scholarly journals Improving Metabolic Stability by Glycosylation: Bifunctional Peptide Derivatives That Are Opioid Receptor Agonists and Neurokinin 1 Receptor Antagonists

2009 ◽  
Vol 52 (16) ◽  
pp. 5164-5175 ◽  
Author(s):  
Takashi Yamamoto ◽  
Padma Nair ◽  
Neil E. Jacobsen ◽  
Josef Vagner ◽  
Vinod Kulkarni ◽  
...  
Keyword(s):  
Opioid Receptor ◽  
Metabolic Stability ◽  
Receptor Antagonists ◽  
Neurokinin 1 Receptor ◽  
Receptor Agonists ◽  
Peptide Derivatives ◽  
Neurokinin 1 ◽  
Opioid Receptor Agonists

Transformation of μ-opioid receptor agonists into biologically potent μ-opioid receptor antagonists

2007 ◽  
Vol 15 (3) ◽  
pp. 1237-1251 ◽  
Author(s):  
Tingyou Li ◽  
Yunden Jinsmaa ◽  
Masahiro Nedachi ◽  
Anna Miyazaki ◽  
Yuko Tsuda ◽  
...  
Keyword(s):  
Opioid Receptor ◽  
Receptor Antagonists ◽  
Receptor Agonists ◽  
Opioid Receptor Antagonists ◽  
Μ Opioid Receptor ◽  
Opioid Receptor Agonists

New Diarylmethylpiperazines as Potent and Selective Nonpeptidic δ Opioid Receptor Agonists with Increased In Vitro Metabolic Stability

2000 ◽  
Vol 43 (21) ◽  
pp. 3878-3894 ◽  
Author(s):  
Niklas Plobeck ◽  
Daniel Delorme ◽  
Zhong-Yong Wei ◽  
Hua Yang ◽  
Fei Zhou ◽  
...  
Keyword(s):  
Opioid Receptor ◽  
Metabolic Stability ◽  
Receptor Agonists ◽  
Δ Opioid Receptor ◽  
Opioid Receptor Agonists
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