Design, Synthesis, and Pharmacological Evaluation of Conformationally Constrained Analogues ofN,N‘-Diaryl- andN-Aryl-N-aralkylguanidines as Potent Inhibitors of Neuronal Na+Channels

1998 ◽  
Vol 41 (16) ◽  
pp. 3048-3061 ◽  
Author(s):  
Michel C. Maillard ◽  
Michael E. Perlman ◽  
Oved Amitay ◽  
Deborah Baxter ◽  
David Berlove ◽  
...  
Keyword(s):  
Na Channels ◽  
Design Synthesis ◽  
Conformationally Constrained ◽  
Pharmacological Evaluation

Design, synthesis and pharmacological evaluation of tricyclic derivatives as selective RXFP4 agonists

2021 ◽  
pp. 104782
Author(s):  
Lin Lin ◽  
Guangyao Lin ◽  
Qingtong Zhou ◽  
Ross A.D. Bathgate ◽  
Grace Qun Gong ◽  
...  
Keyword(s):  
Design Synthesis ◽  
Pharmacological Evaluation

Design, Synthesis, and Pharmacological Evaluation of Glutamate Carboxypeptidase II (GCPII) Inhibitors Based on Thioalkylbenzoic Acid Scaffolds

2012 ◽  
Vol 55 (12) ◽  
pp. 5922-5932 ◽  
Author(s):  
Doris Stoermer ◽  
Dilrukshi Vitharana ◽  
Niyada Hin ◽  
Greg Delahanty ◽  
Bridget Duvall ◽  
...  
Keyword(s):  
Design Synthesis ◽  
Glutamate Carboxypeptidase Ii ◽  
Pharmacological Evaluation ◽  
Glutamate Carboxypeptidase

Design, Synthesis, and Pharmacological Evaluation of Mefloquine-Based Ligands as Novel Antituberculosis Agents

ChemMedChem ◽  
2007 ◽  
Vol 2 (11) ◽  
pp. 1624-1630 ◽  
Author(s):  
Jialin Mao ◽  
Yuehong Wang ◽  
Baojie Wan ◽  
Alan P. Kozikowski ◽  
Scott G. Franzblau
Keyword(s):  
Design Synthesis ◽  
Pharmacological Evaluation

Design, synthesis, and pharmacological evaluation of phenoxy pyridyl derivatives as dual norepinephrine reuptake inhibitors and 5-HT1A partial agonists

2010 ◽  
Vol 20 (3) ◽  
pp. 1114-1117 ◽  
Author(s):  
Amy B. Dounay ◽  
Nancy S. Barta ◽  
Brian M. Campbell ◽  
Corey Coleman ◽  
Elizabeth M. Collantes ◽  
...  
Keyword(s):  
Design Synthesis ◽  
Pharmacological Evaluation ◽  
Partial Agonists ◽  
Norepinephrine Reuptake
Sign in / Sign up

Export Citation Format

Share Document