glycine transporter 1 inhibitor Latest Research Papers

P.0526 Effects of the novel glycine transporter-1 inhibitor bi 425809 on mouse electroencephalography and auditory event-related potential biomarkers related to schizophrenia

European Neuropsychopharmacology ◽

10.1016/j.euroneuro.2021.10.497 ◽

2021 ◽

Vol 53 ◽

pp. S387-S388

Author(s):

N. Schuelert ◽

C. Dorner-Ciossek ◽

H. Rosenbrock

Keyword(s):

Event Related Potential ◽

The Novel ◽

Auditory Event ◽

Glycine Transporter 1 ◽

Glycine Transporter ◽

Potential Biomarkers ◽

Glycine Transporter 1 Inhibitor

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Effects of Cytochrome P450 3A4 Induction and Inhibition on the Pharmacokinetics of BI 425809, a Novel Glycine Transporter 1 Inhibitor

European Journal of Drug Metabolism and Pharmacokinetics ◽

10.1007/s13318-021-00723-y ◽

2021 ◽

Author(s):

Michael Desch ◽

Glen Wunderlich ◽

Markus Goettel ◽

Sophia Goetz ◽

Karl-Heinz Liesenfeld ◽

...

Keyword(s):

Cytochrome P450 ◽

Cytochrome P450 3A4 ◽

Glycine Transporter 1 ◽

Glycine Transporter ◽

Glycine Transporter 1 Inhibitor

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Effect of the glycine transporter 1 inhibitor ALX-5407 on dyskinesia, psychosis-like behaviours and parkinsonism in the MPTP-lesioned marmoset

European Journal of Pharmacology ◽

10.1016/j.ejphar.2021.174452 ◽

2021 ◽

pp. 174452

Author(s):

Imane Frouni ◽

Sébastien Belliveau ◽

Shawn Maddaford ◽

Stephen G. Nuara ◽

Jim C. Gourdon ◽

...

Keyword(s):

Glycine Transporter 1 ◽

Glycine Transporter ◽

Glycine Transporter 1 Inhibitor

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P.555 Effects of the glycine transporter-1 inhibitor bitopertin on rodent electroencephalography and auditory event-related potential biomarkers related to schizophrenia

European Neuropsychopharmacology ◽

10.1016/j.euroneuro.2019.09.558 ◽

2019 ◽

Vol 29 ◽

pp. S390

Author(s):

P. Voehringer ◽

N. Schuelert ◽

A. Plano ◽

C. Dorner-Ciossek ◽

H. Rosenbrock

Keyword(s):

Event Related Potential ◽

Auditory Event ◽

Glycine Transporter 1 ◽

Glycine Transporter ◽

Potential Biomarkers ◽

Glycine Transporter 1 Inhibitor

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Dose-Related Target Occupancy and Effects on Circuitry, Behavior, and Neuroplasticity of the Glycine Transporter-1 Inhibitor PF-03463275 in Healthy and Schizophrenia Subjects

Biological Psychiatry ◽

10.1016/j.biopsych.2017.12.019 ◽

2018 ◽

Vol 84 (6) ◽

pp. 413-421 ◽

Cited By ~ 18

Author(s):

Deepak Cyril D’Souza ◽

Richard E. Carson ◽

Naomi Driesen ◽

Jason Johannesen ◽

Mohini Ranganathan ◽

...

Keyword(s):

Related Target ◽

Glycine Transporter 1 ◽

Glycine Transporter ◽

Glycine Transporter 1 Inhibitor

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Safety, Tolerability and Pharmacokinetics of Oral BI 425809, a Glycine Transporter 1 Inhibitor, in Healthy Male Volunteers: A Partially Randomised, Single-Blind, Placebo-Controlled, First-in-Human Study

European Journal of Drug Metabolism and Pharmacokinetics ◽

10.1007/s13318-017-0440-z ◽

2017 ◽

Vol 43 (2) ◽

pp. 239-249 ◽

Cited By ~ 7

Author(s):

Viktoria Moschetti ◽

Michael Desch ◽

Sophia Goetz ◽

Karl-Heinz Liesenfeld ◽

Holger Rosenbrock ◽

...

