Discovery of 4-Substituted Methoxybenzoyl-aryl-thiazole as Novel Anticancer Agents: Synthesis, Biological Evaluation, and Structure−Activity Relationships

Yan Lu; Chien-Ming Li; Zhao Wang; Charles R. Ross; Jianjun Chen; James T. Dalton; Wei Li; Duane D. Miller

doi:10.1021/jm801449a

Discovery of 4-Substituted Methoxybenzoyl-aryl-thiazole as Novel Anticancer Agents: Synthesis, Biological Evaluation, and Structure−Activity Relationships

Journal of Medicinal Chemistry ◽

10.1021/jm801449a ◽

2009 ◽

Vol 52 (6) ◽

pp. 1701-1711 ◽

Cited By ~ 108

Author(s):

Yan Lu ◽

Chien-Ming Li ◽

Zhao Wang ◽

Charles R. Ross ◽

Jianjun Chen ◽

...

Keyword(s):

Anticancer Agents ◽

Biological Evaluation ◽

Structure Activity Relationships ◽

Structure Activity

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Selective and effective anticancer agents: Synthesis, biological evaluation and structure-activity relationships of novel carbazole derivatives

Bioorganic Chemistry ◽

10.1016/j.bioorg.2021.104991 ◽

2021 ◽

pp. 104991

Author(s):

Wenbo Huang ◽

Zilin Gao ◽

Zhigang Zhang ◽

Wei Fang ◽

Zuoqian Wang ◽

...

Keyword(s):

Anticancer Agents ◽

Biological Evaluation ◽

Carbazole Derivatives ◽

Structure Activity Relationships ◽

Structure Activity

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5-Cinnamoyl-6-aminouracil derivatives as novel anticancer agents. Synthesis, biological evaluation, and structure-activity relationships

Journal of Medicinal Chemistry ◽

10.1021/jm00382a020 ◽

1985 ◽

Vol 28 (4) ◽

pp. 497-502 ◽

Cited By ~ 20

Author(s):

Jean Luc Bernier ◽

Jean Pierre Henichart ◽

Vincent Warin ◽

Chantal Trentesaux ◽

Jean Claude Jardillier

Keyword(s):

Anticancer Agents ◽

Biological Evaluation ◽

Structure Activity Relationships ◽

Structure Activity

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ChemInform Abstract: 5-CINNAMOYL-6-AMINOURACIL DERIVATIVES AS NOVEL ANTICANCER AGENTS. SYNTHESIS, BIOLOGICAL EVALUATION, AND STRUCTURE-ACTIVITY RELATIONSHIPS

Chemischer Informationsdienst ◽

10.1002/chin.198531245 ◽

1985 ◽

Vol 16 (31) ◽

Author(s):

J.-C. BERNIER ◽

J.-P. HENICHART ◽

V. WARIN ◽

C. TRENTESAUX ◽

J.-C. JARDILLIER

Keyword(s):

Anticancer Agents ◽

Biological Evaluation ◽

Structure Activity Relationships ◽

Structure Activity

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Additions and Corrections - 5-Cinnamoyl-6-aminouracil Derivatives as Novel Anticancer Agents. Synthesis, Biological Evaluation, and Structure-Activity Relationships.

Journal of Medicinal Chemistry ◽

10.1021/jm00150a602 ◽

1985 ◽

Vol 28 (12) ◽

pp. 1965-1965

Author(s):

Jean-Luc Bernier ◽

Jean-Pierre Henichart ◽

Vincent Warin ◽

Chantal Trentesaux ◽

Jean-Claude Jardillier

Keyword(s):

Anticancer Agents ◽

Biological Evaluation ◽

Structure Activity Relationships ◽

Structure Activity

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1,3,4-Oxadiazole-containing Hybrids as Potential Anticancer Agents: Recent Developments, Mechanism of Action and Structure-Activity Relationships

Journal of Saudi Chemical Society ◽

10.1016/j.jscs.2021.101284 ◽

2021 ◽

pp. 101284

Author(s):

