Novel 1,3-Dipropyl-8-(1-heteroarylmethyl-1H-pyrazol-4-yl)-xanthine Derivatives as High Affinity and Selective A2B Adenosine Receptor Antagonists.

ChemInform ◽  
2006 ◽  
Vol 37 (16) ◽  
Author(s):  
Elfatih Elzein ◽  
et al. et al.
Keyword(s):  
Adenosine Receptor ◽  
Receptor Antagonists ◽  
A2b Adenosine Receptor ◽  
High Affinity ◽  
Xanthine Derivatives

1,3-Dipropyl-8-(1-phenylacetamide-1H-pyrazol-3-yl)-xanthine derivatives as highly potent and selective human A2B adenosine receptor antagonists

2008 ◽  
Vol 16 (5) ◽  
pp. 2419-2430 ◽  
Author(s):  
Mojgan Aghazadeh Tabrizi ◽  
Pier Giovanni Baraldi ◽  
Delia Preti ◽  
Romeo Romagnoli ◽  
Giulia Saponaro ◽  
...  
Keyword(s):  
Adenosine Receptor ◽  
Receptor Antagonists ◽  
A2b Adenosine Receptor ◽  
Xanthine Derivatives

Selective, high affinity A2B adenosine receptor antagonists: N-1 monosubstituted 8-(pyrazol-4-yl)xanthines

2008 ◽  
Vol 18 (4) ◽  
pp. 1397-1401 ◽  
Author(s):  
Rao V. Kalla ◽  
Elfatih Elzein ◽  
Thao Perry ◽  
Xiaofen Li ◽  
Art Gimbel ◽  
...  
Keyword(s):  
Adenosine Receptor ◽  
Receptor Antagonists ◽  
A2b Adenosine Receptor ◽  
High Affinity

scholarly journals Discovery of 3,4-Dihydropyrimidin-2(1H)-ones As a Novel Class of Potent and Selective A2B Adenosine Receptor Antagonists

2013 ◽  
Vol 4 (11) ◽  
pp. 1031-1036 ◽  
Author(s):  
Abel Crespo ◽  
Abdelaziz El Maatougui ◽  
Pierfrancesco Biagini ◽  
Jhonny Azuaje ◽  
Alberto Coelho ◽  
...  
Keyword(s):  
Adenosine Receptor ◽  
Receptor Antagonists ◽  
A2b Adenosine Receptor

Pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives as adenosine receptor ligands: A starting point for searching A2B adenosine receptor antagonists

2001 ◽  
Vol 53 (2-3) ◽  
pp. 225-235 ◽  
Author(s):  
Pier Giovanni Baraldi ◽  
Barbara Cacciari ◽  
Romeo Romagnoli ◽  
Karl-Norbert Klotz ◽  
Giampiero Spalluto ◽  
...  
Keyword(s):  
Adenosine Receptor ◽  
Receptor Ligands ◽  
Pyrimidine Derivatives ◽  
Receptor Antagonists ◽  
A2b Adenosine Receptor ◽  
Starting Point ◽  
Adenosine Receptor Ligands

Exploring the influence of the substituent at position 4 in a series of 3,4-dihydropyrimidin-2(1H)-one A2B adenosine receptor antagonists

2017 ◽  
Vol 53 (3) ◽  
pp. 316-321 ◽  
Author(s):  
Abel Crespo ◽  
Abdelaziz El Maatougui ◽  
Jhonny Azuaje ◽  
Luz Escalante ◽  
María Majellaro ◽  
...  
Keyword(s):  
Adenosine Receptor ◽  
Receptor Antagonists ◽  
A2b Adenosine Receptor

QSAR and docking analysis of A2B adenosine receptor antagonists based on non-xanthine scaffold

2014 ◽  
Vol 24 (1) ◽  
pp. 394-407 ◽  
Author(s):  
Mahboubeh Mansourian ◽  
Afshin Fassihi ◽  
Lotfollah Saghaie ◽  
Armin Madadkar-Sobhani ◽  
Karim Mahnam ◽  
...  
Keyword(s):  
Adenosine Receptor ◽  
Receptor Antagonists ◽  
Docking Analysis ◽  
A2b Adenosine Receptor

Novel 1,3-Dipropyl-8-(3-benzimidazol-2-yl-methoxy-1-methylpyrazol-5-yl)xanthines as Potent and Selective A2B Adenosine Receptor Antagonists

2012 ◽  
Vol 55 (2) ◽  
pp. 797-811 ◽  
Author(s):  
Pier Giovanni Baraldi ◽  
Stefania Baraldi ◽  
Giulia Saponaro ◽  
Delia Preti ◽  
Romeo Romagnoli ◽  
...  
Keyword(s):  
Adenosine Receptor ◽  
Receptor Antagonists ◽  
A2b Adenosine Receptor
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