Structure-activity relationships among DNA gyrase inhibitors. Synthesis and biological evaluation of 1,2-dihydro-4,4-dimethyl-1-oxo-2-naphthalenecarboxylic acids as 1-carba bioisosteres of oxolinic acid

1984 ◽  
Vol 27 (3) ◽  
pp. 306-310 ◽  
Author(s):  
Thomas Hogberg ◽  
Ish Khanna ◽  
Steven D. Drake ◽  
Lester A. Mitscher ◽  
Linus L. Shen
Keyword(s):  
Dna Gyrase ◽  
Biological Evaluation ◽  
Oxolinic Acid ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
Synthesis And Biological Evaluation ◽  
Gyrase Inhibitors

Taxol structure-activity relationships: synthesis and biological evaluation of 10-deoxytaxol

1993 ◽  
Vol 58 (11) ◽  
pp. 2927-2928 ◽  
Author(s):  
Shu Hui Chen ◽  
Craig Fairchild ◽  
Stephen W. Mamber ◽  
Vittorio Farina
Keyword(s):  
Biological Evaluation ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
Synthesis And Biological Evaluation

scholarly journals Design, synthesis and biological evaluation of 4,5-dibromo-N-(thiazol-2-yl)-1H-pyrrole-2-carboxamide derivatives as novel DNA gyrase inhibitors

2017 ◽  
Vol 25 (1) ◽  
pp. 338-349 ◽  
Author(s):  
Tihomir Tomašič ◽  
Matic Mirt ◽  
Michaela Barančoková ◽  
Janez Ilaš ◽  
Nace Zidar ◽  
...  
Keyword(s):  
Dna Gyrase ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
Synthesis And Biological Evaluation ◽  
Gyrase Inhibitors
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