Potential inhibitors of nucleotide biosynthesis. 2. Halomethyl ketone derivatives of pyrimidine nucleosides

1984 ◽  
Vol 27 (5) ◽  
pp. 680-684 ◽  
Author(s):  
John A. Montgomery ◽  
H. Jeanette Thomas ◽  
R. Wallace Brockman ◽  
Robert D. Elliott
Keyword(s):  
Nucleotide Biosynthesis ◽  
Pyrimidine Nucleosides ◽  
Potential Inhibitors ◽  
Derivatives Of

Analogs of pyrimidine nucleosides. 14. Synthesis and antitumorigenic activity of alkoxyalkyl derivatives of 5-fluorouracil

1980 ◽  
Vol 16 (11) ◽  
pp. 1176-1179 ◽  
Author(s):  
M. Ya. Karpeiskii ◽  
S. M. Mikhailov ◽  
A. S. Tsieminya ◽  
A. A. Ziderman ◽  
I. M. Kravchenko ◽  
...  
Keyword(s):  
Antitumorigenic Activity ◽  
Pyrimidine Nucleosides ◽  
Derivatives Of

Phosphonate monoesters on a thiacalix[4]arene framework as potential inhibitors of protein tyrosine phosphatase 1B

2015 ◽  
Vol 13 (33) ◽  
pp. 8803-8806 ◽  
Author(s):  
Viacheslav V. Trush ◽  
Sergiy G. Kharchenko ◽  
Vsevolod Yu. Tanchuk ◽  
Vitaly I. Kalchenko ◽  
Andriy I. Vovk
Keyword(s):  
Human Serum Albumin ◽  
Serum Albumin ◽  
Human Serum ◽  
Protein Tyrosine Phosphatase ◽  
Tyrosine Phosphatase ◽  
Methylphosphonic Acid ◽  
Protein Tyrosine Phosphatase 1B ◽  
Protein Tyrosine ◽  
Potential Inhibitors ◽  
Derivatives Of

Monoester derivatives of thiacalix[4]arene tetrakis(methylphosphonic) acid were found to be capable of inhibiting protein tyrosine phosphatase 1B. In addition, these compounds can strongly bind to human serum albumin.

PHOSPHORAMIDATE DERIVATIVES OF 2′,5′-DIDEOXYADENOSINE AS POTENTIAL INHIBITORS OF THE EDHF PHENOMENON

2005 ◽  
Vol 24 (5-7) ◽  
pp. 553-555 ◽  
Author(s):  
F. Gavazza ◽  
F. Daverio ◽  
A. T. Chaytor ◽  
T. M. Griffith ◽  
C. McGuigan
Keyword(s):  
Potential Inhibitors ◽  
Derivatives Of
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