Enantioselective Synthesis of Brinzolamide (AL-4862), a New Topical Carbonic Anhydrase Inhibitor. The “DCAT Route” to Thiophenesulfonamides

1999 ◽  
Vol 3 (2) ◽  
pp. 114-120 ◽  
Author(s):  
Raymond E. Conrow ◽  
W. Dennis Dean ◽  
Paul W. Zinke ◽  
Michael E. Deason ◽  
Steven J. Sproull ◽  
...  
Keyword(s):  
Carbonic Anhydrase ◽  
Carbonic Anhydrase Inhibitor ◽  
Enantioselective Synthesis

ChemInform Abstract: Enantioselective Synthesis of Brinzolamide (AL-4862), a New Topical Carbonic Anhydrase Inhibitor. The “DCAT Route” to Thiophenesulfonamides.

ChemInform ◽  
2010 ◽  
Vol 30 (29) ◽  
pp. no-no
Author(s):  
Raymond E. Conrow ◽  
W. Dennis Dean ◽  
Paul W. Zinke ◽  
Michael E. Deason ◽  
Steven J. Sproull ◽  
...  
Keyword(s):  
Carbonic Anhydrase ◽  
Carbonic Anhydrase Inhibitor ◽  
Enantioselective Synthesis

ChemInform Abstract: Enantioselective Synthesis of AL-4414A, a Topically Active Carbonic Anhydrase Inhibitor.

ChemInform ◽  
2010 ◽  
Vol 29 (20) ◽  
pp. no-no
Author(s):  
M. T. DUPRIEST ◽  
P. W. ZINKE ◽  
R. E. CONROW ◽  
D. KUZMICH ◽  
A. P. DANTANARAYANA ◽  
...  
Keyword(s):  
Carbonic Anhydrase ◽  
Carbonic Anhydrase Inhibitor ◽  
Enantioselective Synthesis ◽  
Active Carbonic Anhydrase

Enantioselective Synthesis of AL-4414A, a Topically Active Carbonic Anhydrase Inhibitor

1997 ◽  
Vol 62 (26) ◽  
pp. 9372-9375 ◽  
Author(s):  
Mark T. DuPriest ◽  
Paul W. Zinke ◽  
Raymond E. Conrow ◽  
Daniel Kuzmich ◽  
Anura P. Dantanarayana ◽  
...  
Keyword(s):  
Carbonic Anhydrase ◽  
Carbonic Anhydrase Inhibitor ◽  
Enantioselective Synthesis ◽  
Active Carbonic Anhydrase

The Effect of a Carbonic Anhydrase Inhibitor, Diamox, On Human Pancreatic Secretion

1955 ◽  
Vol 29 (2) ◽  
pp. 262-279 ◽  
Author(s):  
David A. Dreiling ◽  
Henry D. Janowitz ◽  
Mark Halpern
Keyword(s):  
Carbonic Anhydrase ◽  
Pancreatic Secretion ◽  
Carbonic Anhydrase Inhibitor

The Carbonic Anhydrase Inhibitor E7070 Sensitizes Glioblastoma Cells to Radio- and Chemotherapy and Reduces Tumor Growth

2021 ◽  
Author(s):  
Silvia A. Teixeira ◽  
Mariano S. Viapiano ◽  
Augusto F. Andrade ◽  
Mohan S. Nandhu ◽  
Julia A. Pezuk ◽  
...  
Keyword(s):  
Carbonic Anhydrase ◽  
Tumor Growth ◽  
Carbonic Anhydrase Inhibitor ◽  
Glioblastoma Cells

Polypharmacology of epacadostat: a potent and selective inhibitor of the tumor associated carbonic anhydrases IX and XII

2019 ◽  
Vol 55 (40) ◽  
pp. 5720-5723 ◽  
Author(s):  
Andrea Angeli ◽  
Marta Ferraroni ◽  
Alessio Nocentini ◽  
Silvia Selleri ◽  
Paola Gratteri ◽  
...  
Keyword(s):  
Carbonic Anhydrase ◽  
Selective Inhibitor ◽  
Carbonic Anhydrase Inhibitor ◽  
Carbonic Anhydrases ◽  
Indoleamine 2,3 Dioxygenase

Epacadostat (EPA), a selective indoleamine-2,3-dioxygenase 1 (IDO1) inhibitor, has been investigatedin vitroas a human (h) Carbonic Anhydrase Inhibitor (CAI).

Structural modulation of the biological activity of gold nanoparticles functionalized with a carbonic anhydrase inhibitor

2013 ◽  
Vol 36 (5) ◽  
Author(s):  
Francesca Bellissima ◽  
Fabrizio Carta ◽  
Alessio Innocenti ◽  
Andrea Scozzafava ◽  
Piero Baglioni ◽  
...  
Keyword(s):  
Gold Nanoparticles ◽  
Biological Activity ◽  
Carbonic Anhydrase ◽  
Carbonic Anhydrase Inhibitor ◽  
Structural Modulation
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