ChemInform Abstract: Carbonic Anhydrase Inhibitors. Part 53. Synthesis of Substituted-Pyridinium Derivatives of Aromatic Sulfonamides: The First Non-Polymeric Membrane-Impermeable Inhibitors with Selectivity for Isozyme IV.

C. T. SUPURAN; A. SCOZZAFAVA; M. A. ILIES; B. IORGA; T. CRISTEA; F. BRIGANTI; F. CHIRALEU; M. D. BANCIU

doi:10.1002/chin.199852168

ChemInform Abstract: Carbonic Anhydrase Inhibitors. Part 53. Synthesis of Substituted-Pyridinium Derivatives of Aromatic Sulfonamides: The First Non-Polymeric Membrane-Impermeable Inhibitors with Selectivity for Isozyme IV.

ChemInform ◽

10.1002/chin.199852168 ◽

2010 ◽

Vol 29 (52) ◽

pp. no-no

Author(s):

C. T. SUPURAN ◽

A. SCOZZAFAVA ◽

M. A. ILIES ◽

B. IORGA ◽

T. CRISTEA ◽

...

Keyword(s):

Carbonic Anhydrase ◽

Polymeric Membrane ◽

Carbonic Anhydrase Inhibitors ◽

Derivatives Of

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Carbonic anhydrase inhibitors — Part 53. Synthesis of substituted-pyridinium derivatives of aromatic sulfonamides: The first non-polymeric membrane-impermeable inhibitors with selectivity for isozyme IV

European Journal of Medicinal Chemistry ◽

10.1016/s0223-5234(98)80017-2 ◽

1998 ◽

Vol 33 (7-8) ◽

pp. 577-594 ◽

Cited By ~ 56

Author(s):

Claudiu T. Supuran ◽

Andrea Scozzafava ◽

Marc A. Ilies ◽

Bogdan Iorga ◽

Teodora Cristea ◽

...

Keyword(s):

Carbonic Anhydrase ◽

Polymeric Membrane ◽

Carbonic Anhydrase Inhibitors ◽

Derivatives Of

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Bioorganometallic derivatives of 4-hydrazino-benzenesulphonamide as carbonic anhydrase inhibitors: synthesis, characterisation and biological evaluation

Journal of Enzyme Inhibition and Medicinal Chemistry ◽

10.1080/14756366.2020.1724995 ◽

2020 ◽

Vol 35 (1) ◽

pp. 622-628 ◽

Cited By ~ 2

Author(s):

Jeremie Brichet ◽

Rodrigo Arancibia ◽

Emanuela Berrino ◽

Claudiu T. Supuran

Keyword(s):

Carbonic Anhydrase ◽

Biological Evaluation ◽

Carbonic Anhydrase Inhibitors ◽

Derivatives Of

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ChemInform Abstract: Carbonic Anhydrase Inhibitors. Part 2. Membrane-Impermeable Derivatives of 1,3,4-Thiadiazole-2-sulfonamide.

ChemInform ◽

10.1002/chin.199144178 ◽

2010 ◽

Vol 22 (44) ◽

pp. no-no

Author(s):

C. SUPURAN ◽

A. T. BALABAN ◽

M. D. GHEORGHIU ◽

A. SCHICKETANZ ◽

A. DINCULESCU ◽

...

Keyword(s):

Carbonic Anhydrase ◽

Carbonic Anhydrase Inhibitors ◽

Derivatives Of

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Carbonic anhydrase inhibitors. Synthesis of 2,4,6-trimethylpyridinium derivatives of 2-(hydrazinocarbonyl)-3-aryl-1H-indole-5-sulfonamides acting as potent inhibitors of the tumor-associated isoform IX and XII

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2009.04.068 ◽

2009 ◽

Vol 19 (11) ◽

pp. 2931-2934 ◽

Cited By ~ 11

Author(s):

Özlen Güzel ◽

Alfonso Maresca ◽

Andrea Scozzafava ◽

Aydın Salman ◽

Alexandru T. Balaban ◽

...

