Crystal Structures and Structure–Activity Relationships of Imidazothiazole Derivatives as IDO1 Inhibitors

Shingo Tojo; Tetsuya Kohno; Tomoyuki Tanaka; Seiji Kamioka; Yosuke Ota; Takayuki Ishii; Keiko Kamimoto; Shigehiro Asano; Yoshiaki Isobe

doi:10.1021/ml500247w

Crystal Structures and Structure–Activity Relationships of Imidazothiazole Derivatives as IDO1 Inhibitors

ACS Medicinal Chemistry Letters ◽

10.1021/ml500247w ◽

2014 ◽

Vol 5 (10) ◽

pp. 1119-1123 ◽

Cited By ~ 79

Author(s):

Shingo Tojo ◽

Tetsuya Kohno ◽

Tomoyuki Tanaka ◽

Seiji Kamioka ◽

Yosuke Ota ◽

...

Keyword(s):

Crystal Structures ◽

Structure Activity Relationships ◽

Structure Activity

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Contributions of crystal structures, molecular electrostatic potential maps, and lipophilicity data to structure-activity relationships of some conformationally restricted nortropane benzamide neuroleptics

Journal of Crystallographic and Spectroscopic Research ◽

10.1007/bf01160656 ◽

1991 ◽

Vol 21 (4) ◽

pp. 431-443 ◽

Cited By ~ 4

Author(s):

Sonia Collin ◽

Alain Patiny ◽

Daniel P. Vercauteren ◽

Bernadette Norberg ◽

Guy Evrard ◽

...

Keyword(s):

Crystal Structures ◽

Electrostatic Potential ◽

Molecular Electrostatic Potential ◽

Structure Activity Relationships ◽

Conformationally Restricted ◽

Structure Activity ◽

Molecular Electrostatic Potential Maps

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Peptide and Peptide Mimetic Inhibitors of Antigen Presentation by HLA-DR Class II MHC Molecules. Design, Structure−Activity Relationships, and X-ray Crystal Structures

Journal of Medicinal Chemistry ◽

10.1021/jm000034h ◽

2000 ◽

Vol 43 (11) ◽

pp. 2135-2148 ◽

Cited By ~ 68

Author(s):

David R. Bolin ◽

Amy L. Swain ◽

Ramakanth Sarabu ◽

Steven J. Berthel ◽

Paul Gillespie ◽

...

Keyword(s):

Antigen Presentation ◽

Crystal Structures ◽

Class Ii ◽

X Ray ◽

Structure Activity Relationships ◽

Mhc Molecules ◽

Structure Activity ◽

Design Structure ◽

Hla Dr ◽

Class Ii Mhc

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Synthesis, Crystal Structures, Insecticidal Activities, and Structure−Activity Relationships of NovelN′-tert-Butyl-N′-substituted-benzoyl-N-[di(octa)hydro]benzofuran{(2,3-dihydro)benzo[1,3]([1,4])dioxine}carbohydrazide Derivatives

Journal of Agricultural and Food Chemistry ◽

10.1021/jf104196t ◽

2011 ◽

Vol 59 (2) ◽

pp. 635-644 ◽

Cited By ~ 16

Author(s):

Zhiqiang Huang ◽

Yuxiu Liu ◽

Yongqiang Li ◽

Lixia Xiong ◽

Zhipeng Cui ◽

...

Keyword(s):

Crystal Structures ◽

Tert Butyl ◽

Structure Activity Relationships ◽

Structure Activity ◽

Insecticidal Activities

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Structure–activity relationships and crystal structures of some interesting oxazolidinones

Acta Crystallographica Section A Foundations of Crystallography ◽

10.1107/s0108767396089167 ◽

1996 ◽

Vol 52 (a1) ◽

pp. C258-C258

Author(s):

W. Watt ◽

F. Han ◽

J. H. VanDrie ◽

L. M. Thomasco

Keyword(s):

Crystal Structures ◽

Structure Activity Relationships ◽

Structure Activity

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Configuration and preferential solid-state conformations of perindoprilat (S-9780). Comparison with the crystal structures of other ACE inhibitors and conclusions related to structure-activity relationships

Journal of Medicinal Chemistry ◽

10.1021/jm00106a030 ◽

1991 ◽

Vol 34 (2) ◽

pp. 663-669 ◽

Cited By ~ 29

Author(s):

Claudine Pascard ◽

Jean Guilhem ◽

Michel Vincent ◽

Georges Remond ◽

Bernard Portevin ◽

...

Keyword(s):

Solid State ◽

Crystal Structures ◽

Ace Inhibitors ◽

Structure Activity Relationships ◽

Structure Activity

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Structure-Activity Relationships of MDMA-Like Substances

PsycEXTRA Dataset ◽

10.1037/e496472006-001 ◽

1989 ◽

Cited By ~ 3

Author(s):

David E. Nichols ◽

◽

Robert Oberlender

Keyword(s):

Structure Activity Relationships ◽

Structure Activity

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Structure-Activity Relationships in Cannabinoids: An Overview

PsycEXTRA Dataset ◽

10.1037/e496672006-002 ◽

1987 ◽

Author(s):

Raj K. Razdan ◽

Keyword(s):

Structure Activity Relationships ◽

Structure Activity

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Structure-Activity and Selectivity Relationships in Heterogeneous Catalysis, Proceedings of the ACS Symposium on Structure-Activity Relationships in Heterogeneous Catalysis

10.1016/s0167-2991(08)x6047-1 ◽

1991 ◽

Keyword(s):

Heterogeneous Catalysis ◽

Structure Activity Relationships ◽

Structure Activity

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Structure-activity relationships in the acronycine and benzo[b]acronycine series: Role of the pyran ring

Planta Medica ◽

10.1055/s-0028-1084761 ◽

2008 ◽

Vol 74 (09) ◽

Author(s):

Q Do ◽

H Doan Thi Mai ◽

T Gaslonde ◽

B Pfeiffer ◽

S Léonce ◽

...

Keyword(s):

Pyran Ring ◽

Structure Activity Relationships ◽

Structure Activity

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Structure activity-relationships of P-Glycoprotein modulation using a small library of macrocyclic lathyrane diterpenes

Planta Medica ◽

10.1055/s-0032-1320394 ◽

2012 ◽

Vol 78 (11) ◽

Author(s):

M Reis ◽

RJ Ferreira ◽

MMM Santos ◽

DJVA dos Santos ◽

J Molnár ◽

...

Keyword(s):

Structure Activity Relationships ◽

Structure Activity ◽

P Glycoprotein

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