The First Total Synthesis of Solomonsterol B, a Marine Pregnane X Receptor Agonist

2012 ◽  
Vol 2012 (27) ◽  
pp. 5187-5194 ◽  
Author(s):  
Valentina Sepe ◽  
Raffaella Ummarino ◽  
Maria Valeria D'Auria ◽  
Barbara Renga ◽  
Stefano Fiorucci ◽  
...  
Keyword(s):  
Total Synthesis ◽  
Receptor Agonist ◽  
Pregnane X Receptor

Total Synthesis and Pharmacological Characterization of Solomonsterol A, a Potent Marine Pregnane-X-Receptor Agonist Endowed with Anti-Inflammatory Activity

2011 ◽  
Vol 54 (13) ◽  
pp. 4590-4599 ◽  
Author(s):  
Valentina Sepe ◽  
Raffaella Ummarino ◽  
Maria Valeria D’Auria ◽  
Andrea Mencarelli ◽  
Claudio D’Amore ◽  
...  
Keyword(s):  
Total Synthesis ◽  
Receptor Agonist ◽  
Pregnane X Receptor ◽  
Inflammatory Activity ◽  
Pharmacological Characterization ◽  
Anti Inflammatory

An efficient total synthesis of a sphingosine-1-phosphate receptor agonist KRP-203

Tetrahedron ◽  
2008 ◽  
Vol 64 (17) ◽  
pp. 3859-3866 ◽  
Author(s):  
Masao Chino ◽  
Masatoshi Kiuchi ◽  
Kunitomo Adachi
Keyword(s):  
Total Synthesis ◽  
Receptor Agonist ◽  
Sphingosine 1 Phosphate

scholarly journals Solomonsterol A, a Marine Pregnane-X-Receptor Agonist, Attenuates Inflammation and Immune Dysfunction in a Mouse Model of Arthritis

Marine Drugs ◽  
2013 ◽  
Vol 12 (1) ◽  
pp. 36-53 ◽  
Author(s):  
Andrea Mencarelli ◽  
Claudio D'Amore ◽  
Barbara Renga ◽  
Sabrina Cipriani ◽  
Adriana Carino ◽  
...  
Keyword(s):  
Mouse Model ◽  
Receptor Agonist ◽  
Pregnane X Receptor ◽  
Immune Dysfunction

Modification in the side chain of solomonsterol A: discovery of cholestan disulfate as a potent pregnane-X-receptor agonist

2012 ◽  
Vol 10 (31) ◽  
pp. 6350 ◽  
Author(s):  
Valentina Sepe ◽  
Raffaella Ummarino ◽  
Maria Valeria D'Auria ◽  
Gianluigi Lauro ◽  
Giuseppe Bifulco ◽  
...  
Keyword(s):  
Receptor Agonist ◽  
Pregnane X Receptor ◽  
Side Chain

scholarly journals Total Synthesis of a Cyclic Adenosine 5′-Diphosphate Ribose Receptor Agonist

2012 ◽  
Vol 77 (9) ◽  
pp. 4191-4197 ◽  
Author(s):  
Joanna M. Swarbrick ◽  
Barry V. L. Potter
Keyword(s):  
Total Synthesis ◽  
Receptor Agonist

Pregnane X Receptor agonist Increases the Expression Levels of the Plasma Membrane Monoamine Transporter

2014 ◽  
Vol 22 (1) ◽  
pp. 19
Author(s):  
Sung Kweon Cho ◽  
Haejin Oh ◽  
Se Hyang Hong ◽  
Min Soo Park ◽  
Jae Yong Chung
Keyword(s):  
Plasma Membrane ◽  
Receptor Agonist ◽  
Pregnane X Receptor ◽  
Monoamine Transporter ◽  
Expression Levels

A Pregnane X Receptor Agonist with Unique Species-Dependent Stereoselectivity and Its Implications in Drug Development

2005 ◽  
Vol 68 (2) ◽  
pp. 403-413 ◽  
Author(s):  
Ying Mu ◽  
Corey R. J. Stephenson ◽  
Christopher Kendall ◽  
Simrat P. S. Saini ◽  
David Toma ◽  
...  
Keyword(s):  
Drug Development ◽  
Receptor Agonist ◽  
Pregnane X Receptor ◽  
Unique Species

scholarly journals Total Synthesis of (±)-Quinagolide: A Potent D2 Receptor Agonist for the Treatment of Hyperprolactinemia

ACS Omega ◽  
2019 ◽  
Vol 4 (5) ◽  
pp. 8231-8238 ◽  
Author(s):  
Subhash P. Chavan ◽  
Appasaheb L. Kadam ◽  
Sanket A. Kawale
Keyword(s):  
Total Synthesis ◽  
Receptor Agonist ◽  
D2 Receptor ◽  
D2 Receptor Agonist
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