Total Synthesis of (±)-Quinagolide: A Potent D2 Receptor Agonist for the Treatment of Hyperprolactinemia

Subhash P. Chavan; Appasaheb L. Kadam; Sanket A. Kawale

doi:10.1021/acsomega.9b00903

Total Synthesis of (±)-Quinagolide: A Potent D2 Receptor Agonist for the Treatment of Hyperprolactinemia

ACS Omega ◽

10.1021/acsomega.9b00903 ◽

2019 ◽

Vol 4 (5) ◽

pp. 8231-8238 ◽

Cited By ~ 3

Author(s):

Subhash P. Chavan ◽

Appasaheb L. Kadam ◽

Sanket A. Kawale

Keyword(s):

Total Synthesis ◽

Receptor Agonist ◽

D2 Receptor ◽

D2 Receptor Agonist

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Synthesis of 3-Azidopiperidine Skeleton Employing Ceric Ammonium Nitrate (CAN)-Mediated Regioselective Azidoalkoxylation of Enol Ether: Total Synthesis of D2 Receptor Agonist (±)-Quinagolide

Organic Letters ◽

10.1021/acs.orglett.8b02900 ◽

2018 ◽

Vol 20 (22) ◽

pp. 7011-7014 ◽

Cited By ~ 5

Author(s):

Subhash P. Chavan ◽

Appasaheb L. Kadam ◽

Pradeep B. Lasonkar ◽

Rajesh G. Gonnade

Keyword(s):

Total Synthesis ◽

Ammonium Nitrate ◽

Receptor Agonist ◽

D2 Receptor ◽

Ceric Ammonium Nitrate ◽

Enol Ether ◽

D2 Receptor Agonist

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Dopamine D2 receptor agonist treatment, Berlin heart excor implantation and transplantation in 7 patients with terminal heart failure caused by Postpartum Cardiomyopathy (PPCM)

The Thoracic and Cardiovascular Surgeon ◽

10.1055/s-0030-1269067 ◽

2011 ◽

Vol 59 (S 01) ◽

Author(s):

S Eifert ◽

R Sodian ◽

E Scherbaum ◽

P Wellmann ◽

S Güthoff ◽

...

Keyword(s):

Heart Failure ◽

Receptor Agonist ◽

Dopamine D2 Receptor ◽

D2 Receptor ◽

Dopamine D2 ◽

Berlin Heart ◽

Terminal Heart Failure ◽

Postpartum Cardiomyopathy ◽

D2 Receptor Agonist

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Neuroprotective effects of dopamine D2 receptor agonist on neuroinflammatory injury in olfactory bulb neurons in vitro and in vivo in a mouse model of allergic rhinitis

NeuroToxicology ◽

10.1016/j.neuro.2021.10.001 ◽

2021 ◽

Author(s):

Peiqiang Liu ◽

Danxue Qin ◽

Hao Lv ◽

Wenjun Fan ◽

Zezhang Tao ◽

...

Keyword(s):

Allergic Rhinitis ◽

Mouse Model ◽

Olfactory Bulb ◽

Receptor Agonist ◽

Dopamine D2 Receptor ◽

D2 Receptor ◽

Neuroprotective Effects ◽

D2 Receptor Agonist

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Quinelorane, a dopamine D3/D2 receptor agonist, reduces prepulse inhibition of startle and ventral pallidal GABA efflux: Time course studies

Pharmacology Biochemistry and Behavior ◽

10.1016/j.pbb.2008.05.012 ◽

2008 ◽

Vol 90 (4) ◽

pp. 686-690 ◽

Cited By ~ 6

Author(s):

Y QU ◽

N SWERDLOW ◽

M WEBER ◽

D STOUFFER ◽

L PARSONS

Keyword(s):

Prepulse Inhibition ◽

Receptor Agonist ◽

Time Course ◽

D2 Receptor ◽

Dopamine D3 ◽

Efflux Time ◽

D2 Receptor Agonist

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In vivo vulnerability to competition by endogenous dopamine: Comparison of the D2 receptor agonist radiotracer (-)-N-[11C]propyl-norapomorphine ([11C]NPA) with the D2 receptor antagonist radiotracer [11C]-raclopride

Synapse ◽

10.1002/syn.20013 ◽

2004 ◽

Vol 52 (3) ◽

pp. 188-208 ◽

Cited By ~ 111

Author(s):

Rajesh Narendran ◽

Dah-Ren Hwang ◽

Mark Slifstein ◽

Peter S. Talbot ◽

David Erritzoe ◽

...

