Design, Synthesis, and Biological Activity of a Novel Series of Human Sirtuin-2-Selective Inhibitors

2012 ◽  
Vol 55 (12) ◽  
pp. 5760-5773 ◽  
Author(s):  
Takayoshi Suzuki ◽  
Mohammed Naseer Ahmed Khan ◽  
Hideyuki Sawada ◽  
Erika Imai ◽  
Yukihiro Itoh ◽  
...  
Keyword(s):  
Biological Activity ◽  
Selective Inhibitors ◽  
Design Synthesis

scholarly journals Design, synthesis and biological activity of sphingosine kinase 2 selective inhibitors

2012 ◽  
Vol 20 (1) ◽  
pp. 183-194 ◽  
Author(s):  
Mithun R. Raje ◽  
Kenneth Knott ◽  
Yugesh Kharel ◽  
Philippe Bissel ◽  
Kevin R. Lynch ◽  
...  
Keyword(s):  
Biological Activity ◽  
Sphingosine Kinase ◽  
Selective Inhibitors ◽  
Design Synthesis ◽  
Sphingosine Kinase 2

Design, synthesis, and biological activity of potent and selective inhibitors of mast cell tryptase

2005 ◽  
Vol 15 (11) ◽  
pp. 2734-2737 ◽  
Author(s):  
Corey R. Hopkins ◽  
Mark Czekaj ◽  
Steven S. Kaye ◽  
Zhongli Gao ◽  
James Pribish ◽  
...  
Keyword(s):  
Mast Cell ◽  
Biological Activity ◽  
Selective Inhibitors ◽  
Mast Cell Tryptase ◽  
Design Synthesis

Design, Synthesis, and Biological Activity of Potent and Selective Inhibitors of Blood Coagulation Factor Xa

2004 ◽  
Vol 47 (16) ◽  
pp. 4089-4099 ◽  
Author(s):  
J. Adam Willardsen ◽  
Danette A. Dudley ◽  
Wayne L. Cody ◽  
Liguo Chi ◽  
Thomas B. McClanahan ◽  
...  
Keyword(s):  
Biological Activity ◽  
Blood Coagulation ◽  
Factor Xa ◽  
Coagulation Factor ◽  
Selective Inhibitors ◽  
Design Synthesis

Design, Synthesis, and Biological Activity of NCC149 Derivatives as Histone Deacetylase 8-Selective Inhibitors

ChemMedChem ◽  
2014 ◽  
Vol 9 (3) ◽  
pp. 657-664 ◽  
Author(s):  
Takayoshi Suzuki ◽  
Nobusuke Muto ◽  
Masashige Bando ◽  
Yukihiro Itoh ◽  
Ayako Masaki ◽  
...  
Keyword(s):  
Biological Activity ◽  
Histone Deacetylase ◽  
Selective Inhibitors ◽  
Design Synthesis ◽  
Histone Deacetylase 8

Design, Synthesis and Biological Activity of Aromatic Diketone Derivatives as HIV-1 Integrase Inhibitors

2015 ◽  
Vol 11 (2) ◽  
pp. 180-187 ◽  
Author(s):  
Liming Hu ◽  
Zhipeng Li ◽  
Zhanyang Wang ◽  
Gengxin Liu ◽  
Xianzhuo He ◽  
...  
Keyword(s):  
Biological Activity ◽  
Integrase Inhibitors ◽  
Design Synthesis ◽  
Hiv 1

scholarly journals Synthesis, characterization and biological activity of organometallic derivatives of the antimalarial drug mefloquine as new antischistosomal drug candidates

MedChemComm ◽  
2018 ◽  
Vol 9 (11) ◽  
pp. 1905-1909 ◽  
Author(s):  
Faustine d'Orchymont ◽  
Jeannine Hess ◽  
Gordana Panic ◽  
Marta Jakubaszek ◽  
Lea Gemperle ◽  
...  
Keyword(s):  
Biological Activity ◽  
Antimalarial Drug ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
Drug Candidates ◽  
Derivatives Of

The design, synthesis, characterization and biological evaluation of new ferrocenyl and ruthenocenyl derivatives of the antimalarial mefloquine is described.

1-Methyl-3H-pyrazolo[1,2-a]benzo[1,2,3,4]tetrazin-3-ones. Design, Synthesis, and Biological Activity of New Antitumor Agents

2005 ◽  
Vol 48 (8) ◽  
pp. 2859-2866 ◽  
Author(s):  
Anna Maria Almerico ◽  
Francesco Mingoia ◽  
Patrizia Diana ◽  
Paola Barraja ◽  
Antonino Lauria ◽  
...  
Keyword(s):  
Biological Activity ◽  
Antitumor Agents ◽  
Design Synthesis
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