Palladium(0)-Catalyzed Cyclization Reaction of Polymer-Supported Aryl Iodides with 1,2-Allenyl Carboxylic Acids. A Facile Solid-Phase Synthesis of Butenolides†

2000 ◽  
Vol 2 (10) ◽  
pp. 1419-1422 ◽  
Author(s):  
Shengming Ma ◽  
Dehui Duan ◽  
Zhangjie Shi
Keyword(s):  
Carboxylic Acids ◽  
Solid Phase Synthesis ◽  
Solid Phase ◽  
Cyclization Reaction ◽  
Phase Synthesis ◽  
Aryl Iodides ◽  
Polymer Supported

Solid-phase synthesis of (Z)-allyl iodides from 3-acetoxy-2-methylene-alkanoates with recyclable polymer-supported selenium bromide

2007 ◽  
Vol 18 (4) ◽  
pp. 377-379 ◽  
Author(s):  
Shou Ri Sheng ◽  
Ming Gang Hu ◽  
Qin Xin ◽  
Xiao Ling Liu ◽  
Xian Huang
Keyword(s):  
Solid Phase Synthesis ◽  
Solid Phase ◽  
Phase Synthesis ◽  
Polymer Supported

Polymer supported calixarene derivative useful for solid-phase synthesis application

2010 ◽  
Vol 51 (47) ◽  
pp. 6139-6142 ◽  
Author(s):  
Giuseppe Granata ◽  
Grazia M.L. Consoli ◽  
Sebastiano Sciuto ◽  
Corrada Geraci
Keyword(s):  
Solid Phase Synthesis ◽  
Solid Phase ◽  
Phase Synthesis ◽  
Calixarene Derivative ◽  
Polymer Supported

Combinatorial Solid-Phase Synthesis of 6-Aryl-1,3,5-triazines via Suzuki Coupling

2011 ◽  
Vol 64 (5) ◽  
pp. 540 ◽  
Author(s):  
Jae Wook Lee ◽  
Hyung-Ho Ha ◽  
Marc Vendrell ◽  
Jacqueline T. Bork ◽  
Young-Tae Chang
Keyword(s):  
Solid Phase Synthesis ◽  
Solid Phase ◽  
Cross Coupling ◽  
Structural Diversity ◽  
Suzuki Coupling ◽  
Purification Step ◽  
Solid Supports ◽  
Phase Synthesis ◽  
Triazine Derivatives ◽  
Polymer Supported

A synthetic methodology to prepare collections of trisubstituted aryl 1,3,5-triazines with broad structural diversity via Suzuki coupling has been developed. We first optimized the combinatorial derivatization of the triazine core using Suzuki cross-coupling. Second, in order to further expand the methodology for the preparation of negatively charged triazines, we adapted this approach to polymer-supported amino acids and prepared aryl triazines with different charge distribution. With a collection of 160 aryl triazine derivatives in good purities and without any purification step, we proved the viability of this orthogonal scheme for the preparation of triazine libraries using amine/amino acid-captured solid supports and Suzuki cross-coupling.

Solid-phase synthesis of α-alkylserines via phase-transfer catalytic alkylation of polymer-supported 2-phenyl-2-oxazoline-4-carboxylate

Tetrahedron ◽  
2009 ◽  
Vol 65 (43) ◽  
pp. 8839-8843 ◽  
Author(s):  
Jihye Lee ◽  
Min Woo Ha ◽  
Taek-Soo Kim ◽  
Mi-Jeong Kim ◽  
Jin-Mo Ku ◽  
...  
Keyword(s):  
Solid Phase Synthesis ◽  
Phase Transfer ◽  
Solid Phase ◽  
Phase Synthesis ◽  
Catalytic Alkylation ◽  
Polymer Supported
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