Structure-Activity Relationship (SAR) Studies on Oxazolidinone Antibacterial Agents. 2. Relationship between Lipophilicity and Antibacterial Activity in 5-Thiocarbonyl Oxazolidinones.

2001 ◽  
Vol 49 (4) ◽  
pp. 353-360 ◽  
Author(s):  
Ryukou TOKUYAMA ◽  
Yoshiei TAKAHASHI ◽  
Yayoi TOMITA ◽  
Masatoshi TSUBOUCHI ◽  
Toshihiko YOSHIDA ◽  
...  
2001 ◽  
Vol 49 (4) ◽  
pp. 347-352 ◽  
Author(s):  
Ryukou TOKUYAMA ◽  
Yoshiei TAKAHASHI ◽  
Yayoi TOMITA ◽  
Tomio SUZUKI ◽  
Toshihiko YOSHIDA ◽  
...  

2001 ◽  
Vol 49 (4) ◽  
pp. 361-367 ◽  
Author(s):  
Ryukou TOKUYAMA ◽  
Yoshiei TAKAHASHI ◽  
Yayoi TOMITA ◽  
Masatoshi TSUBOUCHI ◽  
Nobuhiko IWASAKI ◽  
...  

ChemInform ◽  
2010 ◽  
Vol 32 (39) ◽  
pp. no-no
Author(s):  
Ryukou Tokuyama ◽  
Yoshiei Takahashi ◽  
Yayoi Tomita ◽  
Tomio Suzuki ◽  
Toshihiko Yoshida ◽  
...  

2020 ◽  
Vol 24 (8) ◽  
pp. 817-854
Author(s):  
Anil Kumar ◽  
Nishtha Saxena ◽  
Arti Mehrotra ◽  
Nivedita Srivastava

Quinolone derivatives have attracted considerable attention due to their medicinal properties. This review covers many synthetic routes of quinolones preparation with their antibacterial properties. Detailed study with structure-activity relationship among quinolone derivatives will be helpful in designing new drugs in this field.


2012 ◽  
Vol 9 (3) ◽  
pp. 329-335 ◽  
Author(s):  
Surajit Kumar Ghosh ◽  
Ashmita Saha ◽  
Bornali Hazarika ◽  
Udaya Pratap Singh ◽  
Hans Raj Bhat ◽  
...  

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