Identification of a Nonpeptidic and Conformationally Restricted Bradykinin B1 Receptor Antagonist with Anti-Inflammatory Activity

2007 ◽  
Vol 50 (4) ◽  
pp. 607-610 ◽  
Author(s):  
Derin C. D'Amico ◽  
Toshi Aya ◽  
Jason Human ◽  
Christopher Fotsch ◽  
Jian Jeffrey Chen ◽  
...  
Keyword(s):  
Receptor Antagonist ◽  
Inflammatory Activity ◽  
Conformationally Restricted ◽  
B1 Receptor ◽  
Bradykinin B1 Receptor ◽  
Anti Inflammatory

scholarly journals The bradykinin B1 receptor antagonist R-954 inhibits Ehrlich tumor growth in rodents

Peptides ◽  
2011 ◽  
Vol 32 (9) ◽  
pp. 1849-1854 ◽  
Author(s):  
Patricia Dias Fernandes ◽  
Niele de Matos Gomes ◽  
Pierre Sirois
Keyword(s):  
Tumor Growth ◽  
Receptor Antagonist ◽  
Ehrlich Tumor ◽  
B1 Receptor ◽  
Bradykinin B1 Receptor

scholarly journals The bradykinin B1 receptor antagonist BI113823 reverses inflammatory hyperalgesia by desensitization of peripheral and spinal neurons

2014 ◽  
Vol 19 (1) ◽  
pp. 132-142 ◽  
Author(s):  
N. Schuelert ◽  
S. Just ◽  
L. Corradini ◽  
R. Kuelzer ◽  
C. Bernloehr ◽  
...  
Keyword(s):  
Receptor Antagonist ◽  
Spinal Neurons ◽  
Inflammatory Hyperalgesia ◽  
B1 Receptor ◽  
Bradykinin B1 Receptor

An Orally Active Bradykinin B1 Receptor Antagonist Engineered as a Bifunctional Chimera of Sunflower Trypsin Inhibitor

2016 ◽  
Vol 60 (1) ◽  
pp. 504-510 ◽  
Author(s):  
Yibo Qiu ◽  
Misako Taichi ◽  
Na Wei ◽  
Huan Yang ◽  
Kathy Qian Luo ◽  
...  
Keyword(s):  
Receptor Antagonist ◽  
Trypsin Inhibitor ◽  
B1 Receptor ◽  
Bradykinin B1 Receptor ◽  
Orally Active

Pharmacological profile of CR3465, a new leukotriene CysLT1 receptor antagonist with broad anti-inflammatory activity

2004 ◽  
Vol 504 (3) ◽  
pp. 223-233 ◽  
Author(s):  
Flora Ferrari ◽  
Laura Mennuni ◽  
Gianfranco Caselli ◽  
Tiziano Zanelli ◽  
Francesco Makovec
Keyword(s):  
Receptor Antagonist ◽  
Inflammatory Activity ◽  
Pharmacological Profile ◽  
Anti Inflammatory

Anti-inflammatory activity of the leukotriene B4 receptor antagonist, SC-41930, in colitic cotton-top tamarins

1994 ◽  
Vol 41 (S2) ◽  
pp. C254-C255 ◽  
Author(s):  
N. Clapp ◽  
M. Henke ◽  
R. Hansard ◽  
R. Carson ◽  
D. Widomski ◽  
...  
Keyword(s):  
Receptor Antagonist ◽  
Leukotriene B4 ◽  
Inflammatory Activity ◽  
Anti Inflammatory ◽  
Leukotriene B4 Receptor
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