ChemInform Abstract: Synthesis and Biological Evaluation of Phospholane and Dihydrophosphole Analogues of the Glutamate Receptor Agonist AP4.

Stuart J. Conway; Jacqueline C. Miller; Andrew D. Bond; Barry P. Clark; David E. Jane

doi:10.1002/chin.200247162

ChemInform Abstract: Synthesis and Biological Evaluation of Phospholane and Dihydrophosphole Analogues of the Glutamate Receptor Agonist AP4.

ChemInform ◽

10.1002/chin.200247162 ◽

2010 ◽

Vol 33 (47) ◽

pp. no-no

Author(s):

Stuart J. Conway ◽

Jacqueline C. Miller ◽

Andrew D. Bond ◽

Barry P. Clark ◽

David E. Jane

Keyword(s):

Glutamate Receptor ◽

Receptor Agonist ◽

Biological Evaluation ◽

Glutamate Receptor Agonist ◽

Synthesis And Biological Evaluation

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Synthesis and biological evaluation of phospholane and dihydrophosphole analogues of the glutamate receptor agonist AP4Electronic supplementry information (ESI) available: mode of epoxide ring-opening and experimental data for 2 and 3. See http://www.rsc.org/suppdata/p1/b2/b204891d/

Journal of the Chemical Society Perkin Transactions 1 ◽

10.1039/b204891d ◽

2002 ◽

pp. 1625-1627 ◽

Cited By ~ 4

Author(s):

Stuart J. Conway ◽

Jacqueline C. Miller ◽

Andrew D. Bond ◽

Barry P. Clark ◽

David E. Jane

Keyword(s):

Experimental Data ◽

Glutamate Receptor ◽

Ring Opening ◽

Receptor Agonist ◽

Biological Evaluation ◽

Epoxide Ring ◽

Epoxide Ring Opening ◽

Glutamate Receptor Agonist ◽

Synthesis And Biological Evaluation

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EFFECTS OF GROUP III METABOTROPIC GLUTAMATE RECEPTOR AGONIST ON THE MICTURITION REFLEX IN URETHANE-ANESTHETIZED RATS

10.26226/morressier.59b63e3fd462b8029238916e ◽

2017 ◽

Author(s):

Masashi Honda

Keyword(s):

Glutamate Receptor ◽

Receptor Agonist ◽

Metabotropic Glutamate Receptor ◽

Group Iii ◽

Micturition Reflex ◽

Metabotropic Glutamate ◽

Anesthetized Rats ◽

Glutamate Receptor Agonist

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Anti-epileptogenic and anticonvulsant activity of l-2-amino-4-phosphonobutyrate, a presynaptic glutamate receptor agonist

Brain Research ◽

10.1016/s0006-8993(97)00098-x ◽

1997 ◽

Vol 755 (2) ◽

pp. 202-212 ◽

Cited By ~ 54

Author(s):

Abdul-Salam Abdul-Ghani ◽

Philip J.E Attwell ◽

Natasha Singh Kent ◽

Henry F Bradford ◽

Martin J Croucher ◽

...

Keyword(s):

Glutamate Receptor ◽

Anticonvulsant Activity ◽

Receptor Agonist ◽

Glutamate Receptor Agonist

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Enzymatic resolution and pharmacological activity of the enantiomers of 3,5-dihydroxyphenylglycine, a metabotropic glutamate receptor agonist

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/0960-894x(95)00013-j ◽

1995 ◽

Vol 5 (3) ◽

pp. 223-228 ◽

Cited By ~ 30

Author(s):

S. Richard Baker ◽

John Goldsworthy ◽

Raymond C. Harden ◽

Craig R. Salhoff ◽

Darryle D. Schoepp

Keyword(s):

Glutamate Receptor ◽

Pharmacological Activity ◽

Receptor Agonist ◽

Metabotropic Glutamate Receptor ◽

Enzymatic Resolution ◽

Metabotropic Glutamate ◽

Glutamate Receptor Agonist

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Protective effect of the metabotropic glutamate receptor agonist, DCG-IV, against excitotoxic neuronal death

European Journal of Pharmacology ◽

10.1016/0014-2999(94)90624-6 ◽

1994 ◽

Vol 256 (1) ◽

pp. 109-112 ◽

Cited By ~ 90

Author(s):

Valeria Bruno ◽

Agata Copani ◽

Giuseppe Battaglia ◽

Rocco Raffaele ◽

Huruiko Shinozaki ◽

...

