ChemInform Abstract: Synthesis and Structure-Activity Relationships in a Series of Ethenesulfonamide Derivatives, a Novel Class of Endothelin Receptor Antagonists.

Hironori Harada; Jun-ichi Kazami; Susumu Watanuki; Ryuji Tsuzuki; Katsumi Sudoh; Akira Fujimori; Tatsuhiro Tokunaga; Akihiro Tanaka; Shin-ichi Tsukamoto; Isao Yanagisawa

doi:10.1002/chin.200217147

ChemInform Abstract: Synthesis and Structure-Activity Relationships in a Series of Ethenesulfonamide Derivatives, a Novel Class of Endothelin Receptor Antagonists.

ChemInform ◽

10.1002/chin.200217147 ◽

2010 ◽

Vol 33 (17) ◽

pp. no-no

Author(s):

Hironori Harada ◽

Jun-ichi Kazami ◽

Susumu Watanuki ◽

Ryuji Tsuzuki ◽

Katsumi Sudoh ◽

...

Keyword(s):

Endothelin Receptor Antagonists ◽

Endothelin Receptor ◽

Receptor Antagonists ◽

Structure Activity Relationships ◽

Structure Activity

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Synthesis and Structure−Activity Relationships of 2-Substitutedd-Tryptophan-Containing Peptidic Endothelin Receptor Antagonists: Importance of the C-2 Substituent of thed-Tryptophan Residue for Endothelin A and B Receptor Subtype Selectivity

Journal of Medicinal Chemistry ◽

10.1021/jm9600914 ◽

1996 ◽

Vol 39 (12) ◽

pp. 2313-2330 ◽

Cited By ~ 14

Author(s):

Takehiro Fukami ◽

Takeru Yamakawa ◽

Kenji Niiyama ◽

Hisaki Kojima ◽

Yuuka Amano ◽

...

Keyword(s):

Tryptophan Residue ◽

Receptor Subtype ◽

Endothelin Receptor Antagonists ◽

Endothelin Receptor ◽

Receptor Antagonists ◽

Structure Activity Relationships ◽

Subtype Selectivity ◽

Structure Activity ◽

Endothelin A

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Structure–Activity relationships of 2-substituted 5,7-Diarylcyclopenteno[1,2-b]pyridine-6-carboxylic acids as a novel class of endothelin receptor antagonists

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/s0960-894x(02)00663-7 ◽

2002 ◽

Vol 12 (21) ◽

pp. 3041-3045 ◽

Cited By ~ 7

Author(s):

Kenji Niiyama ◽

Hirobumi Takahashi ◽

Toshio Nagase ◽

Hisaki Kojima ◽

Yuka Amano ◽

...

Keyword(s):

Carboxylic Acids ◽

Endothelin Receptor Antagonists ◽

Endothelin Receptor ◽

Receptor Antagonists ◽

Structure Activity Relationships ◽

Structure Activity

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Synthesis and Structure-Activity Relationships in a Series of Ethenesulfonamide Derivatives, a Novel Class of Endothelin Receptor Antagonists.

Chemical and Pharmaceutical Bulletin ◽

10.1248/cpb.49.1593 ◽

2001 ◽

Vol 49 (12) ◽

pp. 1593-1603 ◽

Cited By ~ 7

Author(s):

Hironori HARADA ◽

Jun-ichi KAZAMI ◽

Susumu WATANUKI ◽

Ryuji TSUZUKI ◽

Katsumi SUDOH ◽

...

Keyword(s):

Endothelin Receptor Antagonists ◽

Endothelin Receptor ◽

Receptor Antagonists ◽

Structure Activity Relationships ◽

Structure Activity

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Structure—Activity Relationships of 2-Substituted 5,7-Diarylcyclopenteno[1,2-b]pyridine-6-carboxylic Acids as a Novel Class of Endothelin Receptor Antagonists.

ChemInform ◽

10.1002/chin.200309133 ◽

2003 ◽

Vol 34 (9) ◽

Author(s):

Kenji Niiyama ◽

et al. et al.

