12031-019-01471-0 ◽

2020 ◽

Vol 70 (5) ◽

pp. 647-658 ◽

Cited By ~ 3

Author(s):

Mostafa M. H. Ibrahim ◽

Khaggeswar Bheemanapally ◽

Hussain N. Alhamami ◽

Karen P. Briski

Keyword(s):

Glycogen Phosphorylase ◽

Glycogen Content ◽

Male Rat ◽

Ampk Activity ◽

Glycogen Phosphorylase Inhibitor

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Multiscale time-resolved fluorescence study of a glycogen phosphorylase inhibitor combined with quantum chemistry calculations

Physical Chemistry Chemical Physics ◽

10.1039/c8cp07538g ◽

2019 ◽

Vol 21 (14) ◽

pp. 7685-7696 ◽

Cited By ~ 2

Author(s):

Valentin Maffeis ◽

Konstantinos Mavreas ◽

Filippo Monti ◽

Michael Mamais ◽

Thomas Gustavsson ◽

...

Keyword(s):

Quantum Chemistry ◽

Glycogen Phosphorylase ◽

Potent Inhibitor ◽

Time Resolved Fluorescence ◽

Fluorescence Study ◽

Time Resolved ◽

Quantum Chemistry Calculations ◽

Glycogen Phosphorylase Inhibitor

A study of the first fluorescent potent inhibitor of glycogen phosphorylase showcases how emission is controlled by two independent rotations of two aromatic moieties.

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Novel Liver-targeted conjugates of Glycogen Phosphorylase Inhibitor PSN-357 for the Treatment of Diabetes: Design, Synthesis, Pharmacokinetic and Pharmacological Evaluations

Scientific Reports ◽

10.1038/srep42251 ◽

2017 ◽

Vol 7 (1) ◽

Author(s):

Liying Zhang ◽

Chengjun Song ◽

Guangxin Miao ◽

Lianzhi Zhao ◽

Zhiwei Yan ◽

...

Keyword(s):

Glycogen Phosphorylase ◽

Design Synthesis ◽

Treatment Of Diabetes ◽

Glycogen Phosphorylase Inhibitor

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Insulin Sensitivity is Modified by a Glycogen Phosphorylase Inhibitor: Glucopyranosylidene-Spiro-Thiohydantoin in Streptozotocin-Induced Diabetic Rats

Current Topics in Medicinal Chemistry ◽

10.2174/1568026615666150622091407 ◽

2015 ◽

Vol 15 (23) ◽

pp. 2390-2394 ◽

Cited By ~ 23

Author(s):

Tibor Docsa ◽

Balazs Marics ◽

Jozsef Nemeth ◽

Csaba Huse ◽

Laszlo Somsak ◽

...

Keyword(s):

Insulin Sensitivity ◽

Glycogen Phosphorylase ◽

Diabetic Rats ◽

Glycogen Phosphorylase Inhibitor

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Cover Picture: Structure-Activity Relationships of Glycogen Phosphorylase Inhibitor FR258900 and Its Analogues: A Combined Synthetic, Enzyme Kinetics, and Computational Study (ChemPlusChem 11/2014)

ChemPlusChem ◽

10.1002/cplu.201402403 ◽

2014 ◽

Vol 79 (11) ◽

pp. 1535-1535

Author(s):

László Juhász ◽

Gergely Varga ◽

Andrea Sztankovics ◽

Ferenc Béke ◽

Tibor Docsa ◽

...

Keyword(s):

Enzyme Kinetics ◽

Glycogen Phosphorylase ◽

Computational Study ◽

Structure Activity Relationships ◽

Structure Activity ◽

Glycogen Phosphorylase Inhibitor

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Structure-Activity Relationships of Glycogen Phosphorylase Inhibitor FR258900 and Its Analogues: A Combined Synthetic, Enzyme Kinetics, and Computational Study

ChemPlusChem ◽

10.1002/cplu.201402302 ◽

2014 ◽

Vol 79 (11) ◽

pp. 1536-1536

Author(s):

László Juhász ◽

Gergely Varga ◽

Andrea Sztankovics ◽

Ferenc Béke ◽

Tibor Docsa ◽

...

Keyword(s):

Enzyme Kinetics ◽

Glycogen Phosphorylase ◽

Computational Study ◽

Structure Activity Relationships ◽

Structure Activity ◽

Glycogen Phosphorylase Inhibitor

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Structure-Activity Relationships of Glycogen Phosphorylase Inhibitor FR258900 and Its Analogues: A Combined Synthetic, Enzyme Kinetics, and Computational Study

ChemPlusChem ◽

10.1002/cplu.201402181 ◽

2014 ◽

Vol 79 (11) ◽

pp. 1558-1568 ◽

Cited By ~ 3

Author(s):

László Juhász ◽

Gergely Varga ◽

Andrea Sztankovics ◽

Ferenc Béke ◽

Tibor Docsa ◽

...

