Diastereomeric 6-desoxy-6-spiro-.alpha.-methylene-.gamma.-butyrolactone derivatives of naltrexone and oxymorphone. Selective irreversible inhibition of naltrexone binding in an opioid receptor preparation by a conformationally restricted Michael acceptor ligand

1984 ◽  
Vol 27 (12) ◽  
pp. 1718-1723 ◽  
Author(s):  
Gary A. Koolpe ◽  
Wendel L. Nelson ◽  
T. L. Gioannini ◽  
Lloyd Angel ◽  
Eric J. Simon
Keyword(s):  
Opioid Receptor ◽  
Conformationally Restricted ◽  
Irreversible Inhibition ◽  
Michael Acceptor ◽  
Derivatives Of ◽  
Gamma Butyrolactone

ChemInform Abstract: Derivatives of 17-(2-Methylallyl)-substituted Noroxymorphone: Variation of the Delta Address and Its Effects on Affinity and Selectivity for the Delta Opioid Receptor.

ChemInform ◽  
2010 ◽  
Vol 33 (8) ◽  
pp. no-no
Author(s):  
Thomas Ullrich ◽  
Christina M. Dersch ◽  
Richard B. Rothman ◽  
Arthur E. Jacobson ◽  
Kenner C. Rice
Keyword(s):  
Opioid Receptor ◽  
Delta Opioid Receptor ◽  
Derivatives Of

14β-Chlorocinnamoylamino derivatives of metopon interact differentially with the mu opioid receptor

1994 ◽  
Vol 54 (1) ◽  
pp. 187-188 ◽  
Author(s):  
J.P. McLaughlin ◽  
A. Sebastian ◽  
S. Archer ◽  
J.M. Bidlack
Keyword(s):  
Opioid Receptor ◽  
Mu Opioid Receptor ◽  
Mu Opioid ◽  
Derivatives Of
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