Structure–activity relationships in platelet-activating factor. Part 13: Synthesis and biological evaluation of piperazine derivatives with dual anti-PAF and anti-HIV-1 or pure antiretroviral activity

Nawal Serradji; Okkacha Bensaid; Marc Martin; Wafa Sallem; Nathalie Dereuddre-Bosquet; Houcine Benmehdi; Catherine Redeuilh; Aazdine Lamouri; Georges Dive; Pascal Clayette; Françoise Heymans

doi:10.1016/j.bmc.2006.07.031

Structure–activity relationships in platelet-activating factor. Part 13: Synthesis and biological evaluation of piperazine derivatives with dual anti-PAF and anti-HIV-1 or pure antiretroviral activity

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2006.07.031 ◽

2006 ◽

Vol 14 (23) ◽

pp. 8109-8125 ◽

Cited By ~ 13

Author(s):

Nawal Serradji ◽

Okkacha Bensaid ◽

Marc Martin ◽

Wafa Sallem ◽

Nathalie Dereuddre-Bosquet ◽

...

Keyword(s):

Platelet Activating Factor ◽

Biological Evaluation ◽

Structure Activity Relationships ◽

Piperazine Derivatives ◽

Structure Activity ◽

Synthesis And Biological Evaluation ◽

Anti Hiv ◽

Hiv 1 ◽

Antiretroviral Activity

Download Full-text

Structure–activity relationships in platelet-activating factor. Part 14: Synthesis and biological evaluation of piperazine derivatives with dual anti-PAF and anti-HIV-1 activity

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2006.07.043 ◽

2006 ◽

Vol 14 (23) ◽

pp. 7999-8013 ◽

Cited By ~ 10

Author(s):

Wafa Sallem ◽

Nawal Serradji ◽

Nathalie Dereuddre-Bosquet ◽

Georges Dive ◽

Pascal Clayette ◽

...

Keyword(s):

Platelet Activating Factor ◽

Biological Evaluation ◽

Structure Activity Relationships ◽

Piperazine Derivatives ◽

Structure Activity ◽

Synthesis And Biological Evaluation ◽

Anti Hiv ◽

Hiv 1

Download Full-text

Structure−Activity Relationships in Platelet-Activating Factor. 12. Synthesis and Biological Evaluation of Platelet-Activating Factor Antagonists with Anti-HIV-1 Activity

Journal of Medicinal Chemistry ◽

10.1021/jm040860g ◽

2004 ◽

Vol 47 (25) ◽

pp. 6410-6419 ◽

Cited By ~ 12

Author(s):

Nawal Serradji ◽

Marc Martin ◽

Okkacha Bensaid ◽

Salvatore Cisternino ◽

Christophe Rousselle ◽

...

Keyword(s):

Platelet Activating Factor ◽

Biological Evaluation ◽

Structure Activity Relationships ◽

Structure Activity ◽

Synthesis And Biological Evaluation ◽

Anti Hiv ◽

Hiv 1

Download Full-text

Synthesis and Biological Evaluation of 14-Alkoxymorphinans. 18.1N-Substituted 14-Phenylpropyloxymorphinan-6-ones with Unanticipated Agonist Properties: Extending the Scope of Common Structure−Activity Relationships

Journal of Medicinal Chemistry ◽

10.1021/jm021118o ◽

2003 ◽

Vol 46 (9) ◽

pp. 1758-1763 ◽

Cited By ~ 23

Author(s):

Elisabeth Greiner ◽

Mariana Spetea ◽

Roland Krassnig ◽

Falko Schüllner ◽

Mario Aceto ◽

...

Keyword(s):

Biological Evaluation ◽

Structure Activity Relationships ◽

Common Structure ◽

Structure Activity ◽

Synthesis And Biological Evaluation

Download Full-text

Synthesis and Biological Evaluation of 8-Hydroxyquinoline-hydrazones for Anti-HIV-1 and Anticancer Potential

ChemistrySelect ◽

10.1002/slct.201802283 ◽

2018 ◽

Vol 3 (38) ◽

pp. 10727-10731 ◽

Cited By ~ 5

Author(s):

Purvi Shah ◽

Leila F. Abadi ◽

Shraddha Gaikwad ◽

Dasharath Chaudhari ◽

Varun Kushwah ◽

...