Keyword(s):

Receptor Antagonist ◽

Receptor Agonist ◽

D2 Receptor ◽

Endogenous Dopamine ◽

D2 Receptor Agonist

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The effect of the dopamine D2 receptor agonist cabergoline on the content of catecholamines and expression of BDNF mRNA in the rat midbrain and hypothalamus

Zhurnal nevrologii i psikhiatrii im S S Korsakova ◽

10.17116/jnevro201911911154 ◽

2019 ◽

Vol 119 (11) ◽

pp. 54

Author(s):

P. K. Anokhin ◽

A. G. Veretinskaya ◽

V. V. Pavshintsev ◽

I. Yu. Shamakina

Keyword(s):

Receptor Agonist ◽

Dopamine D2 Receptor ◽

D2 Receptor ◽

Bdnf Mrna ◽

Dopamine D2 ◽

D2 Receptor Agonist

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THE PUTATIVE DOPAMINE D3 RECEPTOR ANTAGONIST PNU 99194A POTENTIATES THE DISCRIMINATIVE STIMULUS INDUCED BYTHE DOPAMINE D3/D2 RECEPTOR AGONIST 7-OH-DPAT

Behavioural Pharmacology ◽

10.1097/00008877-199808000-00052 ◽

1998 ◽

Vol 9 (1) ◽

pp. S31

Author(s):

R. Depoortere ◽

G. h. Perrault ◽

D. J. Sanger

Keyword(s):

Receptor Antagonist ◽

Discriminative Stimulus ◽

Receptor Agonist ◽

D2 Receptor ◽

Dopamine D3 Receptor ◽

D3 Receptor ◽

Dopamine D3 ◽

D2 Receptor Agonist

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Discriminative stimulus properties of S32504, a novel D3/D2 receptor agonist and antiparkinson agent, in rats: attenuation by the antipsychotics, aripiprazole, bifeprunox, N-desmethylclozapine, and by selective antagonists at dopamine D2 but not D3 receptors

Psychopharmacology ◽

10.1007/s00213-006-0567-0 ◽

2006 ◽

Vol 191 (3) ◽

pp. 767-782 ◽

Cited By ~ 12

Author(s):

Mark J. Millan ◽

Loretta Iob ◽

Jean-Louis Péglion ◽

Anne Dekeyne

Keyword(s):

Discriminative Stimulus ◽

Receptor Agonist ◽

D2 Receptor ◽

Stimulus Properties ◽

D3 Receptors ◽

Dopamine D2 ◽

Selective Antagonists ◽

Discriminative Stimulus Properties ◽

D2 Receptor Agonist

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Age-dependent dystonia in striatal Gγ7 deficient mice is reversed by the dopamine D2 receptor agonist pramipexole

Journal of Neurochemistry ◽

10.1111/jnc.12149 ◽

2013 ◽

Vol 124 (6) ◽

pp. 844-854 ◽

Cited By ~ 7

Author(s):

Keita Sasaki ◽

Tatsuro Yamasaki ◽

Idowu O. Omotuyi ◽

Masayoshi Mishina ◽

Hiroshi Ueda

Keyword(s):

Receptor Agonist ◽

Dopamine D2 Receptor ◽

D2 Receptor ◽

Dopamine D2 ◽

Age Dependent ◽

D2 Receptor Agonist ◽

Deficient Mice

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Biochemical and pharmacological studies on pramipexole, a potent and selective dopamine D2 receptor agonist

European Journal of Pharmacology ◽

10.1016/0014-2999(92)90024-x ◽

1992 ◽

Vol 215 (2-3) ◽

pp. 161-170 ◽

Cited By ~ 94

Author(s):

Joachim Mierau ◽

Günter Schingnitz

Keyword(s):

Receptor Agonist ◽

Dopamine D2 Receptor ◽

D2 Receptor ◽

Dopamine D2 ◽

Pharmacological Studies ◽

D2 Receptor Agonist ◽

Selective Dopamine

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