Keyword(s):

Human Study ◽

Healthy Male ◽

Glycine Transporter 1 ◽

Glycine Transporter ◽

Healthy Male Volunteers ◽

Male Volunteers ◽

Single Blind ◽

Glycine Transporter 1 Inhibitor

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P4-010: Improving Cognitive Function in Rodents Via Increasing Glycine Levels in Brain by the Novel Glycine Transporter-1 Inhibitor BI 425809

Alzheimer s & Dementia ◽

10.1016/j.jalz.2016.06.2099 ◽

2016 ◽

Vol 12 ◽

pp. P1018-P1018 ◽

Cited By ~ 3

Author(s):

Holger Rosenbrock ◽

Riccardo Giovannini ◽

Bernhard Schmid ◽

Gert Kramer ◽

Roberto Arban ◽

...

Keyword(s):

Cognitive Function ◽

The Novel ◽

Glycine Transporter 1 ◽

Glycine Transporter ◽

Glycine Transporter 1 Inhibitor

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Identification of 1-Methyl-N-(propan-2-yl)-N-({2-[4-(trifluoromethoxy)phenyl]pyridin-4-yl}methyl)-1H-imidazole-4-carboxamide as a Potent and Orally Available Glycine Transporter 1 Inhibitor

Chemical and Pharmaceutical Bulletin ◽

10.1248/cpb.c16-00610 ◽

2016 ◽

Vol 64 (11) ◽

pp. 1630-1640 ◽

Cited By ~ 1

Author(s):

Shuji Yamamoto ◽

Hiroshi Ohta ◽

Kumi Abe ◽

Daiji Kambe ◽

Naohiro Tsukiyama ◽

...

Keyword(s):

Glycine Transporter 1 ◽

Glycine Transporter ◽

Glycine Transporter 1 Inhibitor

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Discovery of 3-Chloro-N-{(S)-[3-(1-ethyl-1H-pyrazol-4-yl)phenyl][(2S)-piperidine-2-yl]methyl}-4-(trifluoromethyl)pyridine-2-carboxamide as a Potent Glycine Transporter 1 Inhibitor

Chemical and Pharmaceutical Bulletin ◽

10.1248/cpb.c16-00314 ◽

2016 ◽

Vol 64 (9) ◽

pp. 1321-1337

Author(s):

Shuji Yamamoto ◽

Tsuyoshi Shibata ◽

Kumi Abe ◽

Koji Oda ◽

Takeshi Aoki ◽

...

Keyword(s):

Glycine Transporter 1 ◽

Glycine Transporter ◽

Glycine Transporter 1 Inhibitor

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Efficacy of a glycine transporter 1 inhibitor TASP0315003 in animal models of cognitive dysfunction and negative symptoms of schizophrenia

Psychopharmacology ◽

10.1007/s00213-015-3920-3 ◽

2015 ◽

Vol 232 (15) ◽

pp. 2849-2861 ◽

Cited By ~ 12

Author(s):

Shigeyuki Chaki ◽

Toshiharu Shimazaki ◽

Jun-ichi Karasawa ◽

Takeshi Aoki ◽

Ayaka Kaku ◽

...

