scholarly journals Fluorine in fragrances: exploring the difluoromethylene (CF2) group as a conformational constraint in macrocyclic musk lactones

2016 ◽  
Vol 14 (1) ◽  
pp. 211-219 ◽  
Author(s):  
Michael J. Corr ◽  
Rodrigo A. Cormanich ◽  
Cortney N. von Hahmann ◽  
Michael Bühl ◽  
David B. Cordes ◽  
...  
Keyword(s):  
Conformational Constraint

The synthesis of a series of selectively fluorinated musk lactones is reported with CF2 groups at various locations to bias conformation the ring.

Conformational Constraint of the Glycerol Moiety of Lysophosphatidylserine Affords Compounds with Receptor Subtype Selectivity

2016 ◽  
Vol 59 (8) ◽  
pp. 3750-3776 ◽  
Author(s):  
Sejin Jung ◽  
Asuka Inoue ◽  
Sho Nakamura ◽  
Takayuki Kishi ◽  
Akiharu Uwamizu ◽  
...  
Keyword(s):  
Receptor Subtype ◽  
Glycerol Moiety ◽  
Subtype Selectivity ◽  
Conformational Constraint

Backbone cyclization as a tool for imposing conformational constraint on peptides

1993 ◽  
pp. 482-485 ◽  
Author(s):  
Chaim Gilon ◽  
Irena Zeltser ◽  
Vered Rashti-Bahar ◽  
Dan Muller ◽  
Gal Bitan ◽  
...  
Keyword(s):  
Conformational Constraint ◽  
Backbone Cyclization

scholarly journals Tuning the Morphology of Nanostructured Peptide Films by the Introduction of a Secondary Structure Conformational Constraint: A Case Study of Hierarchical Self-Assembly

2018 ◽  
Vol 122 (24) ◽  
pp. 6305-6313 ◽  
Author(s):  
Marta De Zotti ◽  
Beatrice Muzzi ◽  
Emanuela Gatto ◽  
Benedetta Di Napoli ◽  
Claudia Mazzuca ◽  
...  
Keyword(s):  
Secondary Structure ◽  
Self Assembly ◽  
Conformational Constraint

Stereospecific synthesis of (2R,3S)-3-amino-2-piperidineacetic acid derivatives for use as conformational constraint in peptides

1993 ◽  
Vol 34 (22) ◽  
pp. 3593-3594 ◽  
Author(s):  
Isabel Gómez-Monterrey ◽  
Rosario González-Muñiz ◽  
Rosario Herranz ◽  
M.a Teresa Garcia-Gomez
Keyword(s):  
Stereospecific Synthesis ◽  
Conformational Constraint

A conformational constraint improves a β-secretase inhibitor but for an unexpected reason

2009 ◽  
Vol 19 (17) ◽  
pp. 4993-4995 ◽  
Author(s):  
Ivory D. Hills ◽  
M. Katharine Holloway ◽  
Pablo de León ◽  
Ashley Nomland ◽  
Hong Zhu ◽  
...  
Keyword(s):  
Conformational Constraint ◽  
Secretase Inhibitor

Design and Validation of Bicyclic Iminopyrimidinones As Beta Amyloid Cleaving Enzyme-1 (BACE1) Inhibitors: Conformational Constraint to Favor a Bioactive Conformation

2012 ◽  
Vol 55 (21) ◽  
pp. 9331-9345 ◽  
Author(s):  
Mihirbaran Mandal ◽  
Zhaoning Zhu ◽  
Jared N. Cumming ◽  
Xiaoxiang Liu ◽  
Corey Strickland ◽  
...  
Keyword(s):  
Beta Amyloid ◽  
Bioactive Conformation ◽  
Conformational Constraint

Conformational constraint in ferroelectric liquid crystals incorporating a pyrrolidine‐type ring: FLC materials comprising parallel dipolar moments

2007 ◽  
Vol 34 (4) ◽  
pp. 431-440
Author(s):  
Fernando Ely ◽  
Rodrigo Cristiano ◽  
Ricardo L. Longo ◽  
Rafael Vergara‐Toloza ◽  
Eduardo Soto‐Bustamante ◽  
...  
Keyword(s):  
Liquid Crystals ◽  
Ferroelectric Liquid Crystals ◽  
Conformational Constraint
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