Strategy for the Identification of GPR23/LPA4 Receptor Agonists and Inverse Agonists

Soo Hang Wong; Rommel Mallari; Melissa Graham; Larissa Atangan; Shu-Chen Lu; Xiaoning Zhao; Wei Gu; Paul H. Lee

doi:10.1089/adt.2009.0261

Strategy for the Identification of GPR23/LPA4 Receptor Agonists and Inverse Agonists

Assay and Drug Development Technologies ◽

10.1089/adt.2009.0261 ◽

2010 ◽

Vol 8 (4) ◽

pp. 459-470 ◽

Cited By ~ 5

Author(s):

Soo Hang Wong ◽

Rommel Mallari ◽

Melissa Graham ◽

Larissa Atangan ◽

Shu-Chen Lu ◽

...

Keyword(s):

Inverse Agonists ◽

Receptor Agonists

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”Audiogenic seizures in DBA/2 mice discriminate sensitivity between low efficacy benzodiazepine receptor agonists and inverse agonists,”

Life Sciences ◽

10.1016/0024-3205(83)90731-2 ◽

1983 ◽

Vol 33 (17) ◽

pp. 1731

Keyword(s):

Benzodiazepine Receptor ◽

Audiogenic Seizures ◽

Inverse Agonists ◽

Receptor Agonists

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β-Carbolines characterized as benzodiazepine receptor agonists and inverse agonists produce bi-directional changes in palatable food consumption

Brain Research Bulletin ◽

10.1016/0361-9230(86)90194-2 ◽

1986 ◽

Vol 17 (5) ◽

pp. 627-637 ◽

Cited By ~ 18

Author(s):

Steven J. Cooper

Keyword(s):

Food Consumption ◽

Benzodiazepine Receptor ◽

Palatable Food ◽

Inverse Agonists ◽

Receptor Agonists

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INTERACTION OF BENZODIAZEPINE RECEPTOR AGONISTS AND INVERSE AGONISTS WITH THE GABA BENZODIAZEPINE RECEPTOR COMPLEX

Clinical Neuropharmacology ◽

10.1097/00002826-198406001-00436 ◽

1984 ◽

Vol 7 ◽

pp. S473

Author(s):

M. Karobath

Keyword(s):

Benzodiazepine Receptor ◽

Receptor Complex ◽

Inverse Agonists ◽

Receptor Agonists

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Cardiovascular and somatic startle and defense: Concordant and discordant actions of benzodiazepine receptor agonists and inverse agonists

Behavioural Brain Research ◽

10.1016/s0166-4328(97)00097-1 ◽

1998 ◽

Vol 90 (2) ◽

pp. 175-186 ◽

Cited By ~ 9

Author(s):

S Hart ◽

M Sarter ◽

G.G Berntson

Keyword(s):

Benzodiazepine Receptor ◽

Inverse Agonists ◽

Receptor Agonists

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Design, Evaluation, and Comparison of Ghrelin Receptor Agonists and Inverse Agonists as Suitable Radiotracers for PET Imaging

Bioconjugate Chemistry ◽

10.1021/bc2005889 ◽

2012 ◽

Vol 23 (4) ◽

pp. 771-784 ◽

Cited By ~ 24

Author(s):

Constance Chollet ◽

Ralf Bergmann ◽

Jens Pietzsch ◽

Annette G. Beck-Sickinger

Keyword(s):

Pet Imaging ◽

Design Evaluation ◽

Inverse Agonists ◽

Ghrelin Receptor ◽

Receptor Agonists

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Chronic treatment with lorazepam and FG 7142 may change the effects of benzodiazepine receptor agonists, antagonists and inverse agonists by different mechanisms

European Journal of Pharmacology ◽

10.1016/0014-2999(87)90027-6 ◽

1987 ◽

Vol 133 (3) ◽

pp. 309-317 ◽

Cited By ~ 32

Author(s):

Erling N. Petersen ◽

Leif H. Jensen

Keyword(s):

Chronic Treatment ◽

Benzodiazepine Receptor ◽

Fg 7142 ◽

Inverse Agonists ◽

Receptor Agonists

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Audiogenic seizures in DBA/2 mice discriminate sensitively between low efficacy benzodazepine receptor agonists and inverse agonists

Life Sciences ◽

10.1016/s0024-3205(83)80014-9 ◽

1983 ◽

Vol 33 (4) ◽

pp. 393-399 ◽

Cited By ~ 128

Author(s):

Leif H. Jensen ◽

Erling N. Petersen ◽

Claus Braestrup

Keyword(s):

Audiogenic Seizures ◽

Inverse Agonists ◽

Receptor Agonists

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Interaction of benzodiazepine receptor agonists and inverse agonists with the GABA benzodiazepine receptor complex

Pharmacology Biochemistry and Behavior ◽

10.1016/0091-3057(85)90435-6 ◽

1985 ◽

Vol 23 (4) ◽

pp. 671-674 ◽

Cited By ~ 12

Author(s):

Manfred Karobath ◽

Porntip Supavilai

Keyword(s):

Benzodiazepine Receptor ◽

Receptor Complex ◽

Inverse Agonists ◽

Receptor Agonists

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Benzodiazepine receptor agonists and inverse agonists yield concordant rather than opposing effects on startle responses

Journal of Psychopharmacology ◽

10.1177/026988119601000409 ◽

1996 ◽

Vol 10 (4) ◽

pp. 309-312 ◽

Cited By ~ 5

Author(s):

G. Berntson ◽

M. Sarter ◽

S. Ruland ◽

S. Hart ◽

V. Ronis

Keyword(s):

Benzodiazepine Receptor ◽

Inverse Agonists ◽

Receptor Agonists ◽

Opposing Effects

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The affinities, potencies and efficacies of some benzodiazepine-receptor agonists, antagonists and inverse-agonists at rat hippocampal GABAA-receptors

British Journal of Pharmacology ◽

10.1111/j.1476-5381.1987.tb11253.x ◽

1987 ◽

Vol 91 (3) ◽

pp. 601-608 ◽

Cited By ~ 38

Author(s):

J.A. Kemp ◽

G.R. Marshall ◽

E.H.F. Wong ◽

G.N. Woodruff

Keyword(s):

Gabaa Receptors ◽

Benzodiazepine Receptor ◽

Inverse Agonists ◽

Receptor Agonists

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