Keyword(s):

Animal Models ◽

Cognitive Dysfunction ◽

Negative Symptoms ◽

Glycine Transporter 1 ◽

Glycine Transporter ◽

Glycine Transporter 1 Inhibitor

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glycine transporter 1 inhibitor
Recently Published Documents

TOTAL DOCUMENTS

H-INDEX

P.0526 Effects of the novel glycine transporter-1 inhibitor bi 425809 on mouse electroencephalography and auditory event-related potential biomarkers related to schizophrenia

Effects of Cytochrome P450 3A4 Induction and Inhibition on the Pharmacokinetics of BI 425809, a Novel Glycine Transporter 1 Inhibitor

Effect of the glycine transporter 1 inhibitor ALX-5407 on dyskinesia, psychosis-like behaviours and parkinsonism in the MPTP-lesioned marmoset

P.555 Effects of the glycine transporter-1 inhibitor bitopertin on rodent electroencephalography and auditory event-related potential biomarkers related to schizophrenia

Dose-Related Target Occupancy and Effects on Circuitry, Behavior, and Neuroplasticity of the Glycine Transporter-1 Inhibitor PF-03463275 in Healthy and Schizophrenia Subjects

Safety, Tolerability and Pharmacokinetics of Oral BI 425809, a Glycine Transporter 1 Inhibitor, in Healthy Male Volunteers: A Partially Randomised, Single-Blind, Placebo-Controlled, First-in-Human Study

P4-010: Improving Cognitive Function in Rodents Via Increasing Glycine Levels in Brain by the Novel Glycine Transporter-1 Inhibitor BI 425809

Identification of 1-Methyl-N-(propan-2-yl)-N-({2-[4-(trifluoromethoxy)phenyl]pyridin-4-yl}methyl)-1H-imidazole-4-carboxamide as a Potent and Orally Available Glycine Transporter 1 Inhibitor

Discovery of 3-Chloro-N-{(S)-[3-(1-ethyl-1H-pyrazol-4-yl)phenyl][(2S)-piperidine-2-yl]methyl}-4-(trifluoromethyl)pyridine-2-carboxamide as a Potent Glycine Transporter 1 Inhibitor

Efficacy of a glycine transporter 1 inhibitor TASP0315003 in animal models of cognitive dysfunction and negative symptoms of schizophrenia

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glycine transporter 1 inhibitorRecently Published Documents

TOTAL DOCUMENTS

H-INDEX

P.0526 Effects of the novel glycine transporter-1 inhibitor bi 425809 on mouse electroencephalography and auditory event-related potential biomarkers related to schizophrenia

Effects of Cytochrome P450 3A4 Induction and Inhibition on the Pharmacokinetics of BI 425809, a Novel Glycine Transporter 1 Inhibitor

Effect of the glycine transporter 1 inhibitor ALX-5407 on dyskinesia, psychosis-like behaviours and parkinsonism in the MPTP-lesioned marmoset

P.555 Effects of the glycine transporter-1 inhibitor bitopertin on rodent electroencephalography and auditory event-related potential biomarkers related to schizophrenia

Dose-Related Target Occupancy and Effects on Circuitry, Behavior, and Neuroplasticity of the Glycine Transporter-1 Inhibitor PF-03463275 in Healthy and Schizophrenia Subjects

Safety, Tolerability and Pharmacokinetics of Oral BI 425809, a Glycine Transporter 1 Inhibitor, in Healthy Male Volunteers: A Partially Randomised, Single-Blind, Placebo-Controlled, First-in-Human Study

P4-010: Improving Cognitive Function in Rodents Via Increasing Glycine Levels in Brain by the Novel Glycine Transporter-1 Inhibitor BI 425809

Identification of 1-Methyl-N-(propan-2-yl)-N-({2-[4-(trifluoromethoxy)phenyl]pyridin-4-yl}methyl)-1H-imidazole-4-carboxamide as a Potent and Orally Available Glycine Transporter 1 Inhibitor

Discovery of 3-Chloro-N-{(S)-[3-(1-ethyl-1H-pyrazol-4-yl)phenyl][(2S)-piperidine-2-yl]methyl}-4-(trifluoromethyl)pyridine-2-carboxamide as a Potent Glycine Transporter 1 Inhibitor

Efficacy of a glycine transporter 1 inhibitor TASP0315003 in animal models of cognitive dysfunction and negative symptoms of schizophrenia

glycine transporter 1 inhibitor
Recently Published Documents