Synthesis, SAR studies, and pharmacological evaluation of 3-anilino-4-(3-indolyl) maleimides with conformationally restricted structure as orally bioavailable PKCβ-selective inhibitors

2006 ◽  
Vol 14 (17) ◽  
pp. 5781-5794 ◽  
Author(s):  
Masahiro Tanaka ◽  
Shoichi Sagawa ◽  
Jun-ichi Hoshi ◽  
Fumito Shimoma ◽  
Katsutaka Yasue ◽  
...  
Keyword(s):  
Selective Inhibitors ◽  
Conformationally Restricted ◽  
Pharmacological Evaluation ◽  
Sar Studies ◽  
Orally Bioavailable

scholarly journals SAR Studies of 5-Aminopyrazole-4-carboxamide Analogues as Potent and Selective Inhibitors of Toxoplasma gondii CDPK1

2015 ◽  
Vol 6 (12) ◽  
pp. 1184-1189 ◽  
Author(s):  
Wenlin Huang ◽  
Kayode K. Ojo ◽  
Zhongsheng Zhang ◽  
Kasey Rivas ◽  
Rama Subba Rao Vidadala ◽  
...  
Keyword(s):  
Toxoplasma Gondii ◽  
Selective Inhibitors ◽  
Sar Studies

scholarly journals Design, Synthesis, and SAR Studies of 4-Substituted Methoxylbenzoyl-aryl-thiazoles Analogues as Potent and Orally Bioavailable Anticancer Agents

2011 ◽  
Vol 54 (13) ◽  
pp. 4678-4693 ◽  
Author(s):  
Yan Lu ◽  
Chien-Ming Li ◽  
Zhao Wang ◽  
Jianjun Chen ◽  
Michael L. Mohler ◽  
...  
Keyword(s):  
Anticancer Agents ◽  
Design Synthesis ◽  
Sar Studies ◽  
Orally Bioavailable

scholarly journals Discovery of Orally Bioavailable Selective Inhibitors of the Sodium-Phosphate Cotransporter NaPi2a (SLC34A1)

2018 ◽  
Vol 9 (5) ◽  
pp. 440-445 ◽  
Author(s):  
Kevin J. Filipski ◽  
Matthew F. Sammons ◽  
Samit K. Bhattacharya ◽  
Jane Panteleev ◽  
Janice A. Brown ◽  
...  
Keyword(s):  
Sodium Phosphate ◽  
Selective Inhibitors ◽  
Orally Bioavailable
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