Keyword(s):

Enzyme Kinetics ◽

Glycogen Phosphorylase ◽

Computational Study ◽

Structure Activity Relationships ◽

Structure Activity ◽

Glycogen Phosphorylase Inhibitor

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Sourcing the affinity of flavonoids for the glycogen phosphorylase inhibitor site via crystallography, kinetics and QM/MM-PBSA binding studies: Comparison of chrysin and flavopiridol

Food and Chemical Toxicology ◽

10.1016/j.fct.2012.12.030 ◽

2013 ◽

Vol 61 ◽

pp. 14-27 ◽

Cited By ~ 16

Author(s):

Katerina E. Tsitsanou ◽

Joseph M. Hayes ◽

Maria Keramioti ◽

Michalis Mamais ◽

Nikos G. Oikonomakos ◽

...

Keyword(s):

Glycogen Phosphorylase ◽

Binding Studies ◽

Glycogen Phosphorylase Inhibitor

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glycogen phosphorylase inhibitor
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Glycogen phosphorylase inhibitor, 2,3‐bis[(2E)‐3‐(4‐hydroxyphenyl)prop‐2‐enamido] butanedioic acid (BF142), improves baseline insulin secretion of MIN6 insulinoma cells

Synthetic flavonoid derivatives targeting the glycogen phosphorylase inhibitor site: QM/MM-PBSA motivated synthesis of substituted 5,7-dihydroxyflavones, crystallography, in vitro kinetics and ex-vivo cellular experiments reveal novel potent inhibitors

Effects of Intracerebroventricular Glycogen Phosphorylase Inhibitor CP-316,819 Infusion on Hypothalamic Glycogen Content and Metabolic Neuron AMPK Activity and Neurotransmitter Expression in Male Rat

Multiscale time-resolved fluorescence study of a glycogen phosphorylase inhibitor combined with quantum chemistry calculations

Novel Liver-targeted conjugates of Glycogen Phosphorylase Inhibitor PSN-357 for the Treatment of Diabetes: Design, Synthesis, Pharmacokinetic and Pharmacological Evaluations

Insulin Sensitivity is Modified by a Glycogen Phosphorylase Inhibitor: Glucopyranosylidene-Spiro-Thiohydantoin in Streptozotocin-Induced Diabetic Rats

Cover Picture: Structure-Activity Relationships of Glycogen Phosphorylase Inhibitor FR258900 and Its Analogues: A Combined Synthetic, Enzyme Kinetics, and Computational Study (ChemPlusChem 11/2014)

Structure-Activity Relationships of Glycogen Phosphorylase Inhibitor FR258900 and Its Analogues: A Combined Synthetic, Enzyme Kinetics, and Computational Study

Structure-Activity Relationships of Glycogen Phosphorylase Inhibitor FR258900 and Its Analogues: A Combined Synthetic, Enzyme Kinetics, and Computational Study

Sourcing the affinity of flavonoids for the glycogen phosphorylase inhibitor site via crystallography, kinetics and QM/MM-PBSA binding studies: Comparison of chrysin and flavopiridol

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glycogen phosphorylase inhibitorRecently Published Documents

TOTAL DOCUMENTS

H-INDEX

Glycogen phosphorylase inhibitor, 2,3‐bis[(2E)‐3‐(4‐hydroxyphenyl)prop‐2‐enamido] butanedioic acid (BF142), improves baseline insulin secretion of MIN6 insulinoma cells

Synthetic flavonoid derivatives targeting the glycogen phosphorylase inhibitor site: QM/MM-PBSA motivated synthesis of substituted 5,7-dihydroxyflavones, crystallography, in vitro kinetics and ex-vivo cellular experiments reveal novel potent inhibitors

Effects of Intracerebroventricular Glycogen Phosphorylase Inhibitor CP-316,819 Infusion on Hypothalamic Glycogen Content and Metabolic Neuron AMPK Activity and Neurotransmitter Expression in Male Rat

Multiscale time-resolved fluorescence study of a glycogen phosphorylase inhibitor combined with quantum chemistry calculations

Novel Liver-targeted conjugates of Glycogen Phosphorylase Inhibitor PSN-357 for the Treatment of Diabetes: Design, Synthesis, Pharmacokinetic and Pharmacological Evaluations

Insulin Sensitivity is Modified by a Glycogen Phosphorylase Inhibitor: Glucopyranosylidene-Spiro-Thiohydantoin in Streptozotocin-Induced Diabetic Rats

Cover Picture: Structure-Activity Relationships of Glycogen Phosphorylase Inhibitor FR258900 and Its Analogues: A Combined Synthetic, Enzyme Kinetics, and Computational Study (ChemPlusChem 11/2014)

Structure-Activity Relationships of Glycogen Phosphorylase Inhibitor FR258900 and Its Analogues: A Combined Synthetic, Enzyme Kinetics, and Computational Study

Structure-Activity Relationships of Glycogen Phosphorylase Inhibitor FR258900 and Its Analogues: A Combined Synthetic, Enzyme Kinetics, and Computational Study

Sourcing the affinity of flavonoids for the glycogen phosphorylase inhibitor site via crystallography, kinetics and QM/MM-PBSA binding studies: Comparison of chrysin and flavopiridol

glycogen phosphorylase inhibitor
Recently Published Documents