Keyword(s):

Carbonic Anhydrase ◽

Carbonic Anhydrase Inhibitors ◽

Derivatives Of

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QSAR Studies on Carbonic Anhydrase Inhibitors: A Case of Ureido and Thioureido Derivatives of Aromatic/Heterocyclic Sulfonamides

Bioorganic & Medicinal Chemistry ◽

10.1016/s0968-0896(02)00123-2 ◽

2002 ◽

Vol 10 (9) ◽

pp. 2993-2999 ◽

Cited By ~ 19

Author(s):

Vijay K. Agrawal ◽

Ruchi Sharma ◽

Padmakar V. Khadikar

Keyword(s):

Carbonic Anhydrase ◽

Carbonic Anhydrase Inhibitors ◽

Qsar Studies ◽

Derivatives Of ◽

Aromatic Heterocyclic

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ChemInform Abstract: Carbonic Anhydrase Inhibitors. Part 49. Synthesis of Substituted Ureido and Thioureido Derivatives of Aromatic/Heterocyclic Sulfonamides with Increased Affinities for Isozyme I.

ChemInform ◽

10.1002/chin.199829111 ◽

2010 ◽

Vol 29 (29) ◽

pp. no-no

Author(s):

C. T. SUPURAN ◽

A. SCOZZAFAVA ◽

B. C. JURCA ◽

M. A. ILIES

Keyword(s):

Carbonic Anhydrase ◽

Carbonic Anhydrase Inhibitors ◽

Derivatives Of ◽

Aromatic Heterocyclic

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Carbonic Anhydrase Inhibitors: Ureido and Thioureido Derivatives of Aromatic Sulfonamides Possessing Increased Affinities for Isozyme I. A Novel Route To 2,5-Disubstituted-L,3,4-Thiadiazoles Via Thioureas, and Their Interaction with Isozymes I, II and IV

Journal of Enzyme Inhibition ◽

10.3109/14756369809035830 ◽

1998 ◽

Vol 13 (2) ◽

pp. 103-123 ◽

Cited By ~ 24

Author(s):

Andrea Scozzafava ◽

Claudiu T. Supuran

Keyword(s):

Carbonic Anhydrase ◽

Carbonic Anhydrase Inhibitors ◽

Derivatives Of

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Bile acid derivatives of 5-amino-1,3,4-thiadiazole-2-sulfonamide as new carbonic anhydrase inhibitors: synthesis and investigation of inhibition effects

Bioorganic & Medicinal Chemistry ◽

10.1016/s0968-0896(02)00104-9 ◽

2002 ◽

Vol 10 (8) ◽

pp. 2561-2567 ◽

Cited By ~ 23

Author(s):

Metin Bülbül ◽

Nurullah Saraçoğlu ◽

Ö. İrfan Küfrevioğlu ◽

Mehmet Çiftçi

Keyword(s):

Bile Acid ◽

Carbonic Anhydrase ◽

Carbonic Anhydrase Inhibitors ◽

Bile Acid Derivatives ◽

Derivatives Of

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Topically active carbonic anhydrase inhibitors. 1. O-Acyl derivatives of 6-hydroxybenzothiazole-2-sulfonamide

Journal of Medicinal Chemistry ◽

10.1021/jm00131a011 ◽

1989 ◽

Vol 32 (11) ◽

pp. 2486-2492 ◽

Cited By ~ 33

Author(s):

O. W. Woltersdorf ◽

H. Schwam ◽

J. B. Bicking ◽

S. L. Brown ◽

S. J. DeSolms ◽

...

Keyword(s):

Carbonic Anhydrase ◽

Carbonic Anhydrase Inhibitors ◽

Derivatives Of ◽

Acyl Derivatives ◽

Active Carbonic Anhydrase

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Carbonic anhydrase inhibitors - Part 49: Synthesis of substituted ureido and thioureido derivatives of aromatic/heterocyclic sulfonamides with increased affinities for isozyme I

European Journal of Medicinal Chemistry ◽

10.1016/s0223-5234(98)80033-0 ◽

1998 ◽

Vol 33 (2) ◽

pp. 83-93 ◽

Cited By ~ 113

Author(s):

Claudiu T. Supuran ◽

Andrea Scozzafava ◽

Bogdan C. Jurca ◽

Marc A. Ilies

Keyword(s):

Carbonic Anhydrase ◽

Carbonic Anhydrase Inhibitors ◽

Derivatives Of ◽

Aromatic Heterocyclic

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