Total Syntheses of the Non-Peptide Bradykinin B1 Receptor Antagonist Velutinol A and Its Analogs, seco-Pregnanes with a Cage-Like Moiety

2019 ◽  
Vol 92 (9) ◽  
pp. 1474-1494
Author(s):  
Minoru Tamiya ◽  
Nobuhisa Isaka ◽  
Takaaki Kitazawa ◽  
Atsushi Hasegawa ◽  
Kazuya Ishizawa ◽  
...  
Keyword(s):  
Receptor Antagonist ◽  
Total Syntheses ◽  
B1 Receptor ◽  
Bradykinin B1 Receptor

scholarly journals The bradykinin B1 receptor antagonist R-954 inhibits Ehrlich tumor growth in rodents

Peptides ◽  
2011 ◽  
Vol 32 (9) ◽  
pp. 1849-1854 ◽  
Author(s):  
Patricia Dias Fernandes ◽  
Niele de Matos Gomes ◽  
Pierre Sirois
Keyword(s):  
Tumor Growth ◽  
Receptor Antagonist ◽  
Ehrlich Tumor ◽  
B1 Receptor ◽  
Bradykinin B1 Receptor

Identification of a Nonpeptidic and Conformationally Restricted Bradykinin B1 Receptor Antagonist with Anti-Inflammatory Activity

2007 ◽  
Vol 50 (4) ◽  
pp. 607-610 ◽  
Author(s):  
Derin C. D'Amico ◽  
Toshi Aya ◽  
Jason Human ◽  
Christopher Fotsch ◽  
Jian Jeffrey Chen ◽  
...  
Keyword(s):  
Receptor Antagonist ◽  
Inflammatory Activity ◽  
Conformationally Restricted ◽  
B1 Receptor ◽  
Bradykinin B1 Receptor ◽  
Anti Inflammatory

scholarly journals The bradykinin B1 receptor antagonist BI113823 reverses inflammatory hyperalgesia by desensitization of peripheral and spinal neurons

2014 ◽  
Vol 19 (1) ◽  
pp. 132-142 ◽  
Author(s):  
N. Schuelert ◽  
S. Just ◽  
L. Corradini ◽  
R. Kuelzer ◽  
C. Bernloehr ◽  
...  
Keyword(s):  
Receptor Antagonist ◽  
Spinal Neurons ◽  
Inflammatory Hyperalgesia ◽  
B1 Receptor ◽  
Bradykinin B1 Receptor

An Orally Active Bradykinin B1 Receptor Antagonist Engineered as a Bifunctional Chimera of Sunflower Trypsin Inhibitor

2016 ◽  
Vol 60 (1) ◽  
pp. 504-510 ◽  
Author(s):  
Yibo Qiu ◽  
Misako Taichi ◽  
Na Wei ◽  
Huan Yang ◽  
Kathy Qian Luo ◽  
...  
Keyword(s):  
Receptor Antagonist ◽  
Trypsin Inhibitor ◽  
B1 Receptor ◽  
Bradykinin B1 Receptor ◽  
Orally Active

A Concise Total Synthesis of the Non-peptide Bradykinin B1 Receptor Antagonist Velutinol A

2011 ◽  
Vol 2012 (4) ◽  
pp. 665-668 ◽  
Author(s):  
Nobuhisa Isaka ◽  
Minoru Tamiya ◽  
Atsushi Hasegawa ◽  
Masaji Ishiguro
Keyword(s):  
Total Synthesis ◽  
Receptor Antagonist ◽  
B1 Receptor ◽  
Bradykinin B1 Receptor

DesArg9D-Arg[Hyp3,Thi5,D-Tic7,Oic8]bradykinin (desArg10-[Hoe140]) is a bradykinin B1 receptor antagonist

1991 ◽  
Vol 205 (2) ◽  
pp. 217-218 ◽  
Author(s):  
Klaus Wirth ◽  
Gerhard Breipohl ◽  
Jens Stechl ◽  
Jochen Knolle ◽  
Stephan Henke ◽  
...  
Keyword(s):  
Receptor Antagonist ◽  
B1 Receptor ◽  
Bradykinin B1 Receptor
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