Structure–activity relationship of nonsecosteroidal vitamin D receptor modulators

Sachiko Yamada; Makoto Makishima

doi:10.1016/j.tips.2014.04.008

Structure–activity relationship of nonsecosteroidal vitamin D receptor modulators

Trends in Pharmacological Sciences ◽

10.1016/j.tips.2014.04.008 ◽

2014 ◽

Vol 35 (7) ◽

pp. 324-337 ◽

Cited By ~ 28

Author(s):

Sachiko Yamada ◽

Makoto Makishima

Keyword(s):

Vitamin D ◽

Vitamin D Receptor ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Structure Activity ◽

Relationship Of ◽

Receptor Modulators

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Structure–activity relationship of benzodiazepine derivatives as LXXLL peptide mimetics that inhibit the interaction of vitamin D receptor with coactivators

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2012.11.042 ◽

2013 ◽

Vol 21 (4) ◽

pp. 993-1005 ◽

Cited By ~ 17

Author(s):

Yusuke Mita ◽

Kosuke Dodo ◽

Tomomi Noguchi-Yachide ◽

Yuichi Hashimoto ◽

Minoru Ishikawa

Keyword(s):

Vitamin D ◽

Vitamin D Receptor ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Peptide Mimetics ◽

Structure Activity ◽

Benzodiazepine Derivatives ◽

Relationship Of

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Synthesis and structure–activity relationship of p-carborane-based non-secosteroidal vitamin D analogs

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2014.01.015 ◽

2014 ◽

Vol 22 (4) ◽

pp. 1227-1235 ◽

Cited By ~ 12

Author(s):

Shinya Fujii ◽

Atsushi Kano ◽

Chalermkiat Songkram ◽

Hiroyuki Masuno ◽

Yoshiyuki Taoda ◽

...

Keyword(s):

Vitamin D ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Vitamin D Analogs ◽

Structure Activity ◽

Relationship Of

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The Structure–Activity Relationship of a Tetrahydroisoquinoline Class ofN-Methyl-d-Aspartate Receptor Modulators that Potentiates GluN2B-ContainingN-Methyl-d-Aspartate Receptors

Journal of Medicinal Chemistry ◽

10.1021/acs.jmedchem.7b00239 ◽

2017 ◽

Vol 60 (13) ◽

pp. 5556-5585 ◽

Cited By ~ 10

Author(s):

Katie L. Strong ◽

Matthew P. Epplin ◽

John Bacsa ◽

Christopher J. Butch ◽

Pieter B. Burger ◽

...

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

Aspartate Receptor ◽

Structure Activity ◽

Relationship Of ◽

Receptor Modulators

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Three-dimensional Structure-activity Relationship of Vitamin D Based on Computational and Synthetic Chemistries.

Journal of Synthetic Organic Chemistry Japan ◽

10.5059/yukigoseikyokaishi.59.131 ◽

2001 ◽

Vol 59 (2) ◽

pp. 131-141 ◽

Cited By ~ 1

Author(s):

Keiko Yamamoto ◽

Hiroyuki Masuno ◽

Sachiko Yamada

Keyword(s):

Vitamin D ◽

Three Dimensional ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Dimensional Structure ◽

Three Dimensional Structure ◽

Structure Activity ◽

Relationship Of

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ChemInform Abstract: Three-Dimensional Structure-Activity Relationship of Vitamin D Based on Computational and Synthetic Chemistries

ChemInform ◽

10.1002/chin.200131271 ◽

2010 ◽

Vol 32 (31) ◽

pp. no-no

Author(s):

Keiko Yamamoto ◽

Hiroyuki Masuno ◽

Sachiko Yamada

Keyword(s):

Vitamin D ◽

Three Dimensional ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Dimensional Structure ◽

Three Dimensional Structure ◽

Structure Activity ◽

Relationship Of

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Structure–activity relationship studies on vitamin D lactam derivatives as vitamin D receptor antagonist

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2008.06.095 ◽

2008 ◽

Vol 18 (15) ◽

pp. 4287-4290 ◽

Cited By ~ 12

Author(s):

Kaori Cho ◽

Fumito Uneuchi ◽

Yuko Kato-Nakamura ◽

Jun-ichi Namekawa ◽

Seiichi Ishizuka ◽

...

Keyword(s):

Vitamin D ◽

Receptor Antagonist ◽

Vitamin D Receptor ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Structure Activity

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Selective Estrogen Receptor Modulators with Conformationally Restricted Side Chains. Synthesis and Structure−Activity Relationship of ERα-Selective Tetrahydroisoquinoline Ligands

Journal of Medicinal Chemistry ◽

10.1021/jm040858p ◽

2005 ◽

Vol 48 (2) ◽

pp. 364-379 ◽

Cited By ~ 43

Author(s):

Johanne Renaud ◽

Serge François Bischoff ◽

Thomas Buhl ◽

Philipp Floersheim ◽

Brigitte Fournier ◽

...

Keyword(s):

Estrogen Receptor ◽

Selective Estrogen Receptor Modulators ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Side Chains ◽

Conformationally Restricted ◽

Estrogen Receptor Modulators ◽

Structure Activity ◽

Relationship Of ◽

Receptor Modulators

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C19-Steroids as androgen receptor modulators: Design, discovery, and structure-activity relationship of new steroidal androgen receptor antagonists

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2006.05.022 ◽

2006 ◽

Vol 14 (17) ◽

pp. 5933-5947 ◽

Cited By ~ 18

Author(s):

Padma Marwah ◽

Ashok Marwah ◽

Henry A. Lardy ◽

Hiroshi Miyamoto ◽

Chawnshang Chang

Keyword(s):

Androgen Receptor ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Receptor Antagonists ◽

Structure Activity ◽

Relationship Of ◽

Receptor Modulators ◽

Androgen Receptor Antagonists

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Extending the Structure–Activity Relationship of Anthranilic Acid Derivatives As Farnesoid X Receptor Modulators: Development of a Highly Potent Partial Farnesoid X Receptor Agonist

Journal of Medicinal Chemistry ◽

10.1021/jm500937v ◽

2014 ◽

Vol 57 (19) ◽

pp. 8035-8055 ◽

Cited By ~ 33

Author(s):

Daniel Merk ◽

Christina Lamers ◽

Khalil Ahmad ◽

Roberto Carrasco Gomez ◽

Gisbert Schneider ◽

...

Keyword(s):

Anthranilic Acid ◽

Receptor Agonist ◽

Structure Activity Relationship ◽

Farnesoid X Receptor ◽

Activity Relationship ◽

Structure Activity ◽

Relationship Of ◽

Receptor Modulators ◽

Anthranilic Acid Derivatives

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Synthesis and Structure−Activity Relationship of Novel 6-Aryl-1,4- dihydrobenzo[d][1,3]oxazine-2-thiones as Progesterone Receptor Modulators Leading to the Potent and Selective Nonsteroidal Progesterone Receptor Agonist Tanaproget#

Journal of Medicinal Chemistry ◽

10.1021/jm050358b ◽

2005 ◽

Vol 48 (16) ◽

pp. 5092-5095 ◽

Cited By ~ 64

Author(s):

Andrew Fensome ◽

Reinhold Bender ◽

Rajiv Chopra ◽

Jeff Cohen ◽

Mark A. Collins ◽

...

Keyword(s):

Progesterone Receptor ◽

Receptor Agonist ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Structure Activity ◽

Relationship Of ◽

Receptor Modulators ◽

Progesterone Receptor Modulators

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