Synthesis and Biological Activity of Conformationally Restricted Analogs of Milnacipran:  (1S,2R)-1-Phenyl-2-[(S)-1-aminopropyl]-N,N-diethylcyclopropanecarboxamide, an Efficient NoncompetitiveN-Methyl-d-aspartic Acid Receptor Antagonist

1996 ◽  
Vol 39 (24) ◽  
pp. 4844-4852 ◽  
Author(s):  
Satoshi Shuto ◽  
Shizuka Ono ◽  
Yukako Hase ◽  
Yoshihito Ueno ◽  
Tomohiro Noguchi ◽  
...  
Keyword(s):  
Biological Activity ◽  
Receptor Antagonist ◽  
Aspartic Acid ◽  
Acid Receptor ◽  
Conformationally Restricted ◽  
Conformationally Restricted Analogs

Design of potent ABA receptor antagonists based on a conformational restriction approach

2020 ◽  
Vol 18 (26) ◽  
pp. 4988-4996
Author(s):  
Jun Takeuchi ◽  
Hikaru Nagamiya ◽  
Sayaka Moroi ◽  
Toshiyuki Ohnishi ◽  
Yasushi Todoroki
Keyword(s):  
Abscisic Acid ◽  
Receptor Antagonist ◽  
Receptor Antagonists ◽  
Conformational Restriction ◽  
Acid Receptor ◽  
Conformationally Restricted ◽  
Aba Receptor ◽  
Conformationally Restricted Analogs

Conformationally restricted analogs of (+)-PAO4, an abscisic acid receptor antagonist, were synthesized to improve its potency.

The fibrosis of ketamine, a noncompetitiveN-methyl-d-aspartic acid receptor antagonist dose-dependent change in a ketamine-induced cystitis rat model

2015 ◽  
Vol 39 (2) ◽  
pp. 206-212 ◽  
Author(s):  
Miho Song ◽  
Hwan Yeul Yu ◽  
Ji-Youn Chun ◽  
Dong-Myung Shin ◽  
Soo Hyun Song ◽  
...  
Keyword(s):  
Receptor Antagonist ◽  
Aspartic Acid ◽  
Rat Model ◽  
Acid Receptor ◽  
Dependent Change ◽  
Dose Dependent

N-methyl-d-aspartic acid receptor antagonist–induced frequency oscillations in mice recreate pattern of electrophysiological deficits in schizophrenia

Neuroscience ◽  
2009 ◽  
Vol 158 (2) ◽  
pp. 705-712 ◽  
Author(s):  
R.S. Ehrlichman ◽  
M.J. Gandal ◽  
C.R. Maxwell ◽  
M.T. Lazarewicz ◽  
L.H. Finkel ◽  
...  
Keyword(s):  
Receptor Antagonist ◽  
Aspartic Acid ◽  
Acid Receptor

scholarly journals The N-Methyl-D-Aspartic Acid Receptor Antagonist Memantine Ameliorates and Delays the Development of Arthritis by Enhancing Regulatory T Cells

Neurosignals ◽  
2012 ◽  
Vol 20 (2) ◽  
pp. 61-71 ◽  
Author(s):  
Sofia S. Lindblad ◽  
Piotr Mydel ◽  
Annelie Hellvard ◽  
Ing-Marie Jonsson ◽  
Maria I. Bokarewa
Keyword(s):  
T Cells ◽  
Regulatory T Cells ◽  
Receptor Antagonist ◽  
Aspartic Acid ◽  
Acid Receptor
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