Keyword(s):

Carboxylic Acids ◽

Endothelin Receptor Antagonists ◽

Endothelin Receptor ◽

Receptor Antagonists ◽

Structure Activity Relationships ◽

Structure Activity

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Endothelin receptor antagonists: synthesis and structure–activity relationships of substituted benzothiazine-1,1-dioxides

Bioorganic & Medicinal Chemistry ◽

10.1016/s0968-0896(98)00080-7 ◽

1998 ◽

Vol 6 (9) ◽

pp. 1447-1456 ◽

Cited By ~ 10

Author(s):

K.A. Berryman ◽

J.J. Edmunds ◽

A.M. Bunker ◽

S. Haleen ◽

J. Bryant ◽

...

Keyword(s):

Endothelin Receptor Antagonists ◽

Endothelin Receptor ◽

Receptor Antagonists ◽

Structure Activity Relationships ◽

Structure Activity

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Biphenylsulfonamide Endothelin Receptor Antagonists. Part 3: Structure–Activity Relationship of 4′-Heterocyclic Biphenylsulfonamides

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/s0960-894x(01)00791-0 ◽

2002 ◽

Vol 12 (4) ◽

pp. 517-520 ◽

Cited By ~ 4

Author(s):

Natesan Murugesan ◽

Zhengxiang Gu ◽

Philip D. Stein ◽

Steven Spergel ◽

Sharon Bisaha ◽

...

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

Endothelin Receptor Antagonists ◽

Endothelin Receptor ◽

Receptor Antagonists ◽

Structure Activity ◽

Relationship Of

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Endothelin Receptor Antagonists: An Overview of Their Synthesis and Structure-Activity Relationship

Mini-Reviews in Medicinal Chemistry ◽

10.2174/1389557053544010 ◽

2005 ◽

Vol 5 (4) ◽

pp. 381-408 ◽

Cited By ~ 12

Author(s):

Javed Iqbal ◽

Rashmi Sanghi ◽

Saibal Das

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

Endothelin Receptor Antagonists ◽

Endothelin Receptor ◽

Receptor Antagonists ◽

Structure Activity

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ChemInform Abstract: Biphenylsulfonamide Endothelin Receptor Antagonists. Part 3. Structure-Activity Relationship of 4′-Heterocyclic Biphenylsulfonamides.

ChemInform ◽

10.1002/chin.200221114 ◽

2010 ◽

Vol 33 (21) ◽

pp. no-no

Author(s):

Natesan Murugesan ◽

Zhengxiang Gu ◽

Philip D. Stein ◽

Steven Spergel ◽

Sharon Bisaha ◽

...

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

Endothelin Receptor Antagonists ◽

Endothelin Receptor ◽

Receptor Antagonists ◽

Structure Activity ◽

Relationship Of

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Faculty Opinions recommendation of Race and sex differences in response to endothelin receptor antagonists for pulmonary arterial hypertension.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.13489110.15114060 ◽

2012 ◽

Author(s):

Robert Frantz ◽

Vivek Iyer

Keyword(s):

Sex Differences ◽

Pulmonary Arterial Hypertension ◽

Arterial Hypertension ◽

Endothelin Receptor Antagonists ◽

Endothelin Receptor ◽

Receptor Antagonists ◽

Pulmonary Arterial

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ChemInform Abstract: Endothelin Receptor Antagonist Triterpenoid, Myriceric Acid A, Isolated from Myrica cerifera, and Structure Activity Relationships of Its Derivatives.

ChemInform ◽

10.1002/chin.199633208 ◽

2010 ◽

Vol 27 (33) ◽

pp. no-no

Author(s):

K. SAKURAWI ◽

F. YASUDA ◽

T. TOZYO ◽

M. NAKAMURA ◽

T. SATO ◽

...

Keyword(s):

Receptor Antagonist ◽

Endothelin Receptor Antagonist ◽

Endothelin Receptor ◽

Myrica Cerifera ◽

Structure Activity Relationships ◽

Structure Activity ◽

Myriceric Acid A

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