Antagonists of Human CCR5 Receptor Containing 4-(Pyrazolyl)piperidine Side Chains. Part 1. Discovery and SAR Study of 4-Pyrazolylpiperidine Side Chains.

ChemInform ◽  
2004 ◽  
Vol 35 (25) ◽  
Author(s):  
Dong-Ming Shen ◽  
et al. et al.
Keyword(s):  
Side Chains ◽  
Ccr5 Receptor ◽  
Sar Study ◽  
Human Ccr5

Antagonists of human CCR5 receptor containing 4-(pyrazolyl)piperidine side chains. Part 1: Discovery and SAR study of 4-pyrazolylpiperidine side chains

2004 ◽  
Vol 14 (4) ◽  
pp. 935-939 ◽  
Author(s):  
Dong-Ming Shen ◽  
Min Shu ◽  
Sander G. Mills ◽  
Kevin T. Chapman ◽  
Lorraine Malkowitz ◽  
...  
Keyword(s):  
Side Chains ◽  
Ccr5 Receptor ◽  
Sar Study ◽  
Human Ccr5

Antagonists of human CCR5 receptor containing 4-(pyrazolyl)piperidine side chains. Part 3: SAR studies on the benzylpyrazole segment

2004 ◽  
Vol 14 (4) ◽  
pp. 947-952 ◽  
Author(s):  
Min Shu ◽  
Jennifer L Loebach ◽  
Kerry A Parker ◽  
Sander G Mills ◽  
Kevin T Chapman ◽  
...  
Keyword(s):  
Side Chains ◽  
Sar Studies ◽  
Ccr5 Receptor ◽  
Human Ccr5

Antagonists of human CCR5 receptor containing 4-(pyrazolyl)piperidine side chains. Part 2: Discovery of potent, selective, and orally bioavailable compounds

2004 ◽  
Vol 14 (4) ◽  
pp. 941-945 ◽  
Author(s):  
Dong-Ming Shen ◽  
Min Shu ◽  
Christopher A. Willoughby ◽  
Shrenik Shah ◽  
Christopher L. Lynch ◽  
...  
Keyword(s):  
Side Chains ◽  
Ccr5 Receptor ◽  
Orally Bioavailable ◽  
Human Ccr5

Modulators of the human CCR5 receptor. Part 2: SAR of substituted 1-(3,3-diphenylpropyl)-piperidinyl phenylacetamides

2005 ◽  
Vol 15 (22) ◽  
pp. 5012-5015 ◽  
Author(s):  
John G. Cumming ◽  
Anne E. Cooper ◽  
Ken Grime ◽  
Chris J. Logan ◽  
Sharon McLaughlin ◽  
...  
Keyword(s):  
Ccr5 Receptor ◽  
Substituted 1 ◽  
Human Ccr5
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