Design, Synthesis, and Pharmacological Evaluation of Glutamate Carboxypeptidase II (GCPII) Inhibitors Based on Thioalkylbenzoic Acid Scaffolds

2012 ◽  
Vol 55 (12) ◽  
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Author(s):  
Doris Stoermer ◽  
Dilrukshi Vitharana ◽  
Niyada Hin ◽  
Greg Delahanty ◽  
Bridget Duvall ◽  
...  
Keyword(s):  
Design Synthesis ◽  
Glutamate Carboxypeptidase Ii ◽  
Pharmacological Evaluation ◽  
Glutamate Carboxypeptidase

Design, synthesis and pharmacological evaluation of tricyclic derivatives as selective RXFP4 agonists

2021 ◽  
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Lin Lin ◽  
Guangyao Lin ◽  
Qingtong Zhou ◽  
Ross A.D. Bathgate ◽  
Grace Qun Gong ◽  
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Design Synthesis ◽  
Pharmacological Evaluation

S1 pocket of glutamate carboxypeptidase II: A new binding site for amyloid-β degradation

2013 ◽  
Vol 438 (4) ◽  
pp. 765-771 ◽  
Author(s):  
Suk Kyung Lee ◽  
Hyunyoung Kim ◽  
You-Hoon Cheong ◽  
Min-Ju Kim ◽  
Sangmee Ahn Jo ◽  
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Keyword(s):  
Binding Site ◽  
Amyloid Β ◽  
Glutamate Carboxypeptidase Ii ◽  
Glutamate Carboxypeptidase

Design, Synthesis, and Pharmacological Evaluation of Mefloquine-Based Ligands as Novel Antituberculosis Agents

ChemMedChem ◽  
2007 ◽  
Vol 2 (11) ◽  
pp. 1624-1630 ◽  
Author(s):  
Jialin Mao ◽  
Yuehong Wang ◽  
Baojie Wan ◽  
Alan P. Kozikowski ◽  
Scott G. Franzblau
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Design Synthesis ◽  
Pharmacological Evaluation

Design, synthesis, and pharmacological evaluation of phenoxy pyridyl derivatives as dual norepinephrine reuptake inhibitors and 5-HT1A partial agonists

2010 ◽  
Vol 20 (3) ◽  
pp. 1114-1117 ◽  
Author(s):  
Amy B. Dounay ◽  
Nancy S. Barta ◽  
Brian M. Campbell ◽  
Corey Coleman ◽  
Elizabeth M. Collantes ◽  
...  
Keyword(s):  
Design Synthesis ◽  
Pharmacological Evaluation ◽  
Partial Agonists ◽  
Norepinephrine Reuptake

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2020 ◽  
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Gabriele Carullo ◽  
Amer Ahmed ◽  
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Design Synthesis ◽  
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