scholarly journals Discovery of 3,4-Dihydropyrimidin-2(1H)-ones As a Novel Class of Potent and Selective A2B Adenosine Receptor Antagonists

2013 ◽  
Vol 4 (11) ◽  
pp. 1031-1036 ◽  
Author(s):  
Abel Crespo ◽  
Abdelaziz El Maatougui ◽  
Pierfrancesco Biagini ◽  
Jhonny Azuaje ◽  
Alberto Coelho ◽  
...  
Keyword(s):  
Adenosine Receptor ◽  
Receptor Antagonists ◽  
A2b Adenosine Receptor

Pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives as adenosine receptor ligands: A starting point for searching A2B adenosine receptor antagonists

2001 ◽  
Vol 53 (2-3) ◽  
pp. 225-235 ◽  
Author(s):  
Pier Giovanni Baraldi ◽  
Barbara Cacciari ◽  
Romeo Romagnoli ◽  
Karl-Norbert Klotz ◽  
Giampiero Spalluto ◽  
...  
Keyword(s):  
Adenosine Receptor ◽  
Receptor Ligands ◽  
Pyrimidine Derivatives ◽  
Receptor Antagonists ◽  
A2b Adenosine Receptor ◽  
Starting Point ◽  
Adenosine Receptor Ligands

Exploring the influence of the substituent at position 4 in a series of 3,4-dihydropyrimidin-2(1H)-one A2B adenosine receptor antagonists

2017 ◽  
Vol 53 (3) ◽  
pp. 316-321 ◽  
Author(s):  
Abel Crespo ◽  
Abdelaziz El Maatougui ◽  
Jhonny Azuaje ◽  
Luz Escalante ◽  
María Majellaro ◽  
...  
Keyword(s):  
Adenosine Receptor ◽  
Receptor Antagonists ◽  
A2b Adenosine Receptor

QSAR and docking analysis of A2B adenosine receptor antagonists based on non-xanthine scaffold

2014 ◽  
Vol 24 (1) ◽  
pp. 394-407 ◽  
Author(s):  
Mahboubeh Mansourian ◽  
Afshin Fassihi ◽  
Lotfollah Saghaie ◽  
Armin Madadkar-Sobhani ◽  
Karim Mahnam ◽  
...  
Keyword(s):  
Adenosine Receptor ◽  
Receptor Antagonists ◽  
Docking Analysis ◽  
A2b Adenosine Receptor

Novel 1,3-Dipropyl-8-(3-benzimidazol-2-yl-methoxy-1-methylpyrazol-5-yl)xanthines as Potent and Selective A2B Adenosine Receptor Antagonists

2012 ◽  
Vol 55 (2) ◽  
pp. 797-811 ◽  
Author(s):  
Pier Giovanni Baraldi ◽  
Stefania Baraldi ◽  
Giulia Saponaro ◽  
Delia Preti ◽  
Romeo Romagnoli ◽  
...  
Keyword(s):  
Adenosine Receptor ◽  
Receptor Antagonists ◽  
A2b Adenosine Receptor

New pyrrolopyrimidin-6-yl benzenesulfonamides: Potent A2B adenosine receptor antagonists

2006 ◽  
Vol 16 (14) ◽  
pp. 3642-3645 ◽  
Author(s):  
Cristina Esteve ◽  
Arsenio Nueda ◽  
José Luis Díaz ◽  
Jorge Beleta ◽  
Alvaro Cárdenas ◽  
...  
Keyword(s):  
Adenosine Receptor ◽  
Receptor Antagonists ◽  
A2b Adenosine Receptor

Antinociceptive Effects of Novel A2B Adenosine Receptor Antagonists

2003 ◽  
Vol 308 (1) ◽  
pp. 358-366 ◽  
Author(s):  
Osama M. Abo-Salem ◽  
Alaa M. Hayallah ◽  
Andras Bilkei-Gorzo ◽  
Barbara Filipek ◽  
Andreas Zimmer ◽  
...  
Keyword(s):  
Adenosine Receptor ◽  
Receptor Antagonists ◽  
A2b Adenosine Receptor ◽  
Antinociceptive Effects

New Pyrrolopyrimidin-6-yl Benzenesulfonamides: Potent A2B Adenosine Receptor Antagonists.

ChemInform ◽  
2006 ◽  
Vol 37 (42) ◽  
Author(s):  
Cristina Esteve ◽  
Arsenio Nueda ◽  
Jose Luis Diaz ◽  
Jorge Beleta ◽  
Alvaro Cardenas ◽  
...  
Keyword(s):  
Adenosine Receptor ◽  
Receptor Antagonists ◽  
A2b Adenosine Receptor

Discovery of N-(5,6-diarylpyridin-2-yl)amide derivatives as potent and selective A2B adenosine receptor antagonists

2010 ◽  
Vol 20 (5) ◽  
pp. 1697-1700 ◽  
Author(s):  
Paul Eastwood ◽  
Jacob Gonzalez ◽  
Sergio Paredes ◽  
Arsenio Nueda ◽  
Teresa Domenech ◽  
...  
Keyword(s):  
Adenosine Receptor ◽  
Receptor Antagonists ◽  
A2b Adenosine Receptor ◽  
Amide Derivatives
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