benzhydryl piperazine
Recently Published Documents

TOTAL DOCUMENTS

10
(FIVE YEARS 0)

H-INDEX

4
(FIVE YEARS 0)
Latest Documents Most Cited Documents Contributed Authors Related Sources Related Keywords

scholarly journals (4-(Bis(4-Fluorophenyl)Methyl)Piperazin-1-yl)(Cyclohexyl)Methanone Hydrochloride (LDK1229): A New Cannabinoid CB1Receptor Inverse Agonist from the Class of Benzhydryl Piperazine Analogs

2014 ◽  
Vol 87 (2) ◽  
pp. 197-206 ◽  
Author(s):  
Mariam M. Mahmoud ◽  
Teresa Olszewska ◽  
Hui Liu ◽  
Derek M. Shore ◽  
Dow P. Hurst ◽  
...  
Keyword(s):  
Inverse Agonist ◽  
Benzhydryl Piperazine

Synthesis of 1-benzhydryl piperazine derivatives and evaluation of their ACE inhibition and antimicrobial activities

2014 ◽  
Vol 23 (6) ◽  
pp. 3207-3219 ◽  
Author(s):  
Amlipur Santhoshi ◽  
Singam Naveen Kumar ◽  
Pombala Sujitha ◽  
Yedla Poornachandra ◽  
Partha Sarathi Sadhu ◽  
...  
Keyword(s):  
Ace Inhibition ◽  
Antimicrobial Activities ◽  
Piperazine Derivatives ◽  
Benzhydryl Piperazine

scholarly journals Synthesis and antimicrobial studies of novel 1-benzhydryl-piperazine sulfonamide and carboxamide derivatives

2008 ◽  
Vol 23 (4) ◽  
pp. 462-469 ◽  
Author(s):  
C. S. Ananda Kumar ◽  
K. Vinaya ◽  
J. Narendra Sharath Chandra ◽  
N. R. Thimmegowda ◽  
S. B. Benaka Prasad ◽  
...  
Keyword(s):  
Antimicrobial Studies ◽  
Benzhydryl Piperazine

Synthesis and Crystal Structure of 1-Benzenesulfonyl-4-benzhydryl-piperazine

2007 ◽  
Vol 469 (1) ◽  
pp. 111-119 ◽  
Author(s):  
C. S. Ananda Kumar ◽  
S. B. Benaka Prasad ◽  
N. R. Thimmegowda ◽  
K. S. Rangappa ◽  
S. Chandrappa ◽  
...  
Keyword(s):  
Crystal Structure ◽  
Synthesis And Crystal Structure ◽  
Benzhydryl Piperazine

Synthesis and evaluation of novel β-lactam inhibitors of human leukocyte elastase

2001 ◽  
Vol 79 (4) ◽  
pp. 377-387 ◽  
Author(s):  
K P Koteva ◽  
André M Cantin ◽  
W A Neugebauer ◽  
E Escher
Keyword(s):  
Serine Protease ◽  
Protease Inhibitors ◽  
Neutrophil Elastase ◽  
Human Leukocyte ◽  
Leukocyte Elastase ◽  
Piperazine Derivatives ◽  
Structure Activity ◽  
Human Leukocyte Elastase ◽  
Benzhydryl Piperazine ◽  
Derivatives Of

A series of β-lactam derivatives were synthesized and tested to determine the structure-activity relationship for inhibition of human leukocyte elastase (HLE), a serine protease involved in several degenerative lung and tissue diseases. The most potent IC50 values were obtained with neutral hydrophobic 7α-methoxy cephalosporanic acid derivatives. Tryptophanyl-9-fluorenylmethyl ester and N-benzhydryl piperazine derivatives of 7α-methoxy cephalosporanic acid represent two novel HLE inhibitors, with length of action persisting beyond 24 h.Key words: β-lactams, neutrophil elastase, protease inhibitors, peptides.

Acid—base equilibria of some benzhydryl piperazine derivatives

1976 ◽  
Vol 86 ◽  
pp. 185-194 ◽  
Author(s):  
M.R Smyth ◽  
W.Franklin Smyth ◽  
R.F Palmer ◽  
J.M Clifford
Keyword(s):  
Acid Base ◽  
Piperazine Derivatives ◽  
Benzhydryl Piperazine
Load More ...
Sign in / Sign up

Export Citation Format

Share Document