The Development of Cyclic Sulfolanes as Novel and High-Affinity P2 Ligands for HIV-1 Protease Inhibitors

1994 ◽  
Vol 37 (8) ◽  
pp. 1177-1188 ◽  
Author(s):  
Arun K. Ghosh ◽  
Hee Yoon Lee ◽  
Wayne J. Thompson ◽  
Chris Culberson ◽  
M. Katharine Holloway ◽  
...  
Keyword(s):  
Protease Inhibitors ◽  
High Affinity ◽  
Hiv 1

ChemInform Abstract: The Development of Cyclic Sulfolanes as Novel and High-Affinity P2 Ligands for HIV-1 Protease Inhibitors.

ChemInform ◽  
2010 ◽  
Vol 25 (33) ◽  
pp. no-no
Author(s):  
A. K. GHOSH ◽  
H. Y. LEE ◽  
W. J. THOMPSON ◽  
C. CULBERSON ◽  
M. K. HOLLOWAY ◽  
...  
Keyword(s):  
Protease Inhibitors ◽  
High Affinity ◽  
Hiv 1

scholarly journals Asymmetric Diels–Alder reaction of 3-(acyloxy)acryloyl oxazolidinones: optically active synthesis of a high-affinity ligand for potent HIV-1 protease inhibitors

RSC Advances ◽  
2019 ◽  
Vol 9 (71) ◽  
pp. 41755-41763
Author(s):  
Arun K. Ghosh ◽  
Alessandro Grillo ◽  
Satish Kovela ◽  
Margherita Brindisi
Keyword(s):  
Protease Inhibitors ◽  
Alder Reaction ◽  
Optically Active ◽  
Diels Alder ◽  
Active Synthesis ◽  
High Affinity ◽  
Affinity Ligand ◽  
Diels Alder Reaction ◽  
High Affinity Ligand ◽  
Hiv 1

Asymmetric Diels–Alder reaction of chiral 3-(acyloxy)acryloyl oxazolidinones and synthesis of hexahydro-4H-3,5-methanofuro[2,3-b]pyranol are described.

ChemInform Abstract: Synthesis and Pharmacokinetics of Potent Carbamate HIV-1 Protease Inhibitors Containing Novel High Affinity Hydroxyethylamine Isosteres.

ChemInform ◽  
2010 ◽  
Vol 27 (14) ◽  
pp. no-no
Author(s):  
W. J. HORNBACK ◽  
J. E. MUNROE ◽  
T. A. SHEPHERD ◽  
S. D. HATCH ◽  
M. A. MUESING ◽  
...  
Keyword(s):  
Protease Inhibitors ◽  
High Affinity ◽  
Hydroxyethylamine Isosteres ◽  
Hiv 1

ChemInform Abstract: A Short Synthesis of 3(R)-Hydroxy-2(R)-isopropyltetrahydrothiophene: A Precursor to a High-Affinity P2-Ligand of HIV-1 Protease Inhibitors.

ChemInform ◽  
2010 ◽  
Vol 25 (17) ◽  
pp. no-no
Author(s):  
B. M. KIM ◽  
H.-Y. LEE ◽  
P. M. MUNSON ◽  
J. P. GUARE ◽  
C. MCDONOUGH
Keyword(s):  
Protease Inhibitors ◽  
High Affinity ◽  
Short Synthesis ◽  
Hiv 1

Thiophene derivatives as extremely high affinity P3′ ligands for the hydroxyethylpiperazine class of HIV-1 protease inhibitors

1995 ◽  
Vol 5 (2) ◽  
pp. 185-190 ◽  
Author(s):  
B. Moon Kim ◽  
James P. Guare ◽  
Joseph D. Vacca ◽  
Stuart R. Michelson ◽  
Paul L. Darke ◽  
...  
Keyword(s):  
Protease Inhibitors ◽  
High Affinity ◽  
Thiophene Derivatives ◽  
Hiv 1

3-Tetrahydrofuran and pyran urethanes as high-affinity P2-ligands for HIV-1 protease inhibitors

1993 ◽  
Vol 36 (2) ◽  
pp. 292-294 ◽  
Author(s):  
Arun K. Ghosh ◽  
Wayne J. Thompson ◽  
Sean P. McKee ◽  
Tien T. Duong ◽  
Terry A. Lyle ◽  
...  
Keyword(s):  
Protease Inhibitors ◽  
High Affinity ◽  
Hiv 1
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