Swarnagowri Nayak ◽

Santosh L. Gaonkar ◽

Ebraheem Abdu Musad ◽

Abdullah Mohammed AL. Dawsar

Keyword(s):

Mechanism Of Action ◽

Anticancer Agents ◽

Structure Activity Relationships ◽

Structure Activity ◽

Recent Developments

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Synthesis and Biological Evaluation of 14-Alkoxymorphinans. 18.1N-Substituted 14-Phenylpropyloxymorphinan-6-ones with Unanticipated Agonist Properties: Extending the Scope of Common Structure−Activity Relationships

Journal of Medicinal Chemistry ◽

10.1021/jm021118o ◽

2003 ◽

Vol 46 (9) ◽

pp. 1758-1763 ◽

Cited By ~ 23

Author(s):

Elisabeth Greiner ◽

Mariana Spetea ◽

Roland Krassnig ◽

Falko Schüllner ◽

Mario Aceto ◽

...

Keyword(s):

Biological Evaluation ◽

Structure Activity Relationships ◽

Common Structure ◽

Structure Activity ◽

Synthesis And Biological Evaluation

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Back Cover: Photochemical Properties and Structure-Activity Relationships of RuII Complexes with Pyridylbenzazole Ligands as Promising Anticancer Agents (Eur. J. Inorg. Chem. 12/2017)

European Journal of Inorganic Chemistry ◽

10.1002/ejic.201700259 ◽

2017 ◽

Vol 2017 (12) ◽

pp. 1842-1842

Author(s):

Dmytro Havrylyuk ◽

David K. Heidary ◽

Leona Nease ◽

Sean Parkin ◽

Edith C. Glazer

Keyword(s):

Anticancer Agents ◽

Back Cover ◽

Structure Activity Relationships ◽

Structure Activity ◽

Photochemical Properties

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125 Synthesis, biological evaluation and structure activity relationships of a novel servies of aromatic hydroxamic acids as potent HDAC inhibitors

European Journal of Cancer Supplements ◽

10.1016/s1359-6349(04)80133-2 ◽

2004 ◽

Vol 2 (8) ◽

pp. 40-41

Author(s):

K. Van Emelen ◽

J. Arts ◽

P. Angibaud ◽

H. De Winter ◽

S. Van Brandt ◽

...

Keyword(s):

Hdac Inhibitors ◽

Hydroxamic Acids ◽

Biological Evaluation ◽

Structure Activity Relationships ◽

Structure Activity

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Biological Evaluation, Structure−Activity Relationships, and Three-Dimensional Quantitative Structure−Activity Relationship Studies of Dihydro-β-agarofuran Sesquiterpenes as Modulators of P-Glycoprotein-Dependent Multidrug Resistance

Journal of Medicinal Chemistry ◽

10.1021/jm070290v ◽

2007 ◽

Vol 50 (20) ◽

pp. 4808-4817 ◽

Cited By ~ 30

Author(s):

Carolina P. Reyes ◽

Francisco Muñoz-Martínez ◽

Ivan R. Torrecillas ◽

Cristina R. Mendoza ◽

Francisco Gamarro ◽

...

Keyword(s):

Multidrug Resistance ◽

Three Dimensional ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Biological Evaluation ◽

Activity Relationship ◽

Quantitative Structure ◽

Structure Activity Relationships ◽

Structure Activity ◽

P Glycoprotein

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Synthesis, Biological Evaluation, and Structure−Activity Relationships of 3-Acylindole-2-carboxylic Acids as Inhibitors of the Cytosolic Phospholipase A2

Journal of Medicinal Chemistry ◽

10.1021/jm960863w ◽

1997 ◽

Vol 40 (17) ◽

pp. 2694-2705 ◽

Cited By ~ 20

Author(s):

Matthias Lehr

Keyword(s):

Phospholipase A2 ◽

Carboxylic Acids ◽

Biological Evaluation ◽

Cytosolic Phospholipase A2 ◽

Structure Activity Relationships ◽

Cytosolic Phospholipase ◽

Structure Activity

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