Design, Synthesis, and Biological Activity of Potent and Orally Available G Protein-Coupled Receptor 40 Agonists

2011 ◽  
Vol 54 (5) ◽  
pp. 1365-1378 ◽  
Author(s):  
Shinobu Sasaki ◽  
Shuji Kitamura ◽  
Nobuyuki Negoro ◽  
Masami Suzuki ◽  
Yoshiyuki Tsujihata ◽  
...  
Keyword(s):  
Biological Activity ◽  
G Protein ◽  
G Protein Coupled Receptor ◽  
Design Synthesis ◽  
G Protein Coupled

Design, synthesis and efficacy of novel G protein-coupled receptor kinase 2 inhibitors

2013 ◽  
Vol 69 ◽  
pp. 384-392 ◽  
Author(s):  
Alfonso Carotenuto ◽  
Ersilia Cipolletta ◽  
Isabel Gomez-Monterrey ◽  
Marina Sala ◽  
Ermelinda Vernieri ◽  
...  
Keyword(s):  
G Protein ◽  
Receptor Kinase ◽  
G Protein Coupled Receptor ◽  
Design Synthesis ◽  
G Protein Coupled

scholarly journals Design, Synthesis, and Evaluation of Novel and Selective G-protein Coupled Receptor 120 (GPR120) Spirocyclic Agonists

2016 ◽  
Vol 8 (1) ◽  
pp. 49-54 ◽  
Author(s):  
Jason M. Cox ◽  
Hong D. Chu ◽  
Mariappan V. Chelliah ◽  
John S. Debenham ◽  
Keith Eagen ◽  
...  
Keyword(s):  
G Protein ◽  
G Protein Coupled Receptor ◽  
Design Synthesis ◽  
G Protein Coupled

Design, Synthesis, and Evaluation of N- and C-Terminal Protein Bioconjugates as G Protein-Coupled Receptor Agonists

2018 ◽  
Vol 29 (2) ◽  
pp. 403-409
Author(s):  
Robert D. Healey ◽  
Jonathan P. Wojciechowski ◽  
Ana Monserrat-Martinez ◽  
Susan L. Tan ◽  
Christopher P. Marquis ◽  
...  
Keyword(s):  
G Protein ◽  
G Protein Coupled Receptor ◽  
Terminal Protein ◽  
Design Synthesis ◽  
Receptor Agonists ◽  
G Protein Coupled

scholarly journals Structure-Based Design, Synthesis, and Biological Evaluation of Highly Selective and Potent G Protein-Coupled Receptor Kinase 2 Inhibitors

2016 ◽  
Vol 59 (8) ◽  
pp. 3793-3807 ◽  
Author(s):  
Helen V. Waldschmidt ◽  
Kristoff T. Homan ◽  
Osvaldo Cruz-Rodríguez ◽  
Marilyn C. Cato ◽  
Jessica Waninger-Saroni ◽  
...  
Keyword(s):  
G Protein ◽  
Biological Evaluation ◽  
Receptor Kinase ◽  
G Protein Coupled Receptor ◽  
Design Synthesis ◽  
G Protein Coupled ◽  
Synthesis And Biological Evaluation

Design, synthesis and evaluation of potent G-protein coupled receptor 40 agonists

2016 ◽  
Vol 27 (1) ◽  
pp. 159-162 ◽  
Author(s):  
Jing Huang ◽  
Bin Guo ◽  
Wen-Jing Chu ◽  
Xin Xie ◽  
Yu-She Yang ◽  
...  
Keyword(s):  
G Protein ◽  
G Protein Coupled Receptor ◽  
Design Synthesis ◽  
G Protein Coupled

G-Protein-Coupled Receptor Affinity Prediction Based on the Use of a Profiling Dataset:  QSAR Design, Synthesis, and Experimental Validation

2005 ◽  
Vol 48 (21) ◽  
pp. 6563-6574 ◽  
Author(s):  
Catherine Rolland ◽  
Rafael Gozalbes ◽  
Eric Nicolaï ◽  
Marie-France Paugam ◽  
Laurent Coussy ◽  
...  
Keyword(s):  
G Protein ◽  
Experimental Validation ◽  
G Protein Coupled Receptor ◽  
Design Synthesis ◽  
Receptor Affinity ◽  
Affinity Prediction ◽  
G Protein Coupled
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