scholarly journals Design and Synthesis of Potent HIV-1 Protease Inhibitors Incorporating Hexahydrofuropyranol-Derived High Affinity P2Ligands: Structure−Activity Studies and Biological Evaluation

2011 ◽  
Vol 54 (2) ◽  
pp. 622-634 ◽  
Author(s):  
Arun K. Ghosh ◽  
Bruno D. Chapsal ◽  
Abigail Baldridge ◽  
Melinda P. Steffey ◽  
D. Eric Walters ◽  
...  
Keyword(s):  
Protease Inhibitors ◽  
Biological Evaluation ◽  
Design And Synthesis ◽  
High Affinity ◽  
Structure Activity ◽  
Hiv 1

scholarly journals Synthesis and biological evaluation of novel allophenylnorstatine-based HIV-1 protease inhibitors incorporating high affinity P2-ligands

2010 ◽  
Vol 20 (3) ◽  
pp. 1241-1246 ◽  
Author(s):  
Arun K. Ghosh ◽  
Sandra Gemma ◽  
Elena Simoni ◽  
Abigail Baldridge ◽  
D. Eric Walters ◽  
...  
Keyword(s):  
Protease Inhibitors ◽  
Biological Evaluation ◽  
High Affinity ◽  
Synthesis And Biological Evaluation ◽  
Hiv 1

scholarly journals Design, synthesis, X-ray studies, and biological evaluation of novel macrocyclic HIV-1 protease inhibitors involving the P1′-P2′ ligands

2017 ◽  
Vol 27 (21) ◽  
pp. 4925-4931 ◽  
Author(s):  
Arun K. Ghosh ◽  
W. Sean Fyvie ◽  
Margherita Brindisi ◽  
Melinda Steffey ◽  
Johnson Agniswamy ◽  
...  
Keyword(s):  
Protease Inhibitors ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
X Ray ◽  
Hiv 1

scholarly journals Probing Lipophilic Adamantyl Group as the P1-Ligand for HIV-1 Protease Inhibitors: Design, Synthesis, Protein X-ray Structural Studies, and Biological Evaluation

2016 ◽  
Vol 59 (14) ◽  
pp. 6826-6837 ◽  
Author(s):  
Arun K. Ghosh ◽  
Heather L. Osswald ◽  
Kristof Glauninger ◽  
Johnson Agniswamy ◽  
Yuan-Fang Wang ◽  
...  
Keyword(s):  
Protease Inhibitors ◽  
Biological Evaluation ◽  
Structural Studies ◽  
Design Synthesis ◽  
X Ray ◽  
Protein X ◽  
Hiv 1

scholarly journals Structure-based design, synthesis, X-ray studies, and biological evaluation of novel HIV-1 protease inhibitors containing isophthalamide-derived P2-ligands

2015 ◽  
Vol 25 (21) ◽  
pp. 4903-4909 ◽  
Author(s):  
Arun K. Ghosh ◽  
Jun Takayama ◽  
Luke A. Kassekert ◽  
Jean-Rene Ella-Menye ◽  
Sofiya Yashchuk ◽  
...  
Keyword(s):  
Protease Inhibitors ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
X Ray ◽  
Hiv 1
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