Keyword(s):

Protective Effect ◽

Glutamate Receptor ◽

Neuronal Death ◽

Receptor Agonist ◽

Metabotropic Glutamate Receptor ◽

Metabotropic Glutamate ◽

Excitotoxic Neuronal Death ◽

Glutamate Receptor Agonist

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Large-scale expression and thermodynamic characterization of a glutamate receptor agonist-binding domain

European Journal of Biochemistry ◽

10.1046/j.1432-1033.2000.01481.x ◽

2000 ◽

Vol 267 (13) ◽

pp. 4281-4289 ◽

Cited By ~ 21

Author(s):

Dean R. Madden ◽

Rupert Abele ◽

Arnold Andersson ◽

Kari Keinänen

Keyword(s):

Glutamate Receptor ◽

Receptor Agonist ◽

Large Scale ◽

Binding Domain ◽

Agonist Binding ◽

Thermodynamic Characterization ◽

Glutamate Receptor Agonist

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LY379268, a potent and selective Group II metabotropic glutamate receptor agonist, is neuroprotective in gerbil global, but not focal, cerebral ischaemia

Neuroscience Letters ◽

10.1016/s0304-3940(99)00663-1 ◽

1999 ◽

Vol 273 (3) ◽

pp. 191-194 ◽

Cited By ~ 51

Author(s):

Ann Bond ◽

Nella Ragumoorthy ◽

James A. Monn ◽

Caroline A. Hicks ◽

Mark A. Ward ◽

...

Keyword(s):

Glutamate Receptor ◽

Cerebral Ischaemia ◽

Receptor Agonist ◽

Metabotropic Glutamate Receptor ◽

Focal Cerebral Ischaemia ◽

Metabotropic Glutamate ◽

Group Ii ◽

Glutamate Receptor Agonist

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The group II metabotropic glutamate receptor agonist LY354740 and the D2 receptor antagonist haloperidol reduce locomotor hyperactivity but fail to rescue spatial working memory in GluA1 knockout mice

European Journal of Neuroscience ◽

10.1111/ejn.13539 ◽

2017 ◽

Vol 45 (7) ◽

pp. 912-921 ◽

Cited By ~ 5

Author(s):

Thomas Boerner ◽

Alexei M. Bygrave ◽

Jingkai Chen ◽

Anushka Fernando ◽

Stephanie Jackson ◽

...

Keyword(s):

Working Memory ◽

Receptor Antagonist ◽

Glutamate Receptor ◽

Knockout Mice ◽

Receptor Agonist ◽

Metabotropic Glutamate Receptor ◽

Spatial Working Memory ◽

D2 Receptor ◽

Metabotropic Glutamate ◽

Glutamate Receptor Agonist

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Expression of the Neural Recognition Molecule L1 by Cultured Neural Cells is influenced by K+and the Glutamate Receptor Agonist NMDA

European Journal of Neuroscience ◽

10.1111/j.1460-9568.1992.tb00905.x ◽

1992 ◽

Vol 4 (6) ◽

pp. 554-562 ◽

Cited By ~ 15

Author(s):

Martin Scherer ◽

Martin Heller ◽

Melitta Schachner

Keyword(s):

Glutamate Receptor ◽

Receptor Agonist ◽

Neural Cells ◽

Glutamate Receptor Agonist ◽

Recognition Molecule

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Potentiation of excitatory postsynaptic potentials by a metabotropic glutamate receptor agonist (1S,3R-ACPD) in frog spinal motoneurons

Brain Research ◽

10.1016/0006-8993(95)00580-j ◽

1995 ◽

Vol 689 (2) ◽

pp. 281-288 ◽

Cited By ~ 11

Author(s):

Hiroyuki Gotani ◽

Miyuki Kuno ◽

Fusao Nakamura ◽

Shiushi Matsuura

Keyword(s):

Glutamate Receptor ◽

Receptor Agonist ◽

Metabotropic Glutamate Receptor ◽

Excitatory Postsynaptic Potentials ◽

Spinal Motoneurons ◽

Postsynaptic Potentials ◽

Metabotropic Glutamate ◽

Glutamate Receptor Agonist

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