Medetomidine Analogs as α2-Adrenergic Ligands. 2. Design, Synthesis, and Biological Activity of Conformationally Restricted Naphthalene Derivatives of Medetomidine

1996 ◽  
Vol 39 (15) ◽  
pp. 3001-3013 ◽  
Author(s):  
Xiaoyan Zhang ◽  
Xiao-Tao Yao ◽  
James T. Dalton ◽  
Gamal Shams ◽  
Longping Lei ◽  
...  
Keyword(s):  
Biological Activity ◽  
Naphthalene Derivatives ◽  
Design Synthesis ◽  
Conformationally Restricted ◽  
Derivatives Of

scholarly journals Synthesis, characterization and biological activity of organometallic derivatives of the antimalarial drug mefloquine as new antischistosomal drug candidates

MedChemComm ◽  
2018 ◽  
Vol 9 (11) ◽  
pp. 1905-1909 ◽  
Author(s):  
Faustine d'Orchymont ◽  
Jeannine Hess ◽  
Gordana Panic ◽  
Marta Jakubaszek ◽  
Lea Gemperle ◽  
...  
Keyword(s):  
Biological Activity ◽  
Antimalarial Drug ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
Drug Candidates ◽  
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The design, synthesis, characterization and biological evaluation of new ferrocenyl and ruthenocenyl derivatives of the antimalarial mefloquine is described.

scholarly journals Design, Synthesis, and Biological Activity of Conformationally Restricted Analogues of Silibinin

ACS Omega ◽  
2020 ◽  
Vol 5 (36) ◽  
pp. 23164-23174
Author(s):  
Mirei Mizuno ◽  
Kazunori Mori ◽  
Keisuke Tsuchiya ◽  
Takashi Takaki ◽  
Takashi Misawa ◽  
...  
Keyword(s):  
Biological Activity ◽  
Design Synthesis ◽  
Conformationally Restricted

Novel Tetracyclic Spermine Derivatives of Cyclotriphosphazene: Design, Synthesis and Biological Activity

2022 ◽  
pp. 132371
Author(s):  
Gönül Yenilmez Çiftçi ◽  
Sümeyra Yoldaş Kılıç ◽  
Fatma Yuksel ◽  
Gulseren Turhal ◽  
Asuman Demiroglu-Zergeroglu
Keyword(s):  
Biological Activity ◽  
Design Synthesis ◽  
Derivatives Of

Design, synthesis and biological activity of amidinobicyclic compounds (derivatives of DX-9065a) as factor Xa inhibitors: SAR study of S1 and aryl binding sites

2004 ◽  
Vol 12 (9) ◽  
pp. 2099-2114 ◽  
Author(s):  
Satoshi Komoriya ◽  
Naoaki Kanaya ◽  
Takayasu Nagahara ◽  
Asako Yokoyama ◽  
Kazue Inamura ◽  
...  
Keyword(s):  
Biological Activity ◽  
Binding Sites ◽  
Factor Xa ◽  
Factor Xa Inhibitors ◽  
Design Synthesis ◽  
Sar Study ◽  
Derivatives Of
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