Facile synthesis of polymer-peptide conjugates via direct amino acid coupling chemistry

2013 ◽  
Vol 51 (22) ◽  
pp. 4853-4859 ◽  
Author(s):  
Gwen F. Chimonides ◽  
Arun A. Sohdi ◽  
Mohammad R. Khaleghi ◽  
Claire R. Hurley ◽  
Dave J. Adams ◽  
...  
Keyword(s):  
Amino Acid ◽  
Facile Synthesis ◽  
Peptide Conjugates

Facile Synthesis of Highly FunctionalizedN-Methyl Amino Acid Esters without Side-Chain Protection

2005 ◽  
Vol 7 (19) ◽  
pp. 4111-4112 ◽  
Author(s):  
Kimberly N. White ◽  
Joseph P. Konopelski
Keyword(s):  
Amino Acid ◽  
Side Chain ◽  
Amino Acid Esters ◽  
Facile Synthesis ◽  
Acid Esters

scholarly journals Corrigendum concerning “Methoxinine—An alternative stable amino acid substitute for oxidation‐sensitive methionine in radiolabelled peptide conjugates”

2020 ◽  
Vol 26 (3) ◽  
Author(s):  
Nathalie M. Grob ◽  
Martin Behe ◽  
Elisabeth Guggenberg ◽  
Roger Schibli ◽  
Thomas L. Mindt
Keyword(s):  
Amino Acid ◽  
Peptide Conjugates ◽  
Radiolabelled Peptide

Facile Synthesis of a “Ready to Use” Precursor of Porphobilinogen and Its Amino Acid Derivatives

2008 ◽  
Vol 73 (2) ◽  
pp. 764-767 ◽  
Author(s):  
Carole Pissot Soldermann ◽  
Ramakrishnan Vallinayagam ◽  
Manuel Tzouros ◽  
Reinhard Neier
Keyword(s):  
Amino Acid ◽  
Amino Acid Derivatives ◽  
Facile Synthesis

Facile Synthesis of Lipophilic δ-Amino Acid Conjugates from 4-Alkoxy-dithionaphthoic Acids

2012 ◽  
Vol 42 (18) ◽  
pp. 2694-2706 ◽  
Author(s):  
Anna C. Worth ◽  
Catherine E. Needham ◽  
Donald B. Franklin ◽  
Andrew J. Lampkins
Keyword(s):  
Amino Acid ◽  
Facile Synthesis ◽  
Amino Acid Conjugates

Amino Acid Derivatives in Organic Synthesis, Part 4 [1]: Facile Synthesis of Heterocycles Containing a Glycine Residue

2000 ◽  
Vol 55 (1) ◽  
pp. 104-108 ◽  
Author(s):  
Laila M. Chabaka ◽  
Yehia A. Allam ◽  
Galal A. M. Nawwar
Keyword(s):  
Amino Acid ◽  
Organic Synthesis ◽  
Acid Group ◽  
The Other ◽  
Amino Acid Derivatives ◽  
Carboxylic Acid Group ◽  
Facile Synthesis ◽  
Peptide Linkage ◽  
Active Methylene Compounds ◽  
Active Methylene

Pyridines, thiazolopyridines and pyrazolopyrans containing glycinate residue were prepared by reacting N-cyanoacryloglycinate ylidenes with active methylene compounds via a Michael addition - intracyclization synthetic pathway.Simple routes for the synthesis of heterocycles with an amino acid residue were previously reported [1-3] as the incorportation of these residues improves the pharmacokinetics and toxicity of active compounds [4,5]. However, trials to deesterify these residues for coupling purposes were unsuccessful. So, we tried herein new approaches for synthesizing heterocyles carrying one or two glycine moieties with free carboxylic acid group to facilitate further peptide linkage [6] on one hand and on the other one could be able to form metal chelates, a property having a significant output on the toxicological behaviour [7]

scholarly journals Methoxinine - an alternative stable amino acid substitute for oxidation-sensitive methionine in radiolabelled peptide conjugates

2017 ◽  
Vol 23 (1) ◽  
pp. 38-44 ◽  
Author(s):  
Nathalie M. Grob ◽  
Martin Behe ◽  
Elisabeth von Guggenberg ◽  
Roger Schibli ◽  
Thomas L. Mindt
Keyword(s):  
Amino Acid ◽  
Peptide Conjugates ◽  
Radiolabelled Peptide
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