Structure-Activity Relationship (SAR) Studies on Oxazolidinone Antibacterial Agents. 1. Conversion of 5-Substituent on Oxazolidinone.

Ryukou TOKUYAMA; Yoshiei TAKAHASHI; Yayoi TOMITA; Tomio SUZUKI; Toshihiko YOSHIDA; Nobuhiko IWASAKI; Noriyuki KADO; Eiichi OKEZAKI; Osamu NAGATA

doi:10.1248/cpb.49.347

Structure-Activity Relationship (SAR) Studies on Oxazolidinone Antibacterial Agents. 1. Conversion of 5-Substituent on Oxazolidinone.

Chemical and Pharmaceutical Bulletin ◽

10.1248/cpb.49.347 ◽

2001 ◽

Vol 49 (4) ◽

pp. 347-352 ◽

Cited By ~ 26

Author(s):

Ryukou TOKUYAMA ◽

Yoshiei TAKAHASHI ◽

Yayoi TOMITA ◽

Tomio SUZUKI ◽

Toshihiko YOSHIDA ◽

...

Keyword(s):

Antibacterial Agents ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Sar Studies ◽

Structure Activity

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Structure-Activity Relationship (SAR) Studies on Oxazolidinone Antibacterial Agents. 2. Relationship between Lipophilicity and Antibacterial Activity in 5-Thiocarbonyl Oxazolidinones.

Chemical and Pharmaceutical Bulletin ◽

10.1248/cpb.49.353 ◽

2001 ◽

Vol 49 (4) ◽

pp. 353-360 ◽

Cited By ~ 35

Author(s):

Ryukou TOKUYAMA ◽

Yoshiei TAKAHASHI ◽

Yayoi TOMITA ◽

Masatoshi TSUBOUCHI ◽

Toshihiko YOSHIDA ◽

...

Keyword(s):

Antibacterial Activity ◽

Antibacterial Agents ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Sar Studies ◽

Structure Activity

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ChemInform Abstract: Structure-Activity Relationship (SAR) Studies on Oxazolidinone Antibacterial Agents. Part 3. Synthesis and Evaluation of 5-Thiocarbamate Oxazolidinones.

ChemInform ◽

10.1002/chin.200139132 ◽

2010 ◽

Vol 32 (39) ◽

pp. no-no

Author(s):

Ryukou Tokuyama ◽

Yoshiei Takahashi ◽

Yayoi Tomita ◽

Masatoshi Tsubouchi ◽

Nobuhiko Iwasaki ◽

...

Keyword(s):

Antibacterial Agents ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Sar Studies ◽

Structure Activity ◽

Abstract Structure

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Structure-Activity Relationship (SAR) Studies on Oxazolidinone Antibacterial Agents. 3. Synthesis and Evaluation of 5-Thiocarbamate Oxazolidinones.

Chemical and Pharmaceutical Bulletin ◽

10.1248/cpb.49.361 ◽

2001 ◽

Vol 49 (4) ◽

pp. 361-367 ◽

Cited By ~ 25

Author(s):

Ryukou TOKUYAMA ◽

Yoshiei TAKAHASHI ◽

Yayoi TOMITA ◽

Masatoshi TSUBOUCHI ◽

Nobuhiko IWASAKI ◽

...

Keyword(s):

Antibacterial Agents ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Sar Studies ◽

Structure Activity

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ChemInform Abstract: Structure-Activity Relationship (SAR) Studies on Oxazolidinone Antibacterial Agents. Part 2. Relationship Between Lipophilicity and Antibacterial Activity in 5-Thiocarbonyl Oxazolidinones.

ChemInform ◽

10.1002/chin.200139131 ◽

2010 ◽

Vol 32 (39) ◽

pp. no-no

Author(s):

Ryukou Tokuyama ◽

Yoshiei Takahashi ◽

Yayoi Tomita ◽

Masatoshi Tsubouchi ◽

Toshihiko Yoshida ◽

...

Keyword(s):

Antibacterial Activity ◽

Antibacterial Agents ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Sar Studies ◽

Structure Activity ◽

Abstract Structure

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ChemInform Abstract: Structure-Activity Relationship (SAR) Studies on Oxazolidinone Antibacterial Agents. Part 1. Conversion of 5-Substituent on Oxazolidinone.

