Molecularly Targeted Approach to Cancer Therapy: Design, Synthesis and Biological Activity of Non-Hydroxamate Histone Deacetylase Inhibitors

ChemInform ◽  
2006 ◽  
Vol 37 (12) ◽  
Author(s):  
Takayoshi Suzuki ◽  
Hidehiko Nakagawa ◽  
Naoki Miyata
Keyword(s):  
Biological Activity ◽  
Cancer Therapy ◽  
Histone Deacetylase ◽  
Histone Deacetylase Inhibitors ◽  
Design Synthesis ◽  
Therapy Design ◽  
Targeted Approach

Design, Synthesis, and Biological Activity of Boronic Acid-Based Histone Deacetylase Inhibitors

2009 ◽  
Vol 52 (9) ◽  
pp. 2909-2922 ◽  
Author(s):  
Nobuaki Suzuki ◽  
Takayoshi Suzuki ◽  
Yosuke Ota ◽  
Tatsuya Nakano ◽  
Masaaki Kurihara ◽  
...  
Keyword(s):  
Biological Activity ◽  
Histone Deacetylase ◽  
Boronic Acid ◽  
Histone Deacetylase Inhibitors ◽  
Design Synthesis

Design, Synthesis, and Biological Activity of Hydroxamic Tertiary Amines as Histone Deacetylase Inhibitors

ChemMedChem ◽  
2012 ◽  
Vol 7 (4) ◽  
pp. 694-702 ◽  
Author(s):  
Stefania Terracciano ◽  
Maria Giovanna Chini ◽  
Raffaele Riccio ◽  
Ines Bruno ◽  
Giuseppe Bifulco
Keyword(s):  
Biological Activity ◽  
Histone Deacetylase ◽  
Histone Deacetylase Inhibitors ◽  
Tertiary Amines ◽  
Design Synthesis

Design, synthesis, and biological activity of folate receptor-targeted prodrugs of thiolate histone deacetylase inhibitors

2007 ◽  
Vol 17 (15) ◽  
pp. 4208-4212 ◽  
Author(s):  
Takayoshi Suzuki ◽  
Shinya Hisakawa ◽  
Yukihiro Itoh ◽  
Nobuaki Suzuki ◽  
Katsumasa Takahashi ◽  
...  
Keyword(s):  
Biological Activity ◽  
Histone Deacetylase ◽  
Histone Deacetylase Inhibitors ◽  
Folate Receptor ◽  
Design Synthesis

Design, synthesis and in vitro evaluation of amidoximes as histone deacetylase inhibitors for cancer therapy

2016 ◽  
Vol 26 (19) ◽  
pp. 4679-4683 ◽  
Author(s):  
Peifu Jiao ◽  
Peng Jin ◽  
Chencan Li ◽  
Lechao Cui ◽  
Lihua Dong ◽  
...  
Keyword(s):  
Cancer Therapy ◽  
Histone Deacetylase ◽  
Histone Deacetylase Inhibitors ◽  
Design Synthesis ◽  
In Vitro Evaluation

scholarly journals Design, Synthesis, and Blood–Brain Barrier Transport Study of Pyrilamine Derivatives as Histone Deacetylase Inhibitors

2018 ◽  
Vol 9 (9) ◽  
pp. 884-888 ◽  
Author(s):  
Seiya Hiranaka ◽  
Yuma Tega ◽  
Kei Higuchi ◽  
Toshiki Kurosawa ◽  
Yoshiharu Deguchi ◽  
...  
Keyword(s):  
Histone Deacetylase ◽  
Blood Brain Barrier ◽  
Histone Deacetylase Inhibitors ◽  
Brain Barrier ◽  
Design Synthesis ◽  
Transport Study ◽  
Blood Brain

scholarly journals Novel 4-Oxoquinazoline-Based N-Hydroxypropenamides as Histone Deacetylase Inhibitors: Design, Synthesis, and Biological Evaluation

ACS Omega ◽  
2021 ◽  
Vol 6 (7) ◽  
pp. 4907-4920
Author(s):  
Duong T. Anh ◽  
Pham-The Hai ◽  
Le D. Huy ◽  
Hoang B. Ngoc ◽  
Trinh T. M. Ngoc ◽  
...  
Keyword(s):  
Histone Deacetylase ◽  
Histone Deacetylase Inhibitors ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
Synthesis And Biological Evaluation
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