Keyword(s):

Biological Evaluation ◽

Synthesis And Biological Evaluation ◽

Anti Hiv ◽

Hiv 1

Download Full-text

Taxol structure-activity relationships: synthesis and biological evaluation of 10-deoxytaxol

The Journal of Organic Chemistry ◽

10.1021/jo00063a001 ◽

1993 ◽

Vol 58 (11) ◽

pp. 2927-2928 ◽

Cited By ~ 32

Author(s):

Shu Hui Chen ◽

Craig Fairchild ◽

Stephen W. Mamber ◽

Vittorio Farina

Keyword(s):

Biological Evaluation ◽

Structure Activity Relationships ◽

Structure Activity ◽

Synthesis And Biological Evaluation

Download Full-text

ChemInform Abstract: Structure-Activity Relationships Among DNA Gyrase Inhibitors. Synthesis and Biological Evaluation of 1,2-Dihydro-4,4-dimethyl-1-oxo-2-naphthalenecarboxylic Acids as 1-Carba Bioisosteres of Oxolinic Acid.

Chemischer Informationsdienst ◽

10.1002/chin.198432158 ◽

1984 ◽

Vol 15 (32) ◽

Author(s):

T. HOEGBERG ◽

I. KHANNA ◽

S. D. DRAKE ◽

L. A. MITSCHER ◽

L. L. SHEN

Keyword(s):

Dna Gyrase ◽

Biological Evaluation ◽

Oxolinic Acid ◽

Structure Activity Relationships ◽

Structure Activity ◽

Abstract Structure ◽

Synthesis And Biological Evaluation ◽

Gyrase Inhibitors

Download Full-text

Structure−Activity Relationships of 2‘-Fluoro-2‘,3‘-unsaturatedd-Nucleosides as Anti-HIV-1 Agents

Journal of Medicinal Chemistry ◽

10.1021/jm010418n ◽

2002 ◽

Vol 45 (6) ◽

pp. 1313-1320 ◽

Cited By ~ 31

Author(s):

Kyeong Lee ◽

Yongseok Choi ◽

Giuseppe Gumina ◽

Wen Zhou ◽

Raymond F. Schinazi ◽

...

Keyword(s):

Structure Activity Relationships ◽

Structure Activity ◽

Anti Hiv ◽

Hiv 1

Download Full-text

Synthesis and biological evaluation of substituted 2-benzoylpyridine thiosemicarbazones: Novel structure–activity relationships underpinning their anti-proliferative and chelation efficacy

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2012.12.044 ◽

2013 ◽

Vol 23 (4) ◽

pp. 967-974 ◽

Cited By ~ 28

Author(s):

Adeline Y. Lukmantara ◽

Danuta S. Kalinowski ◽

Naresh Kumar ◽

Des R. Richardson

Keyword(s):

Biological Evaluation ◽

Structure Activity Relationships ◽

Structure Activity ◽

Novel Structure ◽

Synthesis And Biological Evaluation

Download Full-text

Design, synthesis and biological evaluation of heteroaryl diketohexenoic and diketobutanoic acids as HIV-1 integrase inhibitors endowed with antiretroviral activity

Il Farmaco ◽

10.1016/j.farmac.2005.03.008 ◽

2005 ◽

Vol 60 (5) ◽

pp. 409-417 ◽

Cited By ~ 20

Author(s):

R. Di Santo ◽

R. Costi ◽

M. Artico ◽

R. Ragno ◽

G. Greco ◽

...

Keyword(s):

Biological Evaluation ◽

Integrase Inhibitors ◽

Design Synthesis ◽

Synthesis And Biological Evaluation ◽

Hiv 1 ◽

Antiretroviral Activity

Download Full-text

ChemInform Abstract: Structure-Activity Relationships Study at the 3′-N Position of Paclitaxel. Part 1. Synthesis and Biological Evaluation of the 3′-(t)-Butylaminocarbonyloxy Bearing Paclitaxel Analogues.

ChemInform ◽

10.1002/chin.199812164 ◽

2010 ◽

Vol 29 (12) ◽

pp. no-no

Author(s):

S.-H. CHEN ◽

M. XUE ◽

S. HUANG ◽

B. H. LONG ◽

C. A. FAIRCHILD ◽

...

Keyword(s):

Biological Evaluation ◽

Structure Activity Relationships ◽

Structure Activity ◽

Abstract Structure ◽

Synthesis And Biological Evaluation

Download Full-text