Design, Synthesis, DNA Binding, and Biological Evaluation of Water-Soluble Hybrid Molecules Containing Two Pyrazole Analogues of the Alkylating Cyclopropylpyrroloindole (CPI) Subunit of the Antitumor Agent CC-1065 and Polypyrrole Minor Groove Binders

2001 ◽  
Vol 44 (16) ◽  
pp. 2536-2543 ◽  
Author(s):  
Pier Giovanni Baraldi ◽  
Gianfrano Balboni ◽  
Maria Giovanna Pavani ◽  
Giampiero Spalluto ◽  
Mojgan Aghazadeh Tabrizi ◽  
...  
Keyword(s):  
Dna Binding ◽  
Antitumor Agent ◽  
Minor Groove ◽  
Biological Evaluation ◽  
Water Soluble ◽  
Design Synthesis ◽  
Minor Groove Binders ◽  
Hybrid Molecules ◽  
Groove Binders

Design, Synthesis, and Biological Evaluation of Hybrid Molecules Containing α-Methylene-γ-butyrolactones and Polypyrrole Minor Groove Binders

2004 ◽  
Vol 47 (11) ◽  
pp. 2877-2886 ◽  
Author(s):  
Pier Giovanni Baraldi ◽  
Maria del Carmen Nunez ◽  
Mojgan Aghazadeh Tabrizi ◽  
Erik De Clercq ◽  
Jan Balzarini ◽  
...  
Keyword(s):  
Minor Groove ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
Minor Groove Binders ◽  
Hybrid Molecules ◽  
Groove Binders ◽  
Synthesis And Biological Evaluation

Aromatic analogues of DNA minor groove binders—synthesis and biological evaluation

2004 ◽  
Vol 39 (1) ◽  
pp. 99-105 ◽  
Author(s):  
Anna Pućkowska ◽  
Krzysztof Bielawski ◽  
Anna Bielawska ◽  
Krystyna Midura-Nowaczek
Keyword(s):  
Minor Groove ◽  
Biological Evaluation ◽  
Dna Minor Groove ◽  
Minor Groove Binders ◽  
Groove Binders ◽  
Synthesis And Biological Evaluation

scholarly journals Design, synthesis and antibacterial activity of minor groove binders: The role of non-cationic tail groups

2012 ◽  
Vol 56 ◽  
pp. 39-47 ◽  
Author(s):  
Abedawn I. Khalaf ◽  
Claire Bourdin ◽  
David Breen ◽  
Gavin Donoghue ◽  
Fraser J. Scott ◽  
...  
Keyword(s):  
Antibacterial Activity ◽  
Minor Groove ◽  
Design Synthesis ◽  
Minor Groove Binders ◽  
Groove Binders

Sequence-Specific Conjugates of Oligo(2′-O-methylribonucleotides) and Hairpin Oligocarboxamide Minor-Groove Binders: Design, Synthesis, and Binding Studies with Double-Stranded DNA

2005 ◽  
Vol 2 (7) ◽  
pp. 936-952 ◽  
Author(s):  
Darya S. Novopashina ◽  
Alexandre N. Sinyakov ◽  
Vladimir A. Ryabinin ◽  
Alya G. Venyaminova ◽  
Ludovic Halby ◽  
...  
Keyword(s):  
Minor Groove ◽  
Binding Studies ◽  
Design Synthesis ◽  
Minor Groove Binders ◽  
Double Stranded Dna ◽  
Groove Binders

scholarly journals Synthesis, Biological Evaluation, and Modeling of Dimeric PPI Analogues as Novel DNA Minor Groove Binders

Molecules ◽  
2008 ◽  
Vol 13 (5) ◽  
pp. 1179-1188
Author(s):  
Yan-Hui Yang ◽  
Qing-He Wang ◽  
Han Nie ◽  
Hong Chen ◽  
Mao-Sheng Cheng
Keyword(s):  
Minor Groove ◽  
Biological Evaluation ◽  
Dna Minor Groove ◽  
Minor Groove Binders ◽  
Groove Binders

Dithiocarbamate/piperazine bridged pyrrolobenzodiazepines as DNA-minor groove binders: Synthesis, DNA-binding affinity and cytotoxic activity

2015 ◽  
Vol 59 ◽  
pp. 23-30 ◽  
Author(s):  
Ahmed Kamal ◽  
Kokkonda Sreekanth ◽  
Nagula Shankaraiah ◽  
Manda Sathish ◽  
Shalini Nekkanti ◽  
...  
Keyword(s):  
Dna Binding ◽  
Cytotoxic Activity ◽  
Binding Affinity ◽  
Minor Groove ◽  
Dna Minor Groove ◽  
Minor Groove Binders ◽  
Dna Binding Affinity ◽  
Groove Binders
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