Determination of isokinetic ratios necessary for equimolar incorporation of carboxylic acids in the solid-phase synthesis of mixture-based combinatorial libraries

Achyuta N. Acharya; John M. Ostresh; Richard A. Houghten

doi:10.1002/bip.10206

Determination of isokinetic ratios necessary for equimolar incorporation of carboxylic acids in the solid-phase synthesis of mixture-based combinatorial libraries

Biopolymers ◽

10.1002/bip.10206 ◽

2002 ◽

Vol 65 (1) ◽

pp. 32-39 ◽

Cited By ~ 9

Author(s):

Achyuta N. Acharya ◽

John M. Ostresh ◽

Richard A. Houghten

Keyword(s):

Carboxylic Acids ◽

Solid Phase Synthesis ◽

Solid Phase ◽

Combinatorial Libraries ◽

Phase Synthesis

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Determination of 9-fluorenylmethoxycarbonyl (Fmoc) resin loading in solid‐phase synthesis by RP-HPLC internal standard method

Monatshefte für Chemie - Chemical Monthly ◽

10.1007/s00706-021-02789-5 ◽

2021 ◽

Author(s):

Hynek Mácha ◽

Marek Kořínek ◽

Ladislav Drož ◽

Karel Nesměrák

Keyword(s):

Standard Method ◽

Solid Phase Synthesis ◽

Solid Phase ◽

Internal Standard ◽

Internal Standard Method ◽

Phase Synthesis ◽

Rp Hplc ◽

Resin Loading

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Combinatorial Libraries on Rigid Scaffolds: Solid Phase Synthesis of Variably Substituted Pyrazoles and Isoxazoles

Molecules ◽

10.3390/jan97p5 ◽

1997 ◽

Vol 2 (12) ◽

pp. 17-30 ◽

Cited By ~ 14

Author(s):

Andreas Marzinzik ◽

Eduard Felder

Keyword(s):

Solid Phase Synthesis ◽

Solid Phase ◽

Combinatorial Libraries ◽

Phase Synthesis ◽

Substituted Pyrazoles

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How to Optimize Reactions for Solid-Phase Synthesis of Combinatorial Libraries Using RF-Tagged Microreactors

Optimization of Solid-Phase Combinatorial Synthesis ◽

10.1201/9781482271058-5 ◽

2001 ◽

pp. 69-82

Keyword(s):

Solid Phase Synthesis ◽

Solid Phase ◽

Combinatorial Libraries ◽

Phase Synthesis

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Elimination Chemistry in the Solution- and Solid-Phase Synthesis of Combinatorial Libraries

ChemInform ◽

10.1002/chin.200411244 ◽

2004 ◽

Vol 35 (11) ◽

Author(s):

Demosthenes Fokas ◽

Carmen Baldino

Keyword(s):

Solid Phase Synthesis ◽

Solid Phase ◽

Combinatorial Libraries ◽

Phase Synthesis

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Stereoselective Solid-Phase Synthesis of Cyclopentane and Cyclohexane Derivatives by Two-Component Domino Reactions: Generation of Combinatorial Libraries

Angewandte Chemie International Edition in English ◽

10.1002/anie.199606511 ◽

1996 ◽

Vol 35 (6) ◽

pp. 651-652 ◽

Cited By ~ 43

Author(s):

Lutz F. Tietze ◽

Adrian Steinmetz

Keyword(s):

Solid Phase Synthesis ◽

Solid Phase ◽

Combinatorial Libraries ◽

Domino Reactions ◽

Phase Synthesis ◽

Two Component

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Solid phase synthesis, NMR structure determination of α-KTx3.8, its in silico docking to Kv1.x potassium channels, and electrophysiological analysis provide insights into toxin-channel selectivity

Toxicon ◽

10.1016/j.toxicon.2015.04.018 ◽

2015 ◽

Vol 101 ◽

pp. 70-78 ◽

Cited By ~ 7

Author(s):

Bastian Kohl ◽

Ina Rothenberg ◽

Syed Abid Ali ◽

Mehtab Alam ◽

Guiscard Seebohm ◽

...

Keyword(s):

Potassium Channels ◽

Structure Determination ◽

In Silico ◽

Solid Phase Synthesis ◽

Solid Phase ◽

Nmr Structure Determination ◽

Phase Synthesis ◽

In Silico Docking ◽

Channel Selectivity

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Solid phase synthesis of mixture-based acyclic and heterocyclic small molecule combinatorial libraries from resin-bound polyamides

Biopolymers ◽

10.1002/1097-0282(2001)60:3<212::aid-bip10033>3.0.co;2-d ◽

2001 ◽

Vol 60 (3) ◽

pp. 212-219 ◽

Cited By ~ 8

Author(s):

Adel Nefzi ◽

John M. Ostresh ◽

Richard A. Houghten

Keyword(s):

Small Molecule ◽

Solid Phase Synthesis ◽

Solid Phase ◽

Combinatorial Libraries ◽

Phase Synthesis

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ChemInform Abstract: Solid-Phase Synthesis of Mixture-Based Acyclic and Heterocyclic Small Molecule Combinatorial Libraries from Resin-Bound Polyamides.

ChemInform ◽

10.1002/chin.200225266 ◽

2010 ◽

Vol 33 (25) ◽

pp. no-no

Author(s):

Adel Nefzi ◽

John M. Ostresh ◽

Richard A. Houghten

Keyword(s):

Small Molecule ◽

Solid Phase Synthesis ◽

Solid Phase ◽

Combinatorial Libraries ◽

Phase Synthesis

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Palladium(0)-Catalyzed Cyclization Reaction of Polymer-Supported Aryl Iodides with 1,2-Allenyl Carboxylic Acids. A Facile Solid-Phase Synthesis of Butenolides†

Organic Letters ◽

10.1021/ol0057481 ◽

2000 ◽

Vol 2 (10) ◽

pp. 1419-1422 ◽

Cited By ~ 36

Author(s):

Shengming Ma ◽

Dehui Duan ◽

Zhangjie Shi

Keyword(s):

Carboxylic Acids ◽

Solid Phase Synthesis ◽

Solid Phase ◽

Cyclization Reaction ◽

Phase Synthesis ◽

Aryl Iodides ◽

Polymer Supported

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Faculty Opinions recommendation of Solid phase synthesis of mixture-based acyclic and heterocyclic small molecule combinatorial libraries from resin-bound polyamides.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1003350.35604 ◽

2002 ◽

Author(s):

Morten Meldal

Keyword(s):

Small Molecule ◽

Solid Phase Synthesis ◽

Solid Phase ◽

Combinatorial Libraries ◽

Phase Synthesis

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