ChemInform ◽

10.1002/chin.200139130 ◽

2010 ◽

Vol 32 (39) ◽

pp. no-no

Author(s):

Ryukou Tokuyama ◽

Yoshiei Takahashi ◽

Yayoi Tomita ◽

Tomio Suzuki ◽

Toshihiko Yoshida ◽

...

Keyword(s):

Antibacterial Agents ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Sar Studies ◽

Structure Activity ◽

Abstract Structure

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Structure Activity Relationship of Arylidene Pyrrolo and Pyrido [2,1-b] Quinazolones as Cytotoxic Agents: Synthesis, SAR Studies, Biological Evaluation and Docking Studies

Medicinal Chemistry ◽

10.2174/1573406411309050003 ◽

2013 ◽

Vol 9 (5) ◽

pp. 642-650 ◽

Cited By ~ 3

Author(s):

Veenu Mangla ◽

Kunal Nepali ◽

Gagandip Singh ◽

Jagjeet Singh ◽

Santosh Guru ◽

...

Keyword(s):

Structure Activity Relationship ◽

Docking Studies ◽

Biological Evaluation ◽

Cytotoxic Agents ◽

Activity Relationship ◽

Sar Studies ◽

Structure Activity ◽

Relationship Of

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Design, synthesis and structure–activity relationship (SAR) studies of imidazo[4,5-b]pyridine derived purine isosteres and their potential as cytotoxic agents

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2014.10.037 ◽

2015 ◽

Vol 89 ◽

pp. 21-31 ◽

Cited By ~ 26

Author(s):

Ayyiliath M. Sajith ◽

K.K. Abdul Khader ◽

Nithin Joshi ◽

Manchala Nageswar Reddy ◽

M. Syed Ali Padusha ◽

...

Keyword(s):

Structure Activity Relationship ◽

Cytotoxic Agents ◽

Activity Relationship ◽

Design Synthesis ◽

Sar Studies ◽

Structure Activity

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Structure-activity relationship for antibacterial action of phenolic and aromatic nitro compounds. An attempt at systematic identification of new antibacterial agents.

Chemical and Pharmaceutical Bulletin ◽

10.1248/cpb.33.2821 ◽

1985 ◽

Vol 33 (7) ◽

pp. 2821-2831 ◽

Cited By ~ 5

Author(s):

SETSUKO OIKAWA ◽

MINORU TSUDA ◽

KIKUTAROU ENDOU ◽

HIDEKO ABE ◽

MAYUMI MATSUOKA ◽

...

Keyword(s):

Antibacterial Agents ◽

Structure Activity Relationship ◽

Nitro Compounds ◽

Antibacterial Action ◽

Activity Relationship ◽

Aromatic Nitro Compounds ◽

Structure Activity ◽

Aromatic Nitro ◽

Systematic Identification

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Potent α-amino-β-lactam carbamic acid ester as NAAA inhibitors. Synthesis and structure–activity relationship (SAR) studies

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2016.01.046 ◽

2016 ◽

Vol 111 ◽

pp. 138-159 ◽

Cited By ~ 17

Author(s):

Andrea Nuzzi ◽

Annalisa Fiasella ◽

Jose Antonio Ortega ◽

Chiara Pagliuca ◽

Stefano Ponzano ◽

...

Keyword(s):

Acid Ester ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Carbamic Acid ◽

Sar Studies ◽

Structure Activity

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Structure–activity relationship of novel low-generation dendrimers for gene delivery

Organic & Biomolecular Chemistry ◽

10.1039/c8ob01767k ◽

2018 ◽

Vol 16 (42) ◽

pp. 7833-7842 ◽

Cited By ~ 4

Author(s):

Yong-Guang Gao ◽

Xiao Lin ◽

Kai Dang ◽

Shan-Feng Jiang ◽

Ye Tian ◽

...

Keyword(s):

Gene Delivery ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Sar Studies ◽

Structure Activity ◽

Gene Vectors ◽

Relationship Of

Structure–activity relationship (SAR) studies are very critical to design ideal gene vectors